RecruitingPhase 3NCT06629779

A Study to Learn How PF-06821497 (Mevrometostat) Works in Men With Metastatic Castration-resistant Prostate Cancer.

A PHASE 3, RANDOMIZED, DOUBLE BLIND, PLACEBO CONTROLLED STUDY OF PF-06821497 (MEVROMETOSTAT) WITH ENZALUTAMIDE IN METASTATIC CASTRATION RESISTANT PROSTATE CANCER (MEVPRO-2)


Sponsor

Pfizer

Enrollment

900 participants

Start Date

Oct 22, 2024

Study Type

INTERVENTIONAL

Summary

This study will explore whether a combination of the investigational drug PF-06821497 and enzalutamide will work better than taking enzalutamide alone in participants with mCRPC who are ARSi or abiraterone naïve.


Eligibility

Sex: MALEMin Age: 18 Years

Inclusion Criteria4

  • Histologically or cytologically confirmed adenocarcinoma of the prostate without small cell features.
  • Metastatic disease in bone documented on bone scan, or in soft tissue documented on CT/MRI scan.
  • Progressive disease in the setting of medical or surgical castration.
  • ECOG performance status 0 or 1, with a life expectancy of ≥12 months as assessed by the investigator.

Exclusion Criteria10

  • Any medical or psychiatric condition including recent (within the past year) or active suicidal ideation/behavior or laboratory abnormality that make the participant inappropriate for the study.
  • Known history of active inflammatory gastrointestinal disease, chronic diarrhea, or previous gastric resection or lap-band surgery.
  • Clinically significant cardiovascular disease.
  • Known or suspected brain metastasis or active leptomeningeal disease or clinically significant history of seizure.
  • Any history of myelodysplastic syndrome, acute myeloid leukemia, or any other prior malignancy with a few exceptions.
  • Participants must be treatment naïve at the mCRPC stage, eg, no cytotoxic chemotherapy, radio-ligand therapy (i.e. 177Lu- PSMA-617), CDK4/6 inhibitors, 5-alpha reductase inhibitors for prostate cancer in any setting, androgen receptor signaling inhibitors (ARSi) including enzalutamide, apalutamide, darolutamide, poly ADP-ribose polymerase (PARP) monotherapy or other systemic anti-cancer treatment with the following exceptions:
  • Treatment with first-generation antiandrogen (ADT) agents;
  • Docetaxel treatment is allowed for mCSPC, as long as no signs of failure, or disease progression occurred during treatment or within 3 months of treatment completion.
  • Previous administration with an investigational product (drug or vaccine) within 30 days or 5 half-lives preceding the first dose of study intervention (whichever is longer).
  • Inadequate organ function.

Interventions

DRUGPF-06821497

Oral continuous

DRUGPlacebo

Oral continuous

DRUGEnzalutamide

Oral continuous


Locations(240)

Ironwood Cancer & Research Centers

Chandler, Arizona, United States

Ironwood Cancer & Research Centers

Gilbert, Arizona, United States

Palo Verde Hematology Oncology

Glendale, Arizona, United States

Ironwood Cancer & Research Centers

Glendale, Arizona, United States

Ironwood Cancer & Research Centers

Goodyear, Arizona, United States

Ironwood Cancer & Research Centers

Mesa, Arizona, United States

Ironwood Cancer & Research Centers

Mesa, Arizona, United States

Ironwood Cancer & Research Centers

Phoenix, Arizona, United States

Ironwood Cancer & Research Centers

Scottsdale, Arizona, United States

Highlands Oncology

Fayetteville, Arkansas, United States

Arkansas Urology - Little Rock

Little Rock, Arkansas, United States

Highlands Oncology

Rogers, Arkansas, United States

Highlands Oncology Group

Springdale, Arkansas, United States

Los Angeles Cancer Network (LACN)

Anaheim, California, United States

Los Angeles Cancer Network (LACN)

Fountain Valley, California, United States

Los Angeles Cancer Network (LACN)

Glendale, California, United States

Los Angeles Cancer Network (LACN)

Glendale, California, United States

Los Angeles Cancer Network (LACN)

Los Angeles, California, United States

Los Angeles Cancer Network (LACN)

Los Angeles, California, United States

Medical Oncology Associates of San Diego

San Diego, California, United States

Accellacare of Duly

Lisle, Illinois, United States

Duly Health and Care (Bone Scintigraphy)

Lisle, Illinois, United States

Blessing Hospital

Quincy, Illinois, United States

Blessing Physician Services

Quincy, Illinois, United States

Duly Health and Care (CT and MRI)

