RecruitingPhase 2NCT06593522

A Phase 2 Study of AMG 193 in Participants With MTAP-deleted Advanced NSCLC (MTAPESTRY 201)

A Phase 2 Study Evaluating the Efficacy, Safety, Tolerability, and Pharmacokinetics of AMG 193 in Subjects With Methylthioadenosine Phosphorylase (MTAP)-Deleted Previously Treated Advanced Non-Small Cell Lung Cancer (NSCLC)


Sponsor

Amgen

Enrollment

200 participants

Start Date

Dec 26, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

The main objective of the study is to characterize safety and efficacy of 2 dose levels of AMG 193 by investigator, and to evaluate AMG 193 monotherapy efficacy by Blinded Independent Central Review (BICR).


Eligibility

Min Age: 18 YearsMax Age: 99 Years

Inclusion Criteria6

  • Histologically or cytologically confirmed metastatic or unresectable locally advanced MTAP-deleted (Homozygous deletion of MTAP) NSCLC
  • Participants will have received and progressed or experienced disease recurrence on or after receiving at least 1 prior systemic therapy for locally advanced and unresectable or metastatic disease.
  • Either an archival tissue sample or an archival block must be available.
  • Life expectancy of greater than 3 months, in the opinion of the investigator.
  • Participants who have had brain metastases and have been appropriately treated with radiation therapy or surgery ending at least 14 days before study day 1 are eligible.
  • Participants with untreated asymptomatic brain metastases smaller or equal to 2 cm in size (per lesion if more than one) and not requiring corticosteroid treatment are eligible.

Exclusion Criteria5

  • Disease Related
  • • Tumors harboring the following mutations amenable to targeted therapies: epidermal growth factor receptor (EGFR), ALK receptor tyrosine kinase (ALK), ROS proto-oncogene 1 (ROS1), neurotrophic tyrosine receptor kinase (NTRK), MET proto-oncogene (MET), B-Raf proto-oncogene (BRAF), RET proto-oncogene (RET), Human epidermal growth factor receptor 2 (HER2/ERBB2), KRAS proto-oncogene G12C (KRAS G12C).
  • Other Medical Conditions
  • Major surgery within 28 days of study day 1.
  • Untreated symptomatic central nervous system (CNS) metastatic disease regardless of size or asymptomatic brain metastases greater than 2 cm per lesion.

Interventions

DRUGAMG 193

Film-coated tablet


Locations(91)

