RecruitingPhase 2NCT06855771

A Study of BMS-986504 in Participants With Pre-treated Advanced or Metastatic Non-small Cell Lung Cancer (NSCLC) With Homozygous MTAP Deletion (MountainTAP-9)

A Multicenter, Randomized, Open-label, Phase 2 Study Evaluating the Safety and Efficacy of BMS-986504 Monotherapy in Participants With Advanced or Metastatic Non-small Cell Lung Cancer (NSCLC) With Homozygous MTAP Deletion After Progression on Prior Therapies


Sponsor

Bristol-Myers Squibb

Enrollment

130 participants

Start Date

Sep 9, 2025

Study Type

INTERVENTIONAL

Summary

The purpose of this study is to evaluate the safety and efficacy of BMS-986504 monotherapy in participants with advanced or metastatic Non-small Cell Lung Cancer (NSCLC) with homozygous MTAP deletion after progression on prior therapies.


Eligibility

Min Age: 18 Years

Inclusion Criteria7

  • Histologically confirmed diagnosis of NSCLC and homozygous MTAP deletion detected in tumor tissue and willingness to provide archival/fresh samples at screening for central MTAP status confirmation.
  • Advanced or metastatic NSCLC not amenable to curative therapies after progression on prior therapies at the time of enrollment (based on the American Joint Committee on Cancer, Ninth Edition).
  • At least 1 measurable lesion as per RECIST v1.1.
  • Documented radiographic disease progression on or after the most recent line of treatment.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0-1.
  • Participant must be ≥ 18 years of age (or the legal age of consent in the jurisdiction in which the study is taking place) at the time of signing the ICF.
  • Capability to swallow tablets intact (without chewing or crushing).

Exclusion Criteria4

  • Active brain metastases or carcinomatous meningitis.
  • History of gastrointestinal disease or other gastrointestinal conditions (eg, uncontrolled nausea, vomiting, malabsorption syndrome) likely to alter absorption of study treatment or result in inability to swallow oral medications.
  • Prior treatment with a PRMT5 or MAT2A inhibitor.
  • Known severe hypersensitivity to study treatment and/or any of its excipients.

Interventions

DRUGBMS-986504

Specified dose on specified days


Locations(71)

Alaska Oncology and Hematology

Anchorage, Alaska, United States

Local Institution - 0099

Boise, Idaho, United States

Dana-Farber Cancer Institute

Boston, Massachusetts, United States

Karmanos Cancer Institute

Detroit, Michigan, United States

Washington University School of Medicine

St Louis, Missouri, United States

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Local Institution - 0079

Shirley, New York, United States

Gabrail Cancer Center

Canton, Ohio, United States

Providence Portland Medical Center

Portland, Oregon, United States

Oregon Health and Science University

Portland, Oregon, United States

Fred Hutchison Cancer Center

Seattle, Washington, United States

Local Institution - 0084

Milwaukee, Wisconsin, United States

GenesisCare - Campbelltown

Campbelltown, New South Wales, Australia

Chris O'Brien Lifehouse

Camperdown, New South Wales, Australia

Princess Alexandra Hospital

Woolloongabba, Queensland, Australia

GenesisCare - St Andrew's

Adelaide, South Australia, Australia

Local Institution - 0039

Beijing, Beijing Municipality, China

The First Affiliated hospital of Xiamen University

Xiamen, Fujian, China

Guangxi Medical University Affiliated Tumor Hospital

Nanning, Guangxi, China

The First Affiliated Hospital of Nanchang University

Nanchang, Jiangxi, China

Local Institution - 0056

Changchun, Jilin, China

Shandong Cancer Hospital

Jinan, Shandong, China

Local Institution - 0044

Linyi, Shandong, China

Sir Run Run Shaw Hospital of Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Taizhou Hospital of Zhejiang Province

