RecruitingPhase 1NCT06179160

A Study to Evaluate INCB161734 in Participants With Advanced or Metastatic Solid Tumors With KRAS G12D Mutation

A Phase 1, Open-Label, Multicenter Study of INCB161734 in Participants With Advanced or Metastatic Solid Tumors With KRAS G12D Mutation


Sponsor

Incyte Corporation

Enrollment

710 participants

Start Date

Jan 4, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

This study is conducted to determine the safety and tolerability of INCB161734 as a single agent or in combination with other anticancer therapies.


Eligibility

Min Age: 18 Years

Inclusion Criteria5

  • ≥18 years old.
  • Locally advanced or metastatic solid tumor with KRAS G12D mutation.
  • For Part 1a and Part 2 Combination Groups 1, 2, and 7: Disease progression on prior standard treatment, intolerance to or ineligibility for standard treatment, declined available therapies that are known to confer clinical benefit, or no standard available treatment to improve the disease outcome.
  • Cohort specific requirements aas defined in the protocol.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.

Exclusion Criteria6

  • Prior treatment with any KRAS G12D inhibitor
  • Known additional invasive malignancy within 1 year of the first dose of study drug
  • History of organ transplant, including allogeneic stem cell transplantation
  • Significant, uncontrolled medical condition
  • History or presence of an ECG abnormality
  • Inadequate organ function

Interventions

DRUGINCB161734

INCB161734 will be administered at protocol defined dose.

DRUGCetuximab

Cetuximab will be administered at protocol defined dose.

DRUGRetifanlimab

Retifanlimab will be administered at protocol defined dose.

DRUGGEMNabP

GEMNabP will be administered at protocol defined dose.

DRUGmFOLFIRINOX

mFOLFIRINOX will be administered at protocol defined dose.

DRUGFOLFOX

FOLFOX will be administered at protocol defined dose.

DRUGFOLFIRI

FOLFIRI will be administered at protocol defined dose.

DRUGINCA33890

INCA33890 will be administered at protocol defined dose.


Locations(34)

Centre Leon Berard

Lyon, France

Mayo Clinic Hospital

Phoenix, Arizona, United States

Stanford University

Palo Alto, California, United States

UCLA Healthcare Hematology-Oncology

Santa Monica, California, United States

Sarah Cannon Research Institue At Healthone

Denver, Colorado, United States

Florida Cancer Specialists

Sarasota, Florida, United States

Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Baltimore, Maryland, United States

Dana Farber Cancer Institute

Boston, Massachusetts, United States

Hackensack University Medical Center

Hackensack, New Jersey, United States

Weill Cornell Medicine

New York, New York, United States

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Jefferson University Hospitals

Philadelphia, Pennsylvania, United States

Scri Oncology Partners

Nashville, Tennessee, United States

Md Anderson Cancer Center

Houston, Texas, United States

Chris Obrien Lifehouse

Camperdown, New South Wales, Australia

St Vincent'S Hospital Sydney

Darlinghurst, New South Wales, Australia

The Alfred Hospital

Melbourne, Victoria, Australia

Peter Maccallum Cancer Centre

North Melbourne, Victoria, Australia

Linear Clinical Research

Nedlands, Western Australia, Australia

Cliniques Universitaires Ucl Saint-Luc

Brussels, Belgium

Universitair Ziekenhuis Antwerpen (Uza)

Edegem, Belgium

Universitair Ziekenhuis (Uz) Leuven

Leuven, Belgium

The Ottawa Hospital Cancer Center

Ottawa, Ontario, Canada

Princess Margaret Cancer Center

Toronto, Ontario, Canada

Universitaire Du Cancer de Toulouse Institut Claudius Regaud Iuct-Oncopole

Toulouse, France

Institut Gustave Roussy

Villejuif, France

Fondazione Irccs Istituto Nazionale Dei Tumori

Milan, Italy

Irccs Istituto Clinico Humanitas

Rozzano, Italy

Centro Ricerche Cliniche Di Verona

Verona, Italy

National Cancer Center Hospital East

Chiba, Japan

The Cancer Institute Hospital of Jfcr

Tokyo, Japan

Hospital General Universitario Vall D Hebron

Barcelona, Spain

Fundacion Jimenez Diaz

Madrid, Spain

Hospital Universitario Quironsalud Madrid

Madrid, Spain

View Full Details on ClinicalTrials.gov

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NCT06179160


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