RecruitingPhase 2NCT06963710

A Study Evaluating the Efficacy and Safety of ALG-000184 Compared With Tenofovir Disoproxil Fumarate in Untreated HBeAg-Positive and HBeAg- Negative Adult Subjects With Chronic Hepatitis B (B-SUPREME)

A Randomized, Double-Blind, Active-Controlled Multicenter Phase 2 Study Evaluating the Efficacy and Safety of ALG-000184 Compared With Tenofovir Disoproxil Fumarate in Untreated HBeAg-Positive and HBeAg-Negative Adult Subjects With Chronic Hepatitis B Virus Infection (B-SUPREME)


Sponsor

Aligos Therapeutics

Enrollment

200 participants

Start Date

Jul 15, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This is a Phase 2 study to evaluate efficacy and safety of 48 weeks of oral once daily monotherapy with ALG-000184 versus tenofovir disproxil fumarate (TDF) for chronic HBV infection.


Eligibility

Min Age: 18 YearsMax Age: 65 Years

Inclusion Criteria8

  • Male or female between 18 and 65 years of age, with body mass index (BMI) of 18.0 to 35.0 kg/m2 (or minimun age by local regulatory requirements).
  • HBeAg-positive and anti-HBeAg (HBeAb) negative (Part 1); or HBeAg-negative (Part 2).
  • HBsAg ≥LLOQ.
  • HBV DNA ≥20,000 IU/mL.
  • A history of a clinical diagnosis of chronic HBV infection AND an ALT values of ≤8×ULN during screening.
  • Must have the following chronic hepatitis B virus infection treatment status at screening:
  • Have never received treatment with HBV antiviral medicines (NA, interferon) or investigational anti-HBV agents including a CAM \[i.e., Treatment Naïve (TN) subjects\], OR
  • Have not been on treatment with approved (NA, interferon) or investigational HBV antiviral medicines (e.g., antisense oligonucleotides or small interfering RNAs) within 6 months or 5 half-lives (whichever is longer) prior to randomization (i.e., Currently Not Treated (CNT) subjects).

Exclusion Criteria11

  • Co-infection with hepatitis A, C, D, E or HIV or any evidence of clinically significant liver disease of non-HBV etiology.
  • Positive for anti-HBs antibodies.
  • History or current evidence of cirrhosis.
  • Liver fibrosis that is classified as Metavir Score ≥F3 liver disease.
  • History of, or current evidence of, hepatic decompensation.
  • Evidence of hepatocellular carcinoma (HCC) on a liver ultrasound.
  • Having received an investigational medicinal product or device within 4 weeks (or 5 half-lives, whichever is longer) before the planned first dose of study drug
  • Exclusionary screening laboratory values include:
  • Aspartate aminotransferase (AST) >8×ULN,
  • Bilirubin (total, direct) >1.2×ULN (unless Gilbert's syndrome is suspected)
  • International Normalization Ratio (INR) >1.2×ULN

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Interventions

DRUGALG-000184

300 mg tablet

DRUGTDF

300 mg tablet


Locations(58)

Aligos Investigational Site

Chandler, Arizona, United States

Aligos Investigational Site

Coronado, California, United States

Aligos Investigational Site

Garden Grove, California, United States

Aligos Investigational Site

Los Angeles, California, United States

Aligos Investigational Site

Palo Alto, California, United States

Aligos Investigational Site

Pasadena, California, United States

Aligos Investigational Site

Rialto, California, United States

Aligos Investigational Site

San Francisco, California, United States

Aligos Investigational Site

San Jose, California, United States

Aligos Investigational Site

Miami, Florida, United States

Aligos Investigational Site

Miami, Florida, United States

Aligos Investigational Site

Marrero, Louisiana, United States

Aligos Investigational Site

Baltimore, Maryland, United States

Aligos Investigational Site

Chevy Chase, Maryland, United States

Aligos Investigational Site

Boston, Massachusetts, United States

Aligos Investigational Site

Manhasset, New York, United States

Aligos Investigational Site

New York, New York, United States

Aligos Investigational Site

Durham, North Carolina, United States

Aligos Investigational Site

Sliven, Bulgaria

Aligos Investigational Sites

Sofia, Bulgaria

Aligos Investigational Site

Stara Zagora, Bulgaria

Aligos Investigational Site

Edmonton, Canada

Aligos Investigational Site

Ottawa, Canada

Aligos Investigational Site

Toronto, Canada

Aligos Investigational Sites

Vancouver, Canada

Aligos Investigational Sites

Beijing, China

Aligos Investigational Site

Changchun, China

Aligos Investigational Site

Chengdu, China

Aligos Investigational Site

Chongqing, China

Aligos Investigational Sites

Guangzhou, China

Aligos Investigational Site

Nanjing, China

Aligos Investigational Sites

Shanghai, China

Aligos Investigational Site

Clichy, France

Aligos Investigational Site

Limoges, France

Aligos Investigational Site

Nice, France

Aligos Investigational Site

Rennes, France

Aligos Investigational Site

Rouen, France

Aligos Investigational Site

Toulouse, France

Aligos Investigational Sites

Hong Kong, Hong Kong

Aligos Investigational Site

Milan, Italy

Aligos Investigational Site

Chisinau, Moldova

Aligos Investigational Site

Auckland, New Zealand

Aligos Investigational Sites

Bucharest, Romania

Aligos Investigational Site

Ansan, South Korea

Aligos Investigational Site

Busan, South Korea

Aligos Investigational Sites

Seoul, South Korea

Aligos Investigational Site

Ulsan, South Korea

Aligos Investigational Site

Yangsan, South Korea

Aligos Investigational Site

Barcelona, Spain

Aligos Investigational Site

Pontevedra, Spain

Aligos Investigational Site

Chiayi City, Taiwan

Aligos Investigational Site

Kaohsiung City, Taiwan

Aligos Investigational Site

Taichung, Taiwan

Aligos Investigational Site

Tainan, Taiwan

Aligos Investigational Site

Taipei, Taiwan

Aligos Investigational Site

Glasgow, United Kingdom

Aligos Investigational Site

Leicester, United Kingdom

Aligos Investigational Sites

London, United Kingdom

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NCT06963710


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