Westmont, Illinois, United States

Adult & Pediatric Urology, PC

Omaha, Nebraska, United States

CHRISTUS St. Vincent Regional Cancer Center

Santa Fe, New Mexico, United States

Montefiore Medical Center - Medical Park

The Bronx, New York, United States

Montefiore Medical Center

The Bronx, New York, United States

Salisbury VA Medical Center

Salisbury, North Carolina, United States

AUC Urologists, LLC

Myrtle Beach, South Carolina, United States

Carolina Urologic Research Center, LLC

Myrtle Beach, South Carolina, United States

Grand Strand Medical Center

Myrtle Beach, South Carolina, United States

Parkway Surgery Center

Myrtle Beach, South Carolina, United States

USA Clinical Trials

San Antonio, Texas, United States

Northwest Medical Specialties, PLLC

Bonney Lake, Washington, United States

Northwest Medical Specialties, PLLC

Federal Way, Washington, United States

Northwest Medical Specialties, PLLC

Gig Harbor, Washington, United States

Northwest Medical Specialties, PLLC

Puyallup, Washington, United States

Harborview Medical Center

Seattle, Washington, United States

Fred Hutchinson Cancer Center

Seattle, Washington, United States

University of Washington Medical Center - Montlake

Seattle, Washington, United States

Northwest Medical Specialties, PLLC

Tacoma, Washington, United States

Centro de Urología (CDU)

CABA, Buenos Aires, Argentina

Hospital Sirio Libanes

Capital Federal, Buenos Aires, Argentina

Imagenes Mdq

Mar del Plata, Buenos Aires, Argentina

Instituto de Investigaciones Clínicas Mar del Plata

Mar del Plata, Buenos Aires, Argentina

Centro Medico Privado CEMAIC

Capital, Córdoba Province, Argentina

Hospital Privado Universitario de Córdoba

Córdoba, Córdoba Province, Argentina

IMAXE

Buenos Aires, Argentina

Centro Medico Fleischer

Buenos Aires, Argentina

Oncocentro Servico Medicos e Hospitalares Ltda

Fortaleza, Ceará, Brazil

Hospital São Carlos

Fortaleza, Ceará, Brazil

Oncocentro Oncologia

Fortaleza, Ceará, Brazil

Crio - Centro Regional Integrado de Oncologia

Fortaleza, Ceará, Brazil

Instituto D'Or de Pesquisa e Ensino (IDOR) - Filial Salvador

Salvador, Estado de Bahia, Brazil

Hospital Da Bahia

Salvador, Estado de Bahia, Brazil

Clinica Amo - Rio Vermelho

Salvador, Estado de Bahia, Brazil

Hospital Sirio Libanes

Brasília, Federal District, Brazil

Liga Norte Riograndense Contra o Câncer

Natal, Rio Grande do Norte, Brazil

Hospital São Lucas da PUCRS

Porto Alegre, Rio Grande do Sul, Brazil

MedPlex Eixo Norte

Porto Alegre, Rio Grande do Sul, Brazil

Hospital Nossa Senhora da Conceição

Porto Alegre, Rio Grande do Sul, Brazil

Fundação Pio XII - Hospital de Câncer de Barretos

Barretos, São Paulo, Brazil

CEPHO - Centro de Estudos e Pesquisas de Hematologia e Oncologia

Santo André, São Paulo, Brazil

Fundação Faculdade Regional de Medicina de São José do Rio Preto

São José do Rio Preto, São Paulo, Brazil

Hospital Alemao Oswaldo Cruz

São Paulo, São Paulo, Brazil

Instituto do Cancer Arnaldo Vieira de Carvalho

São Paulo, Brazil

IBCC - Núcleo de Pesquisa e Ensino

São Paulo, Brazil

Multiprofile Hospital for Active Treatment Dr. Tota Venkova AD

Gabrovo, Bulgaria

"University Multiprofile Hospital for Active Treatment - Dr. Georgi Stranski" EAD

