RecruitingPhase 3NCT06357533

Phase III, Open-label, Study of First-line Dato-DXd in Combination With Rilvegostomig for Advanced Non-squamous NSCLC With High PD-L1 Expression (TC ≥ 50%) and Without Actionable Genomic Alterations

A Phase III, Randomised, Open-label, Global Study of Datopotamab Deruxtecan (Dato-DXd) in Combination With Rilvegostomig or Rilvegostomig Monotherapy Versus Pembrolizumab Monotherapy for the First-line Treatment of Participants With Locally-advanced or Metastatic Non-squamous NSCLC With High PD-L1 Expression (TC ≥ 50%) and Without Actionable Genomic Alterations (TROPION-Lung10)


Sponsor

AstraZeneca

Enrollment

675 participants

Start Date

Apr 11, 2024

Study Type

INTERVENTIONAL

Summary

The purpose of this study is to evaluate efficacy and safety of Dato-DXd in combination with rilvegostomig or rilvegostomig monotherapy compared with pembrolizumab monotherapy as a first line therapy in participants with locally advanced or metastatic non-squamous NSCLC with high PD-L1 expression (TC ≥ 50%) and without actionable genomic alterations.


Eligibility

Min Age: 18 Years

Inclusion Criteria8

  • Histologically or cytologically documented non-squamous NSCLC.
  • Stage IIIB or IIIC or Stage IV metastatic NSCLC (according to Edition 8 of the AJCC staging manual) not amenable to curative surgery or definitive chemoradiation.
  • Absence of sensitising EGFR mutations, and ALK and ROS1 rearrangements, and absence of documented local test result for any other known genomic alteration for which there are locally approved and available targeted first-line therapies.
  • Must provide tumor sample to determine PD-L1 status, TROP2 status and other biomarkers.
  • Known tumour PD-L1 expression status defined as TC ≥ 50%
  • At least one lesion, not previously irradiated that qualifies as a RECIST 1.1 target lesion at baseline
  • ECOG performance status of 0 or 1
  • Adequate bone marrow reserve and organ function

Exclusion Criteria13

  • Prior systemic therapy for advanced/metastatic NSCLC.
  • Squamous cell histology, or predominantly squamous cell histology NSCLC; mixed small cell lung cancer; NSCLC histology, sarcomatoid variant.
  • History of another primary malignancy within 3 years
  • Active or prior documented autoimmune or inflammatory disorders (with exceptions)
  • Any evidence of severe or uncontrolled disease that makes it undesirable for the participant to participate in the study or that would jeopardies compliance with the protocol.
  • Has clinically significant third-space fluid retention (for example pleural effusion) and is not amenable for repeated drainage.
  • History of any ILD/pneumonitis, including radiation pneumonitis (apart from radiation pneumonitis that did not require steroids), or drug-induced ILD/pneumonitis, has current or suspected ILD/pneumonitis that cannot be ruled out by imaging at screening.
  • Has significant pulmonary function compromise, as determined by the investigator
  • Spinal cord compression, or brain metastases unless participant treated and no longer symptomatic, radiologically stable, and who require no treatment with corticosteroids or anticonvulsants.
  • History of leptomeningeal carcinomatosis
  • Known clinically significant corneal disease
  • Active infection with TB, HBV, HCV, Hepatitis A, or known HIV infection that is not well controlled
  • History of active primary immunodeficiency

Interventions

DRUGDatopotamab Deruxtecan

Datopotamab Deruxtecan IV (intravenous)

DRUGRilvegostomig

Rilvegostomig IV (intravenous)

DRUGPembrolizumab

Pembrolizumab IV (intravenous)


Locations(281)

Research Site

Anchorage, Alaska, United States

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Tucson, Arizona, United States

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Little Rock, Arkansas, United States

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Springdale, Arkansas, United States

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Anaheim, California, United States

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Beverly Hills, California, United States

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Fountain Valley, California, United States

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Newport Beach, California, United States

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Clermont, Florida, United States

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Gainesville, Florida, United States

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Miami Beach, Florida, United States

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Orange City, Florida, United States

