RecruitingPhase 1Phase 2NCT06244771

A Study Evaluating FMC-376 in Participants With KRAS G12C Mutated Solid Tumors

An Open-Label, Phase 1/2 Dose Escalation, Dose Expansion and Cohort Expansion Study Evaluating the Safety, PK and Clinical Activity of FMC-376 in Participants With KRAS G12C Mutated Locally Advanced Unresectable or Metastatic Solid Tumors


Sponsor

Frontier Medicines Corporation

Enrollment

403 participants

Start Date

Feb 12, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

The goal of this clinical trial is to evaluate FMC-376 in participants with advanced solid tumors with KRAS G12C mutations. This clinical trial will be conducted in 3 parts: Phase 1A (Dose Escalation), Phase 1B (Dose Expansion), and Phase 2 (Cohort Expansion). Multiple dose levels in participants with advanced solid tumors will be evaluated.


Eligibility

Min Age: 18 Years

Inclusion Criteria5

  • Histologically or cytologically confirmed locally advanced unresectable or metastatic solid tumors with KRAS G12C mutation
  • Received and progressed or been intolerant to prior standard therapy OR standard therapy is considered inappropriate OR an investigational agent is considered standard of care
  • Eastern Cooperative Oncology Group (ECOG) performance status 0 or 1
  • Adequate hematological, renal, and hepatic function
  • Agrees not to participate in another interventional study while receiving study drug

Exclusion Criteria5

  • Leptomeningeal disease or carcinomatous meningitis
  • Clinically significant toxicity resulting from prior cancer therapies
  • Known or suspected hypersensitivity to FMC-376 or any components of the study drug
  • Condition that would interfere with study drug absorption
  • Any illness or medical history that would impact safety or compliance with study requirements or impact ability to interpret study data

Interventions

DRUGFMC-376

Oral Capsule Daily


Locations(26)

University of California San Diego (UC San Diego) Health - Jacobs Medical Center - Moores Cancer Center

La Jolla, California, United States

University of California Irvine (UCI) - Chao Family Comprehensive Cancer Center

Orange, California, United States

University of California San Francisco (UCSF) - Helen Diller Family Comprehensive Cancer Center

San Francisco, California, United States

Florida Cancer Specialists and Research Institute

Lake Mary, Florida, United States

Northwest Cancer Centers

Dyer, Indiana, United States

The University of Kansas Cancer Center

Fairway, Kansas, United States

Dana-Farber Cancer Institute

Boston, Massachusetts, United States

Karmanos Cancer Institute

Detroit, Michigan, United States

University of Pennsylvania

Philadelphia, Pennsylvania, United States

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Community Clinical Trials

Kingwood, Texas, United States

South Texas Accelerated Research Therapeutics, LLC

San Antonio, Texas, United States

UT Health San Antonio

San Antonio, Texas, United States

START Mountain Region

West Valley City, Utah, United States

Virginia Cancer Specialists

Fairfax, Virginia, United States

Macquarie University

Macquarie Park, New South Wales, Australia

Tasman Health Care

Southport, Queensland, Australia

Icon Cancer Centre Kurralta Park

Kurralta Park, South Australia, Australia

GenesisCare North Adelaide

North Adelaide, South Australia, Australia

Eastern Health - Box Hill Hospital

Box Hill, Victoria, Australia

Linear Clinical Research Ltd

Nedlands, Western Australia, Australia

Seoul National University Hospital

Seoul, Jongno-gu, South Korea

Severance Hospital

Seoul, Seodaemun-gu, South Korea

Korea University Anam Hospital

Seoul, Seongbuk-gu, South Korea

Seoul National University Bundang Hospital

Gyeonggi-do, Seongnam-si, South Korea

The Catholic University of Korea, St. Vincent's Hospital

Gyeonggi-do, Suwon-si, South Korea

View Full Details on ClinicalTrials.gov

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NCT06244771


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