RecruitingPhase 1Phase 2NCT05490472

JAB-2485 Activity in Adult Patients With Advanced Solid Tumors

A Phase 1/2a, Multi-Center, Open-Label Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Preliminary Evidence of Antitumor Activity of JAB-2485 in Adult Patients With Advanced Solid Tumors


Sponsor

Jacobio Pharmaceuticals Co., Ltd.

Enrollment

102 participants

Start Date

Dec 20, 2022

Study Type

INTERVENTIONAL

Conditions

Summary

This study is to evaluate the safety and tolerability of JAB-2485 monotherapy in adult participants with advanced solid tumors.


Eligibility

Min Age: 18 Years

Inclusion Criteria8

  • Must have Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • Must be able to provide an archived tumor sample
  • Must have histologically or cytologically confirmed metastatic or locally advanced solid tumor
  • Dose Expansion phase cohorts must meet specific expression or gene mutation where indicated
  • Must be refractory to or become intolerant of existing therapy(ies) known to provide clinical benefit for their condition
  • Must have at least 1 measurable lesion per RECIST v1.1
  • Must have adequate organ functions
  • Must be able to swallow and retain orally administered medication

Exclusion Criteria8

  • Has central nervous system (CNS) metastases or carcinomatous meningitis, except if CNS metastases treated and no evidence of radiographic progression or hemorrhage for at least 28 days
  • Active infection requiring systemic treatment within 7 days
  • Active hepatitis B virus (HBV), hepatitis C virus (HCV), or HIV
  • Any severe and/or uncontrolled medical conditions
  • left ventricular ejection fraction (LVEF) ≤50% assessed by echocardiogram (ECHO) or multigated acquisition scan (MUGA)
  • QT interval using Fridericia's formula (QTcF) interval \>470 msec
  • Experiencing unresolved CTCAE 5.0 Grade \>1 toxicities
  • Clinically significant eye disorders

Interventions

DRUGJAB-2485 (Aurora A inhibitor)

Administered orally

DRUGJAB-2485 (Aurora A inhibitor)

Administered orally


Locations(8)

Henry Ford Health System

Detroit, Michigan, United States

Washington University

St Louis, Missouri, United States

Mary Crowley Cancer Research

Dallas, Texas, United States

University of Utah Huntsman Cancer Institute

Salt Lake City, Utah, United States

Cancer Hospital Chinese Academy of Medical Sciences

Beijing, Beijing Municipality, China

Peking University Third Hospital

Beijing, Beijing Municipality, China

Jilin Cancer Hospital

Changchun, Jilin, China

Shandong Cancer Hospital

Jinan, Shandong, China

View Full Details on ClinicalTrials.gov

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NCT05490472


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