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Orlando, Florida, United States

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Orlando, Florida, United States

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West Palm Beach, Florida, United States

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Atlanta, Georgia, United States

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Atlanta, Georgia, United States

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Atlanta, Georgia, United States

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Atlanta, Georgia, United States

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Hinsdale, Illinois, United States

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Noblesville, Indiana, United States

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Paducah, Kentucky, United States

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Annapolis, Maryland, United States

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Boston, Massachusetts, United States

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Boston, Massachusetts, United States

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Dearborn, Michigan, United States

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Farmington Hills, Michigan, United States

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Grand Rapids, Michigan, United States

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Traverse City, Michigan, United States

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Hattiesburg, Mississippi, United States

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Kansas City, Missouri, United States

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Bozeman, Montana, United States

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Grand Island, Nebraska, United States

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Omaha, Nebraska, United States

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Las Vegas, Nevada, United States

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Reno, Nevada, United States

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Voorhees Township, New Jersey, United States

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Stony Brook, New York, United States

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Greenville, North Carolina, United States

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Salisbury, North Carolina, United States

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Cincinnati, Ohio, United States

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Columbus, Ohio, United States

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Maumee, Ohio, United States

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Toledo, Ohio, United States

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Portland, Oregon, United States

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Greenville, South Carolina, United States

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Sioux Falls, South Dakota, United States

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Chattanooga, Tennessee, United States

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Knoxville, Tennessee, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Kingwood, Texas, United States

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Odessa, Texas, United States

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Fort Belvoir, Virginia, United States

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Leesburg, Virginia, United States

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Midlothian, Virginia, United States

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Richmond, Virginia, United States

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Tacoma, Washington, United States

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Vancouver, Washington, United States

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Wenatchee, Washington, United States

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Appleton, Wisconsin, United States

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Birtinya, Australia

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Blacktown, Australia

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Clayton, Australia

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Gosford, Australia

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Melbourne, Australia

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South Brisbane, Australia

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Wodonga, Australia

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Innsbruck, Austria

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Krems, Austria

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Linz, Austria

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Rankweil, Austria

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Vienna, Austria

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Vienna, Austria

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Wels, Austria

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Anderlecht, Belgium

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Bruges, Belgium

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Hasselt, Belgium

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La Louvière, Belgium

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Liège, Belgium

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Barretos, Brazil

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Curitiba, Brazil

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Florianópolis, Brazil

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Ipatinga, Brazil

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Natal, Brazil

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Porto Alegre, Brazil

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Rio de Janeiro, Brazil

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Santa Maria, Brazil

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São Paulo, Brazil

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Taubaté, Brazil

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Vancouver, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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St. John's, Newfoundland and Labrador, Canada

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London, Ontario, Canada

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Newmarket, Ontario, Canada

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Oshawa, Ontario, Canada

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Toronto, Ontario, Canada

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Lévis, Quebec, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Rimouski, Quebec, Canada

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Trois-Rivières, Quebec, Canada

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Saskatoon, Saskatchewan, Canada

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Chicoutimi, Canada

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Beijing, China

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Beijing, China

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Changchun, China

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Changsha, China

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Chengdu, China

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Chengdu, China

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Chongqing, China

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Fuzhou, China

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Guangzhou, China

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Hangzhou, China

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Hangzhou, China

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Hangzhou, China

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Harbin, China

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Hefei, China

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Hefei, China

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Jinan, China

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Jining, China

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Kunming, China

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Lanzhou, China

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Linhai, China

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Linyi, China

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Nanjing, China

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Nanning, China

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Nanning, China

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Shanghai, China

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Shanghai, China

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Shanghai, China

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Shenyang, China

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Taiyuan, China

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Tianjin, China

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Wenzhou, China

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Wuhan, China

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Wuhan, China

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Wuhan, China

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Wuhan, China

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Xi'an, China

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Yangzhou, China

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Zhengzhou, China

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Zhengzhou, China

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Berlin, Germany

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Bonn, Germany

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Düsseldorf, Germany

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Essen, Germany

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Freiburg im Breisgau, Germany