Pleven, Bulgaria

Complex Oncology Center - Plovdiv EOOD

Plovdiv, Bulgaria

University Multiprofile Hospital for Active Treatment Sofiamed

Sofia, Bulgaria

Complex Oncology Center Stara Zagora EOOD

Stara Zagora, Bulgaria

Prostate Cancer Centre

Calgary, Alberta, Canada

Cross Cancer Institute

Edmonton, Alberta, Canada

QEII Health Sciences Centre - Victoria General Site

Halifax, Nova Scotia, Canada

Lakeridge Health

Oshawa, Ontario, Canada

CIUSSS- saguenay-Lac-Saint-Jean

Chicoutimi, Quebec, Canada

Centre Hospitalier de l'Université de Montréal

Montreal, Quebec, Canada

IC La Serena Research

La Serena, Coquimbo Region, Chile

Clinica Universidad Catolica del Maule

Talca, Maule Region, Chile

Centro de Investigacion Clinica del Sur

Temuco, Región de la Araucanía, Chile

Oncocentro Apys

Viña del Mar, Región de Valparaíso, Chile

Fundación Arturo López Pérez

Providencia, Santiago Metropolitan, Chile

Fundacion Arturo Lopez Perez

Providencia, Santiago Metropolitan, Chile

Oncovida

Providencia, Santiago Metropolitan, Chile

Centro de Estudios Clínicos SAGA

Santiago, Santiago Metropolitan, Chile

FALP

Santiago, Santiago Metropolitan, Chile

Bradfordhill

Santiago, Santiago Metropolitan, Chile

Wannan Medical College Yijishan Hospital

Wuhu, Anhui, China

Cancer Hospital Chinese Academy of Medical Science

Beijing, Beijing Municipality, China

Fujian Cancer Hospital

Fuzhou, Fujian, China

Guangzhou First People's Hospital

Guangzhou, Guangdong, China

The Second Affiliated Hospital of Shantou University School of Medicine

Shantou, Guangdong, China

The Second Affiliated Hospital of Guilin Medical University

Guilin, Guangxi, China

The Third Affiliated Hospital of Xinxiang Medical University

Xinxiang, Henan, China

Henan Cancer Hospital

Zhengzhou, Henan, China

Union Hospital Tongji Medical College Huazhong University of Science and Technology

Wuhan, Hubei, China

Hunan Cancer Hospital

Changsha, Hunan, China

Inner Mongolia People's Hospital

Hohhot, Inner Mongolia, China

Huai'an First People's Hospital

Huai'an, Jiangsu, China

Nanjing Drum Tower Hospital The Affiliated Hospital of Nanjing University Medical School

Nanjing, Jiangsu, China

Nantong Tumor Hospital

Nantong, Jiangsu, China

The Second Affiliated Hospital of Soochow University

Suzhou, Jiangsu, China

The First Affiliated Hospital of Xi'an Jiaotong University

Xi'an, Shaanxi, China

Shaanxi Provincial People' Hospital

Xi'an, Shaanxi, China

Shandong Provincial Hospital

Jinan, Shandong, China

The Affiliated Hospital of Qingdao University

Qingdao, Shandong, China

Weifang People's Hospital

Weifang, Shandong, China

Yantai Yuhuangding Hospital

Yantai, Shandong, China

Tongji Hospital of Tongji University

Shanghai, Shanghai Municipality, China

West China Hospital, Sichuan University

Chengdu, Sichuan, China

Sir Run Run Shaw Hospital, Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

The first affiliated hospital of Ningbo university

Ningbo, Zhejiang, China

The First Affiliated Hospital of Wenzhou Medical University

Wenzhou, Zhejiang, China

The First Hospital of Jiaxing

Jiaxing, Zhejiang/nanhu, China

Peking University Third Hospital

Beijing, China

First Affiliated Hospital of China Medical University

Shenyang, China

Fakultni nemocnice Ostrava

Ostrava, Moravskoslezský kraj, Czechia

Fakultní nemocnice Ostrava

Ostrava - Poruba, Moravskoslezský kraj, Czechia

Fakultni nemocnice Olomouc

Olomouc, Olomoucký kraj, Czechia

Multiscan

Pardubice, Pardubický kraj, Czechia

Fakultni nemocnice Kralovske Vinohrady

Prague, Praha 10, Czechia

Urocentrum Praha

Prague, Praha 2, Czechia

Fakultni Thomayerova nemocnice

Prague, Praha 4, Czechia

Krajská nemocnice Liberec

Liberec, Czechia

Næstved Sygehus

Næstved, Region Sjælland, Denmark

Odense Universitetshospital

Odense, Region Syddanmark, Denmark

Vejle Sygehus

Vejle, Region Syddanmark, Denmark

Oulun yliopistollinen sairaala

Oulu, North Ostrobothnia, Finland

Kuopion Yliopistollinen Sairaala

Kuopio, Northern Savonia, Finland

Tampereen yliopistollinen sairaala

Tampere, Pirkanmaa, Finland

Turku University Hospital

Turku, Southwest Finland, Finland

Helsinki university hospital

Helsinki, Finland

Institut Bergonié - Centre Régional de Lutte Contre Le Cancer de Bordeaux et Sud Ouest

