RecruitingPhase 1NCT06238479

A Study of LY4101174 in Participants With Recurrent, Advanced or Metastatic Solid Tumors

A Phase 1 Trial Investigating LY4101174, an Antibody-Drug Conjugate Targeting Nectin-4, in Participants With Recurrent, Advanced or Metastatic Solid Tumors


Sponsor

Eli Lilly and Company

Enrollment

490 participants

Start Date

Mar 5, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to find out whether the study drug, LY4101174, is safe, tolerable and effective in participants with select advanced or metastatic solid tumors. The study is conducted in two parts - phase Ia (dose-escalation, dose-optimization) and phase Ib (dose-expansion). The study will last up to approximately 4 years.


Eligibility

Min Age: 18 Years

Inclusion Criteria20

  • Have one of the following solid tumor cancers:
  • Cohort A1: urothelial carcinoma, triple negative breast cancer, non-small cell lung cancer, esophageal cancer, pancreatic cancer, ovarian cancer, cervical cancer (squamous cell carcinoma), head and neck squamous cell carcinoma or prostate cancer
  • Cohort A2/B1/B2: urothelial carcinoma
  • Cohort C1: triple negative breast cancer
  • Cohort C2: non-small cell lung cancer
  • Cohort C3: ovarian or fallopian tube cancer
  • Cohort C4: cervical cancer
  • Cohort C5: head and neck squamous cell carcinoma
  • Prior Systemic Therapy Criteria:
  • Cohort A1/C1-5: Individual has received all standard therapies for which the participant was deemed to be an appropriate candidate by the treating investigator; OR there is no standard therapy available for the disease. There is no restriction on number of prior therapies
  • Cohort A2/B1/B2: Individual must have received at least one prior regimen in the advanced or metastatic setting. There is no restriction on number of prior therapies.
  • Prior enfortumab vedotin specific requirements:
  • Cohorts A1/A2/C1-5: prior treatment with enfortumab vedotin is allowed, but not required
  • Cohort B1: individual must be enfortumab vedotin naive in the advanced/metastatic setting
  • Cohort B2: individual must have received enfortumab vedotin in the metastatic/advanced setting.
  • Measurability of disease
  • Cohort A1: measurable or non-measurable disease as defined by Response Evaluation Criteria in Solid Tumors v1.1 (RECIST 1.1)
  • Cohorts A2, B1, B2, C1-5: measurable disease required as defined by RECIST v1.1
  • Have an Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • Have adequate archival tumor tissue sample available or undergo a screening biopsy if allowed per country specific regulations

Exclusion Criteria13

  • Individual with known or suspected uncontrolled CNS metastases
  • Individual with uncontrolled hypercalcemia
  • Individual with uncontrolled diabetes
  • Individual with evidence of corneal keratopathy or history of corneal transplant
  • Any serious unresolved toxicities from prior therapy
  • Significant cardiovascular disease
  • Current of history of intestinal obstruction in the previous 3 months
  • Recent thromboembolic event and/or clinically significant bleeding
  • Prolongation of QT interval corrected for heart rate using Fridericia's formula (QTcF) ≥ 470 ms
  • History of pneumonitis/interstitial lung disease
  • History of Grade ≥3 skin toxicity when receiving enfortumab vedotin
  • Individuals who are pregnant, breastfeeding or plan to breastfeed during study or within 30 days of last dose of study intervention
  • Individual with active uncontrolled infection

Interventions

DRUGLY4101174

Intravenous


Locations(28)

AdventHealth Orlando

Orlando, Florida, United States

Emory University

Atlanta, Georgia, United States

Massachusetts General Hospital

Boston, Massachusetts, United States

Washington University School of Medicine

St Louis, Missouri, United States

Perlmutter Cancer Center at NYU Langone Hospital - Long Island

Mineola, New York, United States

Laura & Isaac Perlmutter Cancer Center at NYU Langone Health

New York, New York, United States

Memorial Sloan Kettering Cancer Center

New York, New York, United States

UT Southwestern Medical Center

Dallas, Texas, United States

South Texas Accelerated Research Therapeutics (START)

San Antonio, Texas, United States

Austin Health

Heidelberg, Australia

Icon Cancer Centre Kurralta Park

Kurralta Park, Australia

Institut Jules Bordet

Anderlecht, Belgium

Peking University First Hospital

Beijing, China

Hunan Cancer Hospital

Changsha, China

Shanghai East Hospital

Shanghai, China

Centre Oscar Lambret

Lille, France

Centre Leon Berard

Lyon, France

Institut Paoli-Calmettes

Marseille, France

CHU Strasbourg-Hautepierre

Strasbourg, France

Gustave Roussy

Villejuif, France

National Cancer Center Hospital

Chūōku, Japan

National Cancer Center Hospital East

Kashiwa, Japan

The Cancer Institute Hospital of JFCR

Kōtō City, Japan

Kyoto University Hospital

Kyoto, Japan

Hospital Universitari Vall d'Hebron

Barcelona, Spain

MD Anderson Cancer Center

Madrid, Spain

Hospital Universitario 12 de Octubre

Madrid, Spain

Hospital Universitario Virgen Del Rocio

Seville, Spain

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NCT06238479


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