Cancer Research South Australia

Adelaide, South Australia, Australia

Núcleo de Oncologia da Bahia

Salvador, Estado de Bahia, Brazil

City of Hope National Medical Center

Duarte, California, United States

City of Hope Orange County Lennar Foundation Cancer Center

Duarte, California, United States

Cedars-Sinai Medical Center

Los Angeles, California, United States

Valkyrie Clinical Trials

Los Angeles, California, United States

University of California Los Angeles

Los Angeles, California, United States

Rocky Mountain Cancer Centers

Denver, Colorado, United States

Eastern Connecticut Hematology and Oncology Associates

Norwich, Connecticut, United States

Hartford HealthCare Cancer Institute - Manchester

Plainville, Connecticut, United States

Medstar Georgetown University Hospital

Washington D.C., District of Columbia, United States

Our Lady of the Lake Cancer Institute

Baton Rouge, Louisiana, United States

Trinity Health Saint Joseph Mercy Ann Arbor

Ann Arbor, Michigan, United States

Cancer and Hematology Centers of Western Michigan

Grand Rapids, Michigan, United States

Sarah Cannon Research Institute Oncology Partners

Nashville, Tennessee, United States

United States Oncology Regulatory Affairs Corporate Office

Nashville, Tennessee, United States

Texas Oncology Central/South Texas

Austin, Texas, United States

Sarah Cannon Research Institute

Dallas, Texas, United States

Texas Oncology - Dallas Fort Worth

Dallas, Texas, United States

US Oncology Research Investigational Products Center

Irving, Texas, United States

Texas Oncology Northeast Texas

Tyler, Texas, United States

Virginia Cancer Specialists PC

Fairfax, Virginia, United States

GenesisCare -North Shore Oncology

St Leonards, New South Wales, Australia

Calvary Mater Newcastle Hospital

Waratah, New South Wales, Australia

Mater Hospital Brisbane

South Brisbane, Queensland, Australia

Liga Norte-Riograndense Contra O Cancer

Natal, Rio Grande do Norte, Brazil

Hospital Sao Lucas da Pontificia Universidade Catolica do Rio Grande do Sul

Porto Alegre, Rio Grande do Sul, Brazil

Hospital Nossa Senhora da Conceicao

Porto Alegre, Rio Grande do Sul, Brazil

Fundacao pio xII Barretos

Barretos, São Paulo, Brazil

Fund Faculdade Regional Med Sao Jose Rio Preto

São José do Rio Preto, São Paulo, Brazil

Instituto do Cancer Estado SP Icesp

São Paulo, São Paulo, Brazil

Fundacao Antonio Prudente - Hosp AC Camargo

São Paulo, São Paulo, Brazil

Instituto de Educacao Pesquisa e Gestao em Saude

Rio de Janeiro, Brazil

Centro Paulista de Oncologia

São Paulo, Brazil

Cross Cancer Institute

Edmonton, Alberta, Canada

William Osler Health System - Brampton Civic Hospital

Brampton, Ontario, Canada

London Health Sciences Centre

London, Ontario, Canada

Princess Margaret Cancer Centre

Toronto, Ontario, Canada

McGill University Health Centre Glen Site

Montreal, Quebec, Canada

Beijing Cancer Hospital

Beijing, Beijing Municipality, China

Mengchao Hepatobiliary Hospital of Fujian Medical University

Fuzhou, Fujian, China

Henan Cancer Hospital

Zhengzhou, Henan, China

The First Affiliated Hospital of Zhengzhou University

Zhengzhou, Henan, China

Union Hospital Tongji Medical College Huazhong University of Science and Technology

Wuhan, Hubei, China

The Second Xiangya Hospital of Central South University

Changsha, Hunan, China

Jilin Cancer Hospital

Changchun, Jilin, China

Jinan Central Hospital

Jinan, Shandong, China

Shanghai East Hospital

Shanghai, Shanghai Municipality, China

West China Hospital Sichuan University

Chengdu, Sichuan, China

The First Affiliated Hospital Zhejiang University School Of Medicine

Hangzhou, Zhejiang, China

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

Beijing Cancer Hospital

Beijing, China

Beijing Chest Hospital, Capital Medical University

Beijing, China

Masarykuv onkologicky ustav

Brno, Czechia

Fakultni nemocnice Olomouc

Olomouc, Czechia

Vseobecna fakultni nemocnice v Praze

Prague, Czechia

Fakultni Thomayerova nemocnice

Prague, Czechia

Queen Mary Hospital, The University of Hong Kong

Hong Kong, Hong Kong

Prince of Wales Hospital, Chinese University of Hong Kong

Shatin, New Territories, Hong Kong

Aichi Cancer Center

Nagoya, Aichi-ken, Japan

National Cancer Center Hospital East

Kashiwa-shi, Chiba, Japan

Shizuoka Cancer Center

Sunto-gun, Shizuoka, Japan

National Cancer Center Hospital

Chuo-ku, Tokyo, Japan

The Cancer Institute Hospital of Japanese Foundation for Cancer Research

Koto-ku, Tokyo, Japan

Wakayama Medical University Hospital

Wakayama, Wakayama, Japan

Pauls Stradins Clinical University Hospital

Riga, Latvia

Riga East Clinical University Hospital

Riga, Latvia

Nederlands Kanker Instituut Antoni van Leeuwenhoekziekenhuis

Amsterdam, Netherlands

Sint Jansdal Ziekenhuis

Harderwijk, Netherlands

Erasmus Medisch Centrum

Rotterdam, Netherlands

Unidade Local de Saude de Braga, EPE

Braga, Portugal

Fundacao Champalimaud

Lisbon, Portugal

Hospital Cuf porto

Porto, Portugal

Instituto Portugues de Oncologia do Porto Francisco Gentil, EPE

Porto, Portugal

National University Hospital

Singapore, Singapore

National Cancer Centre Singapore

Singapore, Singapore

Cha Bundang Medical Center, Cha University

Seongnam-si, Gyeonggi-do, South Korea

Severance Hospital Yonsei University Health System

Seoul, South Korea

Ajou University Hospital

Suwon-si Gyeonggi-do, South Korea

The Catholic University of Korea St Vincents Hospital

Suwon-si, Gyeonggi-do, South Korea

Universitaetsspital Basel

Basel, Switzerland

Hopitaux Universitaires de Geneve

Geneva, Switzerland

Kantonsspital Sankt Gallen

Sankt Gallen, Switzerland

Taichung Veterans General Hospital

Taichung, Taiwan

National Cheng Kung University Hospital

Tainan, Taiwan

National Taiwan University Hospital

Taipei, Taiwan

Adana Sehir Egitim ve Arastirma Hastanesi

Adana, Turkey (Türkiye)

Gazi Universitesi Saglik Arastirma ve Uygulama Merkezi Gazi Hastanesi

Ankara, Turkey (Türkiye)

Ankara Bilkent Sehir Hastanesi

Ankara, Turkey (Türkiye)

Memorial Bahcelievler Hastanesi

Istanbul, Turkey (Türkiye)

Bagcilar Medipol Mega Universite Hastanesi

Istanbul, Turkey (Türkiye)

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NCT06593522