RecruitingPhase 3NCT07008976

Clinical Trial of TQB2102 for Injection Versus Trastuzumab Emtansine for Injection in HER2-positive Advanced Breast Cancer

A Randomized, Open-label, Parallel-controlled Phase III Clinical Trial to Evaluate the Efficacy and Safety of TQB2102 for Injection Versus Trastuzumab Emtansine for Injection in Patients With HER2-positive Advanced Breast Cancer


Sponsor

Chia Tai Tianqing Pharmaceutical Group Nanjing Shunxin Pharmaceutical Co., Ltd.

Enrollment

246 participants

Start Date

Jul 7, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This study adopted a randomized, open-label, positive drug-controlled, multi-center trial design. The primary endpoint was PFS evaluated by the Independent Review Committee (IRC). Eligible subjects were randomly assigned in a 1:1 ratio to receive either TQB2102 for injection or trastuzumab emtansine for injection.


Eligibility

Min Age: 18 YearsMax Age: 75 Years

Inclusion Criteria10

  • The subjects voluntarily participated in this study, signed the informed consent form, and had good compliance;
  • Age: 18 - 75 years old (at the time of signing the informed consent form); Eastern Cooperative Oncology Group (ECOG )score ≤ 1; Expected survival period exceeds 3 months;
  • HER2-positive, unresectable, locally advanced or metastatic invasive breast cancer confirmed by histopathological or cytological examination;
  • According to the 2018 version of the American Society of Clinical Oncology (ASCO)/College of American Pathologists (CAP )HumanEpidermalGrowthFactorReceptor2 (HER2) testing guidelines, HER2 positive is defined as: immunohistochemical result of 3+ or Fluorescence In Situ Hybridization (FISH) dual probe positive;
  • The hormone receptor (HR) status has been clearly determined:
  • a) According to the 2020 version of the ASCO/CAP guidelines, HR positive includes ER positive and/or PR positive, that is, the proportion of tumor cells with positive staining among all tumor cells is ≥ 1%.
  • Received anti-HER2 monoclonal antibody and taxane drugs during the recurrence/metastasis stage.
  • Disease progression occurred during or after the most recent treatment or intolerance.
  • At least 1 line of treatment has been received in the recurrence/metastasis stage.
  • According to the Response Evaluation Criteria In Solid Tumors (RECIST) 1.1 standard, at least one measurable lesion exists.

Exclusion Criteria6

  • Excluded are patients with known spinal cord compression or active central nervous system metastases .
  • Patients with only skin and/or intracranial lesions as target lesions.
  • Patients with adverse reactions from previous treatments that have not recovered to a CTCAE v5.0 grade score of ≤1.
  • Patients with poorly controlled blood pressure (systolic blood pressure ≥150 mmHg or diastolic blood pressure ≥100 mmHg).
  • Patients with major cardiovascular diseases
  • Patients with a history of interstitial lung disease/pneumonia (non-infectious type) requiring steroid intervention treatment, or currently having interstitial lung disease/pneumonia, or those with suspected interstitial lung disease/pneumonia indicated by screening period imaging and cannot be excluded.

Interventions

DRUGTQB2102 Injection

TQB2102 Injection is a Human Epidermal Growth Factor Receptor 2 (HER2) bispecific antibody-drug conjugate.

DRUGTrastuzumab Emtansine for Injection

Trastuzumab Emtansine for Injection is HER2-targeting antibody-drug conjugate (ADC).


Locations(31)

The First Affiliated Hospital of Anhui Medical University

Bengbu, Anhui, China

Anhui Provincial Cancer Hospital

Hefei, Anhui, China

The First Affiliated Hospital of Anhui Medical University

Hefei, Anhui, China

Peking University First Hospital

Beijing, Beijing Municipality, China

Beijing Shunyi Hospital

Beijing, Beijing Municipality, China

Fujian Cancer Hospital

Fuzhou, Fujian, China

The First Hospital Of Lanzhou University

Lanzhou, Gansu, China

Jiangmen Central Hospital

Jiangmen, Guangdong, China

Affiliated Cancer Hospital Of Guangxi Medical University

Nanning, Guangxi, China

Cancer Hospital Of Guizhou Medical University

Guiyang, Guizhou, China

Hainan General Hospital

Haikou, Hainan, China

The Fourth Hospital Of Hebei Medical University

Shijiazhuang, Hebei, China

Affiliated Cancer Hospital Of Harbin Medical University

Harbin, Heilongjiang, China

Jiamusi Tuberculosis Hospital (Jiamusi Tumor Hospital)

Jiamusi, Heilongjiang, China

Anyang Cancer Hospital

Anyang, Henan, China

The First Affiliated Hospital Of Henan University Of Science & Technology

Luoyang, Henan, China

Henan Cancer Hospital

Zhengzhou, Henan, China

Hunan Cancer Hospital

Changsha, Hunan, China

Chifeng Municipal Hospital

Chifeng, Inner Mongolia, China

Jiangxi Cancer Hospital

Nanchang, Jiangxi, China

Jilin Cancer Hospital

Changchun, Jilin, China

The First Hospital of Jilin University

Changchun, Jilin, China

The Second Hospital Of Dalian Medical University

Dalian, Liaoning, China

Liaoning Cancer Hospital & Institute

Shenyang, Liaoning, China

Affiliated Hospital Of Jining Medical University

Jining, Shandong, China

Linyi Cancer Hospital

Linyi, Shandong, China

Fudan University Shanghai Cancer Center

Shanghai, Shanghai Municipality, China

Dazhopu Central Hospital

Dazhou, Sichuan, China

Affiliated Hospital of North Sichuan Medical College

Nanchong, Sichuan, China

Tianjin Medical University Cancer Institute & Hospital

Tianjin, Tianjin Municipality, China

Hangzhou Cancer Hospital

Hangzhou, Zhejiang, China

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NCT07008976


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