RecruitingPhase 1NCT05954312

A First-in-Human (FIH) Study to Evaluate the Safety and Tolerability of VVD-130037 in Participants With Advanced Solid Tumors

A Phase 1, Open-label, Multicenter, First-in-Human Study to Evaluate the Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Preliminary Anti-tumor Activity of VVD-130037, a Kelch-like ECH Associated Protein 1 (KEAP1) Activator, in Participants With Advanced Solid Tumors


Sponsor

Vividion Therapeutics, Inc.

Enrollment

290 participants

Start Date

Jul 28, 2023

Study Type

INTERVENTIONAL

Conditions

Summary

A FIH dose escalation and dose expansion study to evaluate VVD-130037 in participants with advanced solid tumors as a single agent, and in combination with docetaxel, paclitaxel, or pembrolizumab.


Eligibility

Min Age: 18 Years

Plain Language Summary

Simplified for easier understanding

This early-phase study is testing a new experimental cancer drug called VVD-130037 in people with advanced solid tumors that have not responded to standard treatments. This is the first time this drug is being tested in humans, so the study focuses primarily on safety and finding the right dose. **You may be eligible if...** - You have confirmed advanced or metastatic solid tumor that has progressed on all prior standard treatments - You have at least one measurable tumor on imaging - Your overall health is adequate (ECOG ≤1) with good organ function - For certain cohorts: You may need to have squamous cell lung cancer, head and neck cancer, or esophageal squamous cell cancer with specific prior treatments **You may NOT be eligible if...** - You have specific genetic mutations (KEAP1 nonsense or frameshift mutations) that are expected to prevent benefit from this drug - You are on anti-epileptic medications or have a history of seizures - Your cancer has spread to the brain or spinal cord - You have had a recent heart attack, congestive heart failure, or serious irregular heartbeat in the past 6 months - You have unresolved significant toxicity from prior cancer treatment Talk to your doctor to see if this trial is right for you.

This summary was AI-generated to explain the trial in plain language. It is not medical advice. Always discuss eligibility with your doctor before enrolling in a clinical trial.

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Interventions

DRUGVVD-130037

Oral tablets

DRUGDocetaxel

IV infusion

DRUGPaclitaxel

IV infusion

DRUGPembrolizumab

IV infusion


Locations(26)

Mayo Clinic Jacksonville

Jacksonville, Florida, United States

Florida Cancer Specialists

Sarasota, Florida, United States

Moffitt Cancer Center

Tampa, Florida, United States

Mayo Clinic Rochester

Rochester, Minnesota, United States

Sarah Cannon Research Institute

Nashville, Tennessee, United States

MDACC

Houston, Texas, United States

NEXT Dallas

Irving, Texas, United States

NEXT Virginia

Fairfax, Virginia, United States

National Cancer Center

Goyang, South Korea

The Catholic University of Korea, St. Vincent's Hospital

Goyang, South Korea

Gachon University Gil Medical Center

Incheon, South Korea

Seoul National University; Bundang Hospital

Seongnam, South Korea

Asan Medical Center

Seoul, South Korea

Samsung Medical Center

Seoul, South Korea

Seoul National University Hospital

Seoul, South Korea

Severance Hospital; Yonsei University Health System

Seoul, South Korea

The Catholic University of Korea, St. Vincent's Hospital

Suwon, South Korea

Hospital Vall d'Hebron

Barcelona, Spain

START Barcelona Hospital HM Nou Delfos

Barcelona, Spain

Hospital Universitario 12 de Octubre

Madrid, Spain

Hospital Universitario Ramon y Cajal

Madrid, Spain

NEXT Madrid

Madrid, Spain

START Madrid CIOCC

Madrid, Spain

Start Madrid-FJD, Hospital Fundacion Jimenez Diaz

Madrid, Spain

Clinica Universitaria de Navarra

Pamplona, Spain

Hospital Clinico Universitario de Valencia

Valencia, Spain

View Full Details on ClinicalTrials.gov

For the most up-to-date information, visit the official listing.

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NCT05954312


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