RecruitingPhase 2NCT07023627

A Study of INCB123667 in Participants With Platinum-Resistant Ovarian Cancer With Cyclin E1 Overexpression

A Phase 2, Single-Arm Study of INCB123667 in Participants With Platinum-Resistant Ovarian Cancer With Cyclin E1 Overexpression (MAESTRA 1)


Sponsor

Incyte Corporation

Enrollment

160 participants

Start Date

Nov 12, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This study will evaluate the safety and efficacy of INCB123667 in Participants With Platinum-Resistant Ovarian Cancer (PROC) With Cyclin E1 Overexpression.


Eligibility

Sex: FEMALEMin Age: 18 YearsMax Age: 99 Years

Inclusion Criteria8

  • Histological diagnosis of a high-grade serous epithelial ovarian, fallopian tube, or primary peritoneal cancer.
  • Have platinum-resistant disease:
  • Participants who have only had 1 line of platinum-based therapy must have received at least 4 cycles of a platinum-containing regimen.
  • Participants who have received 2 to 4 lines of platinum-based therapy must have progressed on or within 6 months after the last dose of platinum.
  • Willingness to undergo a pretreatment biopsy. Note: Tissue from a fresh pretreatment biopsy is preferred, however an archival sample is acceptable as long as the sample is no older than 5 years.
  • Received at least 1 and no more than 4 prior lines of systemic therapy following the initial diagnosis, after which single-agent therapy is considered an appropriate next therapeutic option.
  • Must have received bevacizumab unless there was a contraindication for its use.
  • If the tumor tests positive for FRα, participants must have received mirvetuximab soravtansine unless there is an exception for its use on medical grounds.

Exclusion Criteria6

  • Have endometrioid, clear cell, mucinous, or sarcomatous histology, mixed tumors containing any of these histologies, or low-grade/borderline ovarian cancer.
  • Have primary platinum-refractory disease: either did not respond (CR or PR) to first-line platinum-containing therapy or progressed on or within 3 months after the last dose of the first line platinum-containing therapy.
  • The tumor tests positive for FRα but the participant has not received mirvetuximab soravtansine for any reason other than medical contraindication.
  • Clinically significant or uncontrolled cardiac disease within 6 months before the first dose of study drug.
  • Known active CNS metastases and/or carcinomatous meningitis.
  • Known additional malignancy that is progressing or requires active treatment.

Interventions

DRUGINCB123667

Administered orally twice daily (BID).


Locations(79)

Usa Health Mitchell Cancer Institute

Mobile, Alabama, United States

Uams Winthrop P Rockefeller Cancer Institute

Little Rock, Arkansas, United States

University of California, Los Angeles Medical Center

Los Angeles, California, United States

Scripps Healthscripps Mercy Hospital Prebys Cancer Center

San Diego, California, United States

Medstar Georgetown University Hospital

Washington D.C., District of Columbia, United States

Florida Cancer Specialists & Research Institute

Fort Myers, Florida, United States

Sylvester Comprehensive Cancer Center

Miami, Florida, United States

Mount Sinai Comprehensive Cancer Center

Miami Beach, Florida, United States

Florida Cancer Specialists & Research Institute

West Palm Beach, Florida, United States

Northeast Georgia Medical Center Gainesville

Gainesville, Georgia, United States

Parkview Research Center

Fort Wayne, Indiana, United States

University of Iowa Hospital and Clinics

Iowa City, Iowa, United States

Norton Cancer Institute

Louisville, Kentucky, United States

Trials365, Llc

Shreveport, Louisiana, United States

Greater Baltimore Medical Center

Baltimore, Maryland, United States

John Hopkins University-School of Medicine

Baltimore, Maryland, United States

Massachusetts General Hospital

Boston, Massachusetts, United States

Umass Memorial Medical Center, Inc.

