RecruitingPhase 1NCT06253871

A Phase 1/1b Study of IAM1363 in HER2 Cancers

A Phase 1/1b Study of IAM1363 in Patients With Advanced Cancers Harboring HER2 Alterations


Sponsor

Iambic Therapeutics, Inc

Enrollment

243 participants

Start Date

Mar 25, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

This is a Phase 1/1b open-label, multi-center dose escalation and dose optimization study designed to evaluate the safety and preliminary efficacy of IAM1363 in participants with advanced cancers that harbor HER2 alterations.


Eligibility

Min Age: 18 Years

Inclusion Criteria7

  • Age ≥ 18 years
  • Have relapsed/refractory HER2-altered malignancy
  • Have progression of disease after the last systemic therapy, or be intolerant of last systemic therapy
  • Have radiographically measurable disease by RECIST v1.1 and/or RANO-BM
  • Eastern Cooperative Oncology Group (ECOG) performance score 0-1
  • Have adequate baseline hematologic, liver and renal function
  • Have left ventricular ejection fraction (LVEF) ≥ 50%

Exclusion Criteria8

  • Clinically significant cardiac disease
  • Infection with human immunodeficiency virus (HIV)-1 or HIV-2. Exception: Patients with well-controlled HIV (e.g., CD4 \>350/mm3 and undetectable viral load) are eligible
  • Current active liver disease including hepatitis A, hepatitis B , or hepatitis C
  • Refractory nausea and vomiting, malabsorption, external biliary shunt, or significant small bowel resection that would preclude adequate absorption
  • Uncontrolled diabetes
  • History of solid organ transplantation
  • History of Grade ≥2 CNS hemorrhage, or any CNS hemorrhage within 28 days before C1D1
  • Patients requiring immediate local therapy for brain metastases

Interventions

DRUGIAM1363

Oral, immediate release capsules of IAM1363


Locations(45)

UCSD Moores Cancer Center

La Jolla, California, United States

USC Norris Comprehensive Cancer Center

Los Angeles, California, United States

University of Colorado Cancer Center

Aurora, Colorado, United States

University of Miami

Miami, Florida, United States

Comprehensive Hematology Oncology

St. Petersburg, Florida, United States

University of Chicago

Chicago, Illinois, United States

Dana Farber Cancer Institute

Boston, Massachusetts, United States

University of Michigan

Ann Arbor, Michigan, United States

Henry Ford Cancer Institute

Detroit, Michigan, United States

START - Midwest Cancer Research Center

Grand Rapids, Michigan, United States

Saint Luke's Cancer Institute

Kansas City, Missouri, United States

Washington University School of Medicine

St Louis, Missouri, United States

RUTGERS Cancer Institute

New Brunswick, New Jersey, United States

Icahn School of Medicine at Mount Sinai

New York, New York, United States

Duke Cancer Institute

Durham, North Carolina, United States

University Hospital Cleveland Medical Center

Cleveland, Ohio, United States

Cleveland Clinic

Cleveland, Ohio, United States

OU Health Stephenson Cancer Center

Oklahoma City, Oklahoma, United States

Providence Cancer Institute

Portland, Oregon, United States

SCRI Oncology Partners

Nashville, Tennessee, United States

Vanderbilt Ingram Cancer Center

Nashville, Tennessee, United States

NEXT Oncology - Austin

Austin, Texas, United States

NEXT Oncology - Dallas

Dallas, Texas, United States

Mary Crowley Cancer Research

Dallas, Texas, United States

MD Anderson Cancer Center - University of Texas

Houston, Texas, United States

START Mountain Region

West Valley City, Utah, United States

NEXT Oncology - Virginia Cancer Specialists

Fairfax, Virginia, United States

Fred Hutchinson Cancer Center

Seattle, Washington, United States

Centre Georges François Leclerc

Dijon, France

Institut de Cancerologie de l'Ouest

Saint-Herblain, France

Institut Universitaire du Cancer de Toulouse (IUCT) Oncopole Institut Claudius Regaud "

Toulouse, France

The START center Dublin

Dublin, Dublin, Ireland

Cork University Hospital, Wilton

Cork, Ireland

St. Vincent's University Hospital

Dublin, Ireland

Azienda Ospedaliero Universitaria Careggi - Largo Giovanni Alessandro Brambilla 3

Florence, Italy

Netherlands Cancer Institute-Antoni van Leeuwenhoek

Amsterdam, Netherlands

Seoul National University Hospital

Seoul, South Korea

Severance Hospital - Yonsei Cancer Center

Seoul, South Korea

Asan Medical Center

Seoul, South Korea

Samsung Medical Center

Seoul, South Korea

Hospital Universitario Vall dHebron

Barcelona, Spain

Hospital Universitario 12 de Octubre

Madrid, Spain

START Madrid CIOCC, Hospital Universitario HM Sanchinarro

Madrid, Spain

Hospital Universitario Virgen del Rocio

Seville, Spain

Hospital Clinico Universitario de Valencia (INCLIVA)

Valencia, Spain

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NCT06253871


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