RecruitingPhase 2NCT06931405

Study of BLU-808 in Chronic Inducible Urticaria (CIndU) and Chronic Spontaneous Urticaria (CSU)

A Phase 2 Study to Evaluate the Safety, Tolerability, and Clinical Activity of BLU-808, a Wild Type KIT Inhibitor, in Chronic Inducible Urticaria and Chronic Spontaneous Urticaria


Sponsor

Blueprint Medicines Corporation

Enrollment

105 participants

Start Date

May 28, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This is a 2-part, proof-of-concept study to be conducted globally, designed to evaluate the safety, tolerability, clinical activity, pharmacokinetics, and pharmacodynamics of BLU-808, a wild type KIT inhibitor, in participants with CIndU (Part A) or CSU (Part B).


Eligibility

Min Age: 18 Years

Inclusion Criteria2

  • Part A: Confirmed diagnosis of CIndU for ≥3 months prior to Day 1 that is inadequately controlled with second generation H1-antihistamines.
  • Part B: Confirmed diagnosis of CSU for ≥3 months prior to Day 1 that is inadequately controlled with second generation H1-antihistamines.

Exclusion Criteria6

  • Part A: Any active urticaria that may interfere with study assessments.
  • Part B: Participant has a clearly defined predominant cause of chronic urticaria or sole trigger such as symptomatic dermographism and cold-induced urticaria.
  • Part A and Part B: Any other skin disease associated with chronic itching or angioedema that might influence the study evaluations and results, skin diseases associated with only wheals and no itch, or autoinflammatory diseases with urticarial lesions.
  • Part A and Part B: Significant medical, psychiatric, or surgical conditions, or physical findings that may affect participant safety, study drug metabolism, study participation, or assessment of study results.
  • Part A and Part B: Abnormal laboratory values that may pose risks or interfere with study participation.
  • Part A and Part B: Pregnancy or plans for pregnancy; breastfeeding.

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Interventions

DRUGBLU-808

Oral administration

DRUGPlacebo

Oral administration


Locations(47)

Allervie Clinical Research

Birmingham, Alabama, United States

Acuro Research, Inc.

Little Rock, Arkansas, United States

Modena Allergy & Asthma Clinical Research - La Jolla

La Jolla, California, United States

Allergy & Asthma Associates of Southern California

Laguna Niguel, California, United States

Allergy & Asthma Medical Group and Research Center

San Diego, California, United States

Allergy Affiliates Inc.

Bradenton, Florida, United States

University of South Florida

Tampa, Florida, United States

Treasure Valley Medical Research

Boise, Idaho, United States

Endeavor Health

Northbrook, Illinois, United States

Dawes Fretzin Clinical Research Group, LLC

Indianapolis, Indiana, United States

Southern Indiana Clinical Trials

New Albany, Indiana, United States

The Indiana Clinical Trials Center

Plainfield, Indiana, United States

Equity Medical - Bowling Green

Bowling Green, Kentucky, United States

Johns Hopkins University

Baltimore, Maryland, United States

Institute For Asthma & Allergy

Wheaton, Maryland, United States

Chesapeake Clinical Research

White Marsh, Maryland, United States

Henry Ford Health

Detroit, Michigan, United States

Mayo Clinic

Rochester, Minnesota, United States

The Clinical Research Center LLC.

St Louis, Missouri, United States

Montana Medical Research, Inc.

Missoula, Montana, United States

Equity Medical (at Cameron Dermatology) - New York

New York, New York, United States

Bernstein Clinical Research Center

Cincinnati, Ohio, United States

Allergy & Clinical Immunology Associates

Pittsburgh, Pennsylvania, United States

National Allergy, Asthma & Urticaria Centers of Charleston

Charleston, South Carolina, United States

Medical University of South Carolina (MUSC)

Charleston, South Carolina, United States

Reveal Research Institute

Dallas, Texas, United States

Austin Institute for Clinical Research

Pflugerville, Texas, United States

Odense University Hospital - Odense

Odense, Denmark

Fraunhofer-Institut fuer Translationale Medizin und Pharmakologie ITMP - Standort Berlin

Berlin, Germany

Universitaetsklinikum Carl Gustav Carus Dresden

Dresden, Germany

Universitaetsklinikum Frankfurt - Klinikum der Johann Wolfgang Goethe Universitaet

Frankfurt am Main, Germany

Medizinische Hochschule Hannover (MHH)

Hanover, Germany

Universitaetsmedizin der Johannes Gutenberg - Universitaet Mainz

Mainz, Germany

Universitaetsklinikum Tuebingen

Tübingen, Germany

Azienda Ospedale - Università Padova

Padova, Italy

Azienda Ospedaliero Universitaria Policlinico Umberto

Rome, Italy

Centro Ricerche Cliniche di Verona s.r.l.

Verona, Italy

Hospital del Mar

Barcelona, Spain

Hospital Universitario Vall d'Hebron

Barcelona, Spain

Hospital Universitari de Bellvitge

Barcelona, Spain

Hospital Regional Universitario de Malaga

Málaga, Spain

National Taiwan University Hospital Hsin-Chu Branch

Hsinchu, Taiwan

Kaohsiung Veterans General Hospital (KSVGH)

Kaohsiung City, Taiwan

Taipei Medical University - Shuang Ho Hospital

New Taipei City, Taiwan

China Medical University Hospital

Taichung, Taiwan

National Taiwan University Hospital

Taipei, Taiwan

Linkou Chang Gung Memorial Hospital (CGMHLK)

Taoyuan, Taiwan

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NCT06931405


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