RecruitingPhase 2NCT06793371

AMBER-HFpEF: Assessment of CK-4021586 in a Multi-Center, Blinded Evaluation of Safety and Tolerability Results in HFpEF

A Multi-Center, Randomized, Double-Blind, Placebo-Controlled Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of CK-4021586 in Adults With Symptomatic Heart Failure With Preserved Ejection Fraction


Sponsor

Cytokinetics

Enrollment

60 participants

Start Date

Feb 6, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This is a Phase 2 dose-finding study in adult participants with symptomatic HFpEF.


Eligibility

Min Age: 40 YearsMax Age: 85 Years

Inclusion Criteria7

  • Males and females ≥ 40 years and ≤ 85 years of age at screening.
  • Diagnosed with HF with NYHA functional class II or III.
  • Screening echocardiography with LVEF ≥ 60%.
  • Screening NT-proBNP ≥ 300 pg/mL for participants in sinus rhythm and ≥ 900 pg/mL for participants with comorbid atrial fibrillation or flutter.
  • Body mass index \< 40 kg/m2.
  • Participants on beta-blockers, angiotensin-converting enzyme (ACE)/angiotensin II receptor blocker (ARB) or angiotensin receptor/neprilysin inhibitor (ARNI), must be on stable doses for more than 30 days prior to screening.
  • Participants on a glucagon-like peptide-1 (GLP-1) agonist must be on a stable dose for more than 24 weeks prior to screening with no anticipated plans to change dose during this study.

Exclusion Criteria1

  • History or evidence of any other clinically significant disorder, malignancy, active infection, other condition, or disease that, in the opinion of the investigator or the Medical Monitor, would pose a risk to patient safety or interfere with the study evaluation, procedures, or completion.

Interventions

DRUGCK-4021586 (150 mg, 300 mg, 450 mg, and 600 mg)

CK-4021586 administered orally

DRUGPlacebo to match CK-4021586

Placebo administered orally


Locations(24)

Eastern Shore Research Institute, LLC

Fairhope, Alabama, United States

University of Arizona Sarver Heart Center

Tucson, Arizona, United States

John L. McClellan Memorial Veterans Hospital

Little Rock, Arkansas, United States

BioSolutions Clinical Research Center

Imperial, California, United States

Profound Research LLC

Pasadena, California, United States

University of California, San Francisco - Heart and Vascular Center

San Francisco, California, United States

FOMAT - Comprehensive Cardiovascular Care

Santa Maria, California, United States

Blue Coast Research Center, LLC

Vista, California, United States

New Generation of Medical Research

Hialeah, Florida, United States

Cleveland Clinic Florida

Weston, Florida, United States

Methodist Medical Center of Illinois

Peoria, Illinois, United States

Louisiana Heart Center

Slidell, Louisiana, United States

Massachusetts General Hospital

Boston, Massachusetts, United States

Mayo Clinic

Rochester, Minnesota, United States

Washington University Center for Advanced Medicine

St Louis, Missouri, United States

Morristown Medical Center

Morristown, New Jersey, United States

NYU Langone Health

New York, New York, United States

The Lindner Center for Research & Education at The Christ Hospital

Cincinnati, Ohio, United States

Oregon Health and Science University

Portland, Oregon, United States

University of Texas Southwestern Medical Center, Dallas

Dallas, Texas, United States

Center for Advanced Heart Failure

Houston, Texas, United States

DelRicht Research

Vienna, Virginia, United States

Swedish Heart & Vascular Institute, Advanced Cardiac Support Program

Seattle, Washington, United States

Froedtert Hospital - Center for Advanced Care

Milwaukee, Wisconsin, United States

View Full Details on ClinicalTrials.gov

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NCT06793371