RecruitingPhase 1NCT05231785

A Study to Evaluate the Safety and Tolerability of ALN-APP in Patients With EOAD

A Randomized, Double-blind, Placebo-controlled Single Ascending Dose and Open-label Multi-dose Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Intrathecally Administered ALN-APP in Adult Patients With Early-onset Alzheimer's Disease (EOAD)


Sponsor

Alnylam Pharmaceuticals

Enrollment

60 participants

Start Date

Feb 4, 2022

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to evaluate the safety, tolerability, pharmacodynamics (PD) and pharmacokinetics (PK) of a single dose and multiple doses of ALN-APP administered by intrathecal (IT) injection in adult patients with early-onset Alzheimer's Disease (EOAD). Maximum treatment duration for Part A: single dose. Maximum treatment duration for Part B: 12 months.


Eligibility

Min Age: 18 Years

Inclusion Criteria2

  • Has mild cognitive impairment or mild dementia due to EOAD
  • Has Clinical Dementia Rating (CDR) global score 0.5 or 1.0 and Mini Mental State Examination (MMSE) \>20

Exclusion Criteria5

  • Has Non-Alzheimer's disease dementia
  • Has alanine aminotransferase (ALT) or aspartate aminotransferase (AST) \>2×upper limit of normal (ULN)
  • Has estimated glomerular filtration rate (eGFR) \<45 mL/min/1.73m\^2 at Screening
  • Has recently received an investigational agent
  • Has recent treatment with amyloid-targeting antibody

Interventions

DRUGALN-APP

ALN-APP will be administered intrathecally (IT)

DRUGPlacebo

Placebo will be administered IT


Locations(8)

Clinical Trial Site

La Jolla, California, United States

Clinical Trial Site

Indianapolis, Indiana, United States

Clinical Trial Site

Montreal, Canada

Clinical Trial Site

Toronto, Canada

Clinical Trial Site

Amsterdam, Netherlands

Clinical Trial Site

Groningen, Netherlands

Clinical Trial Site

Huntley Street, United Kingdom

Clinical Trial Site

Sheffield, United Kingdom

View Full Details on ClinicalTrials.gov

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NCT05231785


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