RecruitingPhase 1Phase 2NCT06500676

A Study of GFH375 in Patients With Advanced Solid Tumors With KRAS G12D Mutations

An Open-Label, Phase I/II Clinical Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Efficacy of GFH375 in Patients With KRAS G12D Mutant Advanced Solid Tumors


Sponsor

Genfleet Therapeutics (Shanghai) Inc.

Enrollment

407 participants

Start Date

Jul 9, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

This is a multicenter, open-label, phase I/II study to explore the safety, tolerability, pharmacokinetics (PK), and preliminary efficacy of GFH375 in patients with advanced solid tumors harboring a KRAS G12D mutation.


Eligibility

Min Age: 18 YearsMax Age: 75 Years

Inclusion Criteria7

  • Subjects must voluntarily agree to participate in the trial and sign a written informed consent form.
  • Male or female ≥ 18 years old and ≤75 years old.
  • ECOG performance status of 0-1.
  • With a life expectancy of ≥12 weeks.
  • With histologically or cytologically confirmed advanced or metastatic solid tumors harboring KRAS G12D mutation.
  • Have at least one measurable lesion according to RECIST1.1, and the phase Ia allows no measurable lesion.
  • Adequate laboratory parameters during the screening period.

Exclusion Criteria7

  • Active brain metastases.
  • Prior treatment with a KRAS G12D inhibitor.
  • Palliative radiotherapy was completed within 14 days before the first dose.
  • Have poorly controlled or severe cardiovascular disease.
  • Subjects with active hepatitis B or active hepatitis C.
  • Known allergy to the study drug or its components.
  • Pregnant or lactating women.

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Interventions

DRUGGFH375

GFH375 will be administered at the assigned dose level, orally, until disease progression or intolerable toxicity.


Locations(20)

The First Affiliated Hospital of Anhui Medical University

Hefei, Anhui, China

Cancer Hospital, Chinese Academy of Medical Sciences

Beijing, Beijing Municipality, China

Peking Union Medical College Hospital

Beijing, Beijing Municipality, China

Sun Yat-sen Memorial Hospital, Sun Yat-sen University

Guangzhou, Guangdong, China

The Sixth Affiliated Hospital of Sun Yat-sen University

Guangzhou, Guangdong, China

Guangxi Medical University Cancer Hospital

Nanning, Guangxi, China

Harbin Medical University Cancer Hospital

Haerbin, Heilongjiang, China

The First Affiliated Hospital of Zhengzhou University

Zhengzhou, Henan, China

Union Hospital Tongji Medical College Huazhong University of Science and Technology

Wuhan, Hubei, China

Hunan Cancer Hospital

Changsha, Hunan, China

Jiangsu Province Hospital

Nanjing, Jiangsu, China

Liaoning Cancer Hospital & Institute

Shenyang, Liaoning, China

The First Affiliated Hospital of China Medical University

Shenyang, Liaoning, China

Shandong Cancer Hospital

Jinan, Shandong, China

Shanghai Chest Hospital

Shanhai, Shanghai Municipality, China

Sichuan Cancer Hospital

Chengdu, Sichuan, China

Tianjin Medical University Cancer Institute & Hospital

Tianjing, Tianjing, China

The First Affiliated Hospital Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

The Second Affiliated Hospital Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

View Full Details on ClinicalTrials.gov

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NCT06500676


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