RecruitingPhase 1NCT05978492

A Study of TXN10128 in Subjects With Solid Tumors

A Multicenter, Open-label, Phase 1 Dose Escalation and Expansion Study of TXN10128, an Inhibitor of ENPP1 as Monotherapy and Combination Therapy With Irinotecan or Paclitaxel in Locally Advanced or Metastatic Solid Tumors


Sponsor

Txinno Bioscience Inc.

Enrollment

96 participants

Start Date

Jul 27, 2023

Study Type

INTERVENTIONAL

Conditions

Summary

This is a phase I clinical trial to primarily evaluate the safety, tolerability, and addtionally assess pharmacokinetics, pharmacodynamics, and antitumor activity of investigational product, TXN10128. The target subjects will be consisted of patients with locally advanced (unresectable) or metastatic soild tumors. This study includes a dose-escalation part and a dose-expansion part, and a TXN10128 monotherapy part and a TXN10128 + Irinotecan or Paclitaxel combination therapy part.


Eligibility

Min Age: 19 Years

Inclusion Criteria4

  • Male or female subjects ≥19 years of age at the time of informed consent.
  • Histologically and/or cytologically confirmed any progressive, locally advanced (unresectable), or metastatic solid tumors that have relapsed or are refractory following the last line of treatment and for which prior standard therapy has been ineffective, or standard therapy does not exist or is not considered appropriate.
  • ECOG performance status of 0 or 1.
  • Life expectancy of at least 12 weeks.

Exclusion Criteria4

  • Has leptomeningeal disease.
  • Experienced a Grade ≥3 immune-related adverse events (irAE) with prior immunotherapy with the exception of non-clinically significant laboratory abnormalities.
  • Prior organ transplantation.
  • Known positive human immunodeficiency virus (HIV) infection.

Interested in this trial?

Get notified about updates and connect with the research team.

Interventions

DRUGTXN10128

TXN10128: Oral administration once daily everyday

DRUGIrinotecan

Intravenous (IV) administration at 150 mg/m2 twice (Day 1 and Day 15) at intervals of 2 weeks in one cycle

DRUGPaclitaxel

IV administration at 80 mg/m2 three times (Day 1, Day 8, and Day 15) at intervals of 1 week in one cycle (IV administration at 90 mg/m2 for patients with breast cancer)


Locations(6)

Seoul National University Bundang Hospital

Seongnam-si, Gyeonggi-do, South Korea

Chungbuk National University Hospital

Cheonju, North Chungcheong, South Korea

Seoul National Univ. Hospital

Seoul, Seoul, South Korea

Asan Medical Center

Seoul, Seoul, South Korea

Gachon University Gil Medical Center

Incheon, South Korea

SAMSUNG Medical Center

Seoul, South Korea

View Full Details on ClinicalTrials.gov

For the most up-to-date information, visit the official listing.

Visit

NCT05978492


Related Trials