RecruitingPhase 3NCT07028853

This Study Will Explore Whether a Combination of the Investigational Drug Mevrometostat (PF-06821497) and Enzalutamide Will Work Better Than Taking Enzalutamide Alone in Participants With mCSPC Who Are ARPI naïve.

A Phase 3, Randomized, Double-Blind, Placebo-Controlled Study of Mevrometostat (PF-06821497) With Enzalutamide in Metastatic Castration-Sensitive Prostate Cancer (MEVPRO-3)


Sponsor

Pfizer

Enrollment

1,000 participants

Start Date

Sep 28, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This study will explore whether a combination of the investigational drug mevrometostat (PF-06821497) and enzalutamide will work better than taking enzalutamide alone in participants with mCSPC who are ARPI naïve and have not yet received chemotherapy in the mCSPC