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Gauting, Germany

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Georgsmarienhütte, Germany

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Gera, Germany

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Gütersloh, Germany

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Hamburg, Germany

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Hamburg, Germany

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Heidelberg, Germany

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Kempten, Germany

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Koblenz, Germany

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Ludwigsburg, Germany

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München, Germany

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Nuremberg, Germany

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Potsdam, Germany

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Ravensburg, Germany

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Budapest, Hungary

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Gyöngyös, Hungary

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Gyöngyös - Mátraháza, Hungary

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Győr, Hungary

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Gyula, Hungary

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Kecskemét, Hungary

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Salgótarján, Hungary

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Szekszárd, Hungary

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Székesfehérvár, Hungary

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Törökbálint, Hungary

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Chennai, India

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Dwārka, India

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Jaipur, India

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Kolkata, India

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Marg Jaipur, India

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Nagpur, India

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Nashik, India

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New Delhi, India

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New Delhi, India

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Surat, India

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Thiruvananthapuram, India

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Bergamo, Italy

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Genoa, Italy

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Milan, Italy

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Milan, Italy

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Monza, Italy

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Padua, Italy

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Pavia, Italy

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Ravenna, Italy

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Roma, Italy

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Rozzano, Italy

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Bunkyō City, Japan

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Bunkyō City, Japan

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Fukuoka, Japan

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Fukuoka, Japan

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Hidaka-shi, Japan

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Hirakata-shi, Japan

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Hirosaki-shi, Japan

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Hiroshima, Japan

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Kanazawa, Japan

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Kashiwa, Japan

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Kawasaki-shi, Japan

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Kumamoto, Japan

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Matsusaka-shi, Japan

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Nagoya, Japan

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Niigata, Japan

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Okayama, Japan

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Osaka, Japan

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Osakasayama-shi, Japan

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Sagamihara-shi, Japan

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Sapporo, Japan

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Takaoka-shi, Japan

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Takatsuki-shi, Japan

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Tokushima, Japan

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Tokyo, Japan

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Utsunomiya, Japan

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Yokohama, Japan

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Olsztyn, Poland

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Poznan, Poland

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Przemyśl, Poland

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Warsaw, Poland

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Warsaw, Poland

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San Juan, Puerto Rico

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Changwon, South Korea

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Incheon, South Korea

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Seongnam-si, South Korea

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Seoul, South Korea

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Seoul, South Korea

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Suwon, South Korea

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Suwon, South Korea

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Alicante, Spain

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Barcelona, Spain

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Barcelona, Spain

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Barcelona, Spain

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Jerez de la Frontera, Spain

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Reus,Tarragona, Spain

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Salamanca, Spain

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Kaohsiung City, Taiwan

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New Taipei City, Taiwan

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Taichung, Taiwan

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Taichung, Taiwan

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Tainan, Taiwan

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Taipei, Taiwan

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Taipei, Taiwan

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Taipei, Taiwan

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Taipei, Taiwan

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Taoyuan District, Taiwan

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Bangkok, Thailand

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Hat Yai, Thailand

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Muang, Thailand

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Mueang, Thailand

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Mueang, Thailand

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Adapazarı, Turkey (Türkiye)

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Ankara, Turkey (Türkiye)

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Ankara, Turkey (Türkiye)

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Antalya, Turkey (Türkiye)

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Diyarbakır, Turkey (Türkiye)

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Istanbul, Turkey (Türkiye)

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Istanbul, Turkey (Türkiye)

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Cheltenham, United Kingdom

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Inverness, United Kingdom

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London, United Kingdom

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London, United Kingdom

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London, United Kingdom

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Preston, United Kingdom

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Truro, United Kingdom

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Da Nang, Vietnam

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Hanoi, Vietnam

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Hanoi, Vietnam

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Hà Nội, Vietnam

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Ho Chi Minh City, Vietnam

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Ho Chi Minh City, Vietnam

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Ho Chi Minh City, Vietnam

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Huế, Vietnam

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Vinh, Vietnam

Research Site

Vĩnh Yên, Vietnam

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NCT06357533