Bordeaux, Aquitaine, France

Centre Leon Berard

Lyon Cedex08, Auvergne-Rhône-Alpes, France

Hopitaux Universitaire de Strasbourg - Hopital Hautepierre

Strasbourg, Bas-rhin, France

CHRU de Brest

Brest, Finistère, France

Centre Hospitalier Privé Saint-Grégoire

Saint-Grégoire, Ille-et-vilaine, France

Institut de Cancérologie de l'Ouest

Saint-Herblain, Loire-atlantique, France

Institut Jean Godinot

Reims, Marne, France

Clinique Victor Hugo Le Mans

Le Mans, Pays de la Loire Region, France

Centre Hospitalier Lyon Sud

Pierre-Bénite, Rhône, France

Centre Jean Perrin - Centre Régional de Lutte contre le Cancer d'Auvergne

Clermont-Ferrand, France

Institut Godinot

Reims, France

Studienpraxis Urologie

Nürtingen, Baden-Wurttemberg, Germany

Universitaetsklinikum Tuebingen

Tübingen, Baden-Wurttemberg, Germany

Universitätsklinikum Münster - Albert Schweitzer Campus

Münster, North Rhine-Westphalia, Germany

Universitaetsklinikum Hamburg-Eppendorf

Hamburg, Germany

University Hospital of Patras

Pátrai, Achaḯa, Greece

Alexandra General Hospital of Athens

Athens, Attikí, Greece

Athens Medical Center

Athens, Attikí, Greece

University General Hospital "ATTIKON" - General Hospital of West Attica "H AGIA VARVARA"

Chaïdári, Attikí, Greece

University General Hospital of Larissa

Larissa, Thessalía, Greece

Borsod-Abaúj-Zemplén Vármegyei Központi Kórház és Egyetemi Oktatókórház

Miskolc, Borsod-Abauj Zemplen county, Hungary

Petz Aladar Egyetemi Oktato Korhaz

Győr, Győr-Moson-Sopron, Hungary

Nograd Varmegyei Szent Lazar Korhaz

Salgótarján, Nógrád megye, Hungary

Országos Onkológiai Intézet

Budapest, Pest County, Hungary

IRCCS - Istituto Romagnolo per lo Studio dei Tumori (IRST) "Dino Amadori"

Meldola, Emilia-Romagna, Italy

Istituto Nazionale Tumori Regina Elena

Rome, Lazio, Italy

Fondazione Policlinico Universitario Agostino Gemelli IRCCS - Università Cattolica del Sacro Cuore

Rome, Lazio, Italy

IRCCS Istituto Clinico Humanitas

Rozzano, Milano, Italy

Azienda Socio Sanitaria Territoriale di Cremona

Cremona, Italy

Ospedale San Raffaele

Milan, Italy

Istituto Nazionale Tumori IRCCS Fondazione Pascale

Napoli, Italy

Azienda Ospedaliera Santa Maria Terni

Terni, Italy

APSS- Presidio Ospedaliero S. Chiara

Trento, Italy

Azienda Ospedaliera Universitaria Integrata Verona - Ospedale Borgo Roma

Verona, Italy

Chiba cancer center

Chiba, Chiba, Japan

National Cancer Center Hospital East

Kashiwa, Chiba, Japan

National Hospital Organization Shikoku Cancer Center

Matsuyama, Ehime, Japan

National Hospital Organization Hokkaido Cancer Center

Sapporo, Hokkaido, Japan

Hokkaido University Hospital

Sapporo, Hokkaido, Japan

Kobe University Hospital

Kobe, Hyōgo, Japan

Kanazawa University Hospital

Kanazawa, Ishikawa-ken, Japan

Yokohama City University Medical Center

Yokohama, Kanagawa, Japan

Yokosuka Kyosai Hospital

Yokosuka, Kanagawa, Japan

The University of Osaka Hospital

Suita, Osaka, Japan

Keio university hospital

Shinjuku-ku, Tokyo, Japan

National Hospital Organization Kyushu Cancer Center

Fukuoka, Japan

National Hospital Organization Kumamoto Medical Center

Kumamoto, Japan

Osaka International Cancer Institute

Osaka, Japan

Yamagata University Hospital

Yamagata, Japan

Canisius-Wilhelmina Ziekenhuis

Nijmegen, Gelderland, Netherlands

Frisius Medisch Centrum

Leeuwarden, Provincie Friesland, Netherlands

Franciscus Gasthuis & Vlietland, Locatie Vlietland

Schiedam, South Holland, Netherlands

Imed Radiology

Tauranga, Bay of Plenty, New Zealand

Tauranga Hospital

Tauranga, Bay of Plenty, New Zealand

Christchurch Hospital

Christchurch, Canterbury, New Zealand

Waikato Hospital

Hamilton, Waikato Region, New Zealand

Auckland City Hospital

Auckland, New Zealand

Regionalny Szpital Specjalistyczny im. dr. Władyslawa Biegańskiego

Grudziądz, Kuyavian-Pomeranian Voivodeship, Poland

MICS Centrum Medyczne Torun

Torun, Kuyavian-Pomeranian Voivodeship, Poland

Centrum Badań Klinicznych Jagiellońskie Centrum Innowacji sp. z o.o.

Krakow, Lesser Poland Voivodeship, Poland

Szpital Specjalistyczny im. Ludwika Rydygiera w Krakowie

Krakow, Lesser Poland Voivodeship, Poland

4 Wojskowy Szpital Kliniczny z Polikliniką SPZOZ

Wroclaw, Lower Silesian Voivodeship, Poland

Clinical Best Solutions

Lublin, Lublin Voivodeship, Poland

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie - Panstwowy Instytut Badawczy w Warszawie

Warsaw, Masovian Voivodeship, Poland

Szpital Wojewódzki im. Mikoaja Kopernika w Koszalinie

Koszalin, West Pomeranian Voivodeship, Poland

SP ZOZ Opolskie Centrum Onkologii im. prof. Tadeusza Koszarowskiego w Opolu

Opole, Poland

Provita Profamilia

Piotrkow Trybunalski, Łódź Voivodeship, Poland

CUIMED, s.r.o., Urologicka ambulancia

Bratislava, Slovakia

Univerzitna nemocnica Martin

Martin, Slovakia

Privatna urologicka ambulancia, s.r.o.

Trenčín, Slovakia

Cancercare Langenhoven Drive Oncology Centre

Port Elizabeth, Eastern Cape, South Africa

Wilgers Oncology Centre

Pretoria, Gauteng, South Africa

Wits Clinical Research

Soweto, Gauteng, South Africa

TASK Eden

George, Western Cape, South Africa

Chonnam National University Hwasun Hospital

Hwasun, Jeonranamdo, South Korea

National Cancer Center

Goyang-si, Kyǒnggi-do, South Korea

Seoul National University Hospital

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Severance Hospital, Yonsei University Health System

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Asan Medical Center

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Samsung Medical Center

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Kyungpook National University Chilgok Hospital

Daegu, Taegu-kwangyǒkshi, South Korea

Chungnam national university hospital

Junggu, Taejǒn-kwangyǒkshi, South Korea

Institut Català d'Oncologia - L'Hospitalet

L'Hospitalet de Llobregat, Catalunya [cataluña], Spain

Hospital Universitario 12 de Octubre

Madrid, Madrid, Comunidad de, Spain

Fundación Instituto Valenciano de Oncología

Valencia, Valenciana, Comunitat, Spain

Hospital Universitario Fundación Jiménez Díaz

Madrid, Spain

Hospital Universitario HM Sanchinarro

Madrid, Spain

Södersjukhuset

Stockholm, Stockholms LÄN [se-01], Sweden

Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung City, Taiwan

Taichung Veterans General Hospital

Taichung, Taiwan

National Cheng Kung University Hospital

Tainan, Taiwan

National Taiwan University Hospital

Taipei, Taiwan

Taipei Veterans General Hospital

Taipei, Taiwan

Koç Üniversitesi Hastanesi

Istanbul, İ̇stanbul, Turkey (Türkiye)

TC Saglik Bakanligi Goztepe Prof. Dr. Suleyman Yalcin Sehir Hastanesi

Istanbul, İ̇stanbul, Turkey (Türkiye)

Marmara Universitesi Pendik Egitim Arastirma Hastanesi

Istanbul, İ̇stanbul, Turkey (Türkiye)

I.E.U. Medical Point Hastanesi

Izmir, İ̇zmir, Turkey (Türkiye)

Sbü Gülhane Eğitim Ve Araştirma Hastanesi

Ankara, Turkey (Türkiye)

Memorial Ankara Hastanesi

Ankara, Turkey (Türkiye)

Ankara University Health Practice and Research Hospitals

Ankara, Turkey (Türkiye)

Royal Blackburn Hospital

Blackburn, Blackburn WITH Darwen, United Kingdom

Mid and South Essex NHS Foundation Trust

Chelmsford, Essex, United Kingdom

Royal Derby Hospital

Derby, United Kingdom

The Beatson West of Scotland Cancer Centre

Glasgow, United Kingdom

The Clatterbridge Cancer Centre

Metropolitan Borough of Wirral, United Kingdom

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NCT06629779