Worcester, Massachusetts, United States

University of Michigan Health System

Ann Arbor, Michigan, United States

Minnesota Oncology-Minneapolis

Minneapolis, Minnesota, United States

University of Mississippi Medical Center

Jackson, Mississippi, United States

Washington University

St Louis, Missouri, United States

St. Vincent Regional Hospital - West End Clinic

Billings, Montana, United States

Nebraska Methodist Hospital

Omaha, Nebraska, United States

John Theurer Cancer Center, Hackensack University Medical Center

Hackensack, New Jersey, United States

Laura and Isaac Perlmutter Cancer Center

New York, New York, United States

State University of New York Upstate Medical Unive

Syracuse, New York, United States

Oncology Hematology Care, Inc

Cincinnati, Ohio, United States

The Mark H Zangmeister Cancer Center Ohio

Columbus, Ohio, United States

The Ohio State University Wexner Medical Center Division of Gynecologic Oncology

Hilliard, Ohio, United States

Penn State College of Medicine

Hershey, Pennsylvania, United States

Medical University of South Carolina

Charleston, South Carolina, United States

Texas Oncology-Austin Center

Austin, Texas, United States

Cancer Care Center of South Texas-Medical Center

San Antonio, Texas, United States

Texas Oncology-Tyler

Tyler, Texas, United States

Utah Cancer Specialists

Salt Lake City, Utah, United States

Virginia Cancer Specialists, Pc

Fairfax, Virginia, United States

Carilion Clinic

Roanoke, Virginia, United States

West Virginia University

Morgantown, West Virginia, United States

Froedtert & the Medical College of Wisconsin

Milwaukee, Wisconsin, United States

Blacktown Cancer & Haematology Centre-Blacktown Hospital

Blacktown, New South Wales, Australia

Concord General Repatriation Hospital

Concord, New South Wales, Australia

Burnside War Memorial Hospital - the Brian Fricker Oncology Centre

Adelaide, South Australia, Australia

Hobart Hospital-Royal Hobart Hospital

Hobart, Tasmania, Australia

Cancer Research Sa (Crsa)

Adelaide, Australia

Southern Oncology Clinical Research Unit

South Australia, Australia

Hopital Universitaire de Bruxelles (Hub) - Institut Jules Bordet

Brussels, Belgium

Cliniques Universitaires St Luc Ucl

Brussels, Belgium

Az Groeninge

Kortrijk, Belgium

Universitair Ziekenhuis Leuven

Leuven, Belgium

Chu Liege

Liège, Belgium

Hyogo Cancer Center

Akashi-shi, Japan

Saitama Medical University International Medical Center

Hidaka-shi, Japan

The Cancer Institute Hospital of Jfcr

Kōtoku, Japan

Kurume University Hospital

Kurume, Japan

Shikoku Cancer Center

Matsuyama, Japan

Hokkaido University Hospital

Sapporo Hokkaido, Japan

Shizuoka Cancer Center

Sunto-gun, Japan

Panoncology Trials

San Juan, PR, Puerto Rico

Hospital Universitario Vall D'Hebron

Barcelona, Spain

Hospital Clinic de Barcelona

Barcelona, Spain

Instituto Catalan de Oncologia - Hospital Duran I Reynals

Barcelona, Spain

Hospital Universitario Reina Sofia

Córdoba, Spain

Institut Catala D'Oncologia Girona

Girona, Spain

Clinica Universidad de Navarra - Sede Madrid

Madrid, Spain

Hospital Universitario La Paz

Madrid, Spain

Hospital Universitario Virgen de La Arrixaca

Murcia, Spain

Fundacion Instituto Valenciano de Oncologia

Valencia, Spain

Hospital Clinico Universitario de Valencia (Instituto de Investigacion Sanitaria Incliva)

Valencia, Spain

Istituto Oncologico Della Svizzera Italiana (Iosi) Di Bellinzona

Bellinzona, Switzerland

Kantonsspital Graubunden

Chur, Switzerland

Geneva University Hospitals-Hug

Geneva, Switzerland

Centre Hospitalier Universitaire Vaudois Lausanne (Chuv) - Centre Du Cancer Lausanne-Batiment Hospit

Lausanne, Switzerland

Kantonsspital Baselland (Ksbl) - Standort Liestal - Medizinische Universitatsklinik

Liestal, Switzerland

St Bartholomew'S Hospital

London, United Kingdom

Guy'S Hospital - Guy'S & St Thomas' Nhs Foundation Trust

London, United Kingdom

Royal Marsden Hospital (Sutton) - Royal Marsden Nhs Foundation Trust

London, United Kingdom

Hammersmith Hospital - Imperial College Healthcare Nhs Trust

London, United Kingdom

The Christie Nhs Foundation Trust

Manchester Greater, United Kingdom

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NCT07023627


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