RecruitingPhase 2NCT06651567

A Study to Assess the Efficacy and Safety of ITI-1284 in the Treatment of Agitation Associated With Alzheimer's Dementia

A Multicenter, Randomized, Double-blind, Placebo-controlled, Flexible-dose Study of the Efficacy, Safety, and Tolerability of ITI-1284 in Patients With Agitation Associated With Alzheimer's Dementia


Sponsor

Intra-Cellular Therapies, Inc.

Enrollment

320 participants

Start Date

Oct 22, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

This is a multicenter, randomized, double-blind, placebo-controlled, flexible-dose study of the efficacy, safety, and tolerability of ITI-1284 in patients with agitation associated with Alzheimer's dementia


Eligibility

Min Age: 55 Years

Inclusion Criteria8

  • Can understand the nature of the trial and protocol requirements and provide signed informed consent, if in the judgement of the Investigator is deemed competent to provide consent or if patient is deemed not competent to provide informed consent, with the patient's assent (if capable), consent may be provided by an appropriate person (eg, patient's Legally Authorized Representative \[LAR\]) before the initiation of any study-specific procedures in accordance with local regulations;
  • Meets clinical criteria for Alzheimer's disease based on 2011 National Institute of Aging-Alzheimer's Association (NIA-AA) dementia criteria and biomarker criteria and either:
  • Has a high likelihood for amyloid pathology consistent with Alzheimer's disease, as confirmed by blood-based biomarker at Screening; or
  • Has historical documentation of cerebrospinal fluid (CSF) biomarker or amyloid positron emission tomography (PET) brain scan;
  • Meets all criteria for agitation according to the International Psychogeriatric Association (IPA) consensus definition
  • Has clinically meaningful agitation defined as a Neuropsychiatric Inventory-Agitation/Aggression (NPI-AA) domain total score of ≥ 4 at both Screening and Baseline;
  • CGI-S score ≥ 4 at Screening and Baseline;
  • Has Mini-Mental State Examination, 2nd Edition™: Standard Version (MMSE-2®:SV) score of 6 to 24 at Screening;

Exclusion Criteria7

  • Agitation symptoms are attributable to concomitant medications, adverse environmental conditions, substance abuse, or active medical or psychiatric conditions as per Investigator's judgment;
  • Has been diagnosed with one or more of the following psychiatric conditions:
  • Schizophrenia, schizoaffective disorder, or other psychotic disorder that is not related to Alzheimer's dementia;
  • Bipolar disorder;
  • Major depressive disorder, unless it is considered stable and treated for at least 8 weeks prior to Screening;
  • Has a significant risk for suicidal behavior during the course of their participation in the study, or is considered to be an imminent danger to themselves or others, in the opinion of the investigator, and/or as assessed by Columbia Suicide Severity Rating Scale (C-SSRS); or the patient has had 1 or more suicide attempts within the 2 years prior to Screening;
  • The patient has known hypersensitivity or intolerance to ITI-1284 or lumateperone, or to any of their excipients.

Interventions

DRUGITI-1284

ITI-1284 10 mg or 20 mg rapidly disintegrating tablet, taken once daily, sublingual administration

DRUGPlacebo

Placebo rapidly disintegrating tablet, taken once daily, sublingual administration


Locations(69)

Clinical Site

Bratislava, Slovakia

Clinical Site

Košice, Slovakia

Clinical Site

Krompachy, Slovakia

Clinical Site

Svidník, Slovakia

Clinical Site

Anaheim, California, United States

Clinical Site

Costa Mesa, California, United States

Clinical Site

Garden Grove, California, United States

Clinical Site

Boca Raton, Florida, United States

Clinical Site

Bonita Springs, Florida, United States

Clinical Site

Brandon, Florida, United States

Clinical Site

Delray Beach, Florida, United States

Clinical Site

Doral, Florida, United States

Clinical Site

Hialeah, Florida, United States

Clinical Site

Homestead, Florida, United States

Clinical Site_2

Maitland, Florida, United States

Clinical Site

Maitland, Florida, United States

Clinical Site

Miami, Florida, United States

Clinical Site_2

Miami, Florida, United States

Clinical Site_3

Miami, Florida, United States

Clinical Site

Miami, Florida, United States

Clinical Site

Miami, Florida, United States

Clinical Site

Miami, Florida, United States

Clinical Site

Miami, Florida, United States

Clinical Site

Miami, Florida, United States

Clinical Site

Orlando, Florida, United States

Clinical Site

Orlando, Florida, United States

Clinical Site_2

Tampa, Florida, United States

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Tampa, Florida, United States

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West Palm Beach, Florida, United States

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Boston, Massachusetts, United States

Clinical Site

Las Vegas, Nevada, United States

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Toms River, New Jersey, United States

Clinical Site

Raleigh, North Carolina, United States

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San Antonio, Texas, United States

Clinical Site

Lovech, Bulgaria

Clinical Site

Pleven, Bulgaria

Clinical Site

Sofia, Bulgaria

Clinical Site

Sofia, Bulgaria

Clinical Site

Sofia, Bulgaria

Clinical Site

Sofia, Bulgaria

Clinical Site

Stara Zagora, Bulgaria

Clinical Site_2

Zagreb, Croatia

Clinical Site_3

Zagreb, Croatia

Clinical Site

Zagreb, Croatia

Clinical Site

Zagreb, Croatia

Clinical Site

Brno, Czechia

Clinical Site

Choceň, Czechia

Clinical Site

Kutná Hora, Czechia

Clinical Site

Pilsen, Czechia

Clinical Site

Prague, Czechia

Clinical Site

Prague, Czechia

Clinical Site

Bucharest, Romania

Clinical Site

Bucharest, Romania

Clinical Site

Bucharest, Romania

Clinical Site

Bucharest, Romania

Clinical Site

Sânpetru, Romania

Clinical Site

Sibiu, Romania

Clinical Site_2

Belgrade, Serbia

Clinical Site

Belgrade, Serbia

Clinical Site

Kovin, Serbia

Clinical Site

Niš, Serbia

Clinical Site

Novi Kneževac, Serbia

Clinical Site

Banská Bystrica, Slovakia

Clinical Site

Vranov nad Topľou, Slovakia

Clinical Site

Albacete, Spain

Clinical Site

Barcelona, Spain

Clinical Site

Málaga, Spain

Clinical Site

Zamora, Spain

Clinical Site

Zaragoza, Spain

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NCT06651567