Linhai, Zhejiang, China

Local Institution - 0045

Marseille, Bouches-du-Rhône, France

Chu Grenoble Alpes

La Tronche, Isère, France

Hôpital Nord Guillaume-et-René-Laennec / CHU de Nantes

Saint-Herblain, Loire-Atlantique, France

Centre Hospitalier Régional Universitaire de Nancy - Hôpitaux de Brabois

Vandœuvre-lès-Nancy, Meurthe-et-Moselle, France

Hospices Civils de Lyon - Hopital Louis Pradel

Bron, Rhône, France

Hopitaux Universitaires Paris Centre-Hopital Cochin

Paris, France

Local Institution - 0107

Paris, France

Hôpital Tenon

Paris, France

Groupe hospitalier Paris saint Joseph

Paris, Île-de-France Region, France

Klinikum der Ludwig-Maximilians-Universitaet Muenchen

München, Bavaria, Germany

Universitätsklinikum Frankfurt Goethe-Universität

Frankfurt am Main, Hesse, Germany

Krankenhaus Martha-Maria Halle-Dölau

Halle, Saxony-Anhalt, Germany

Universitaetsklinikum Koeln

Cologne, Germany

Universitaetsklinikum Wuerzburg

Würzburg, Germany

AOU della Campania Luigi Vanvitelli

Napoli, Campania, Italy

Istituto Nazionale Tumori IRCCS Fondazione Pascale

Napoli, Campania, Italy

Fondazione IRCCS San Gerardo dei Tintori

Monza, Lombardy, Italy

ASST Grande Ospedale Metropolitano Niguarda

Milan, Milano, Italy

Istituto Oncologico Veneto IRCCS

Padua, Veneto, Italy

IRCCS Azienda Ospedaliero-Universitaria di Bologna, Policlinico di Sant'Orsola

Bologna, Italy

Fondazione IRCCS Istituto Nazionale dei Tumori

Milan, Italy

Local Institution - 0092

Kashiwa, Chiba, Japan

Local Institution - 0094

Sendai, Miyagi, Japan

Local Institution - 0093

Hirakata, Osaka, Japan

Mazowiecki Szpital Onkologiczny

Wieliszew, Masovian Voivodeship, Poland

Szpital Specjalistyczny w Prabutach Spolka z o.o.

Prabuty, Poland

Institutul Oncologic Bucuresti "Prof. Dr. Alexandru Trestioreanu"

Bucharest, București, Romania

SC Radiotherapy Center Cluj SRL

Florești, Cluj, Romania

Centrul de Oncologie "Sfântul Nectarie"

Craiova, Dolj, Romania

Centrul de Diagnostic si Tratament Provita

Bucharest, Romania

Institutul Oncologic Cluj

Cluj-Napoca, Romania

S.C. Centrul de Oncologie Euroclinic S.R.L.

Iași, Romania

Institutul Regional de Oncologie

Iași, Romania

Hospital Universitari Vall d'Hebron

Barcelona, Barcelona [Barcelona], Spain

Institut Català d'Oncologia - L'Hospitalet

Hospitalet, Barcelona [Barcelona], Spain

Hospital Universitario Ramón y Cajal

Madrid, Madrid, Comunidad de, Spain

Hospital Universitario 12 de Octubre

Madrid, Madrid, Comunidad de, Spain

Hospital Universitario La Paz

Madrid, Madrid, Comunidad de, Spain

H.R.U Málaga - Hospital General

Málaga, Spain

Hospital Universitario Virgen Del Rocio

Seville, Spain

Hospital Universitari i Politecnic La Fe

Valencia, Spain

Karolinska Universitetssjukhuset Solna

Solna, Stockholms Län [se-01], Sweden

Sahlgrenska Universitetssjukhuset

Gothenburg, Västra Götalands Län [se-14], Sweden

Queen Elizabeth Hospital Birmingham

Birmingham, England, United Kingdom

Sarah Cannon Research Institute UK

London, London, City of, United Kingdom

Freeman Hospital

Newcastle upon Tyne, United Kingdom

View Full Details on ClinicalTrials.gov

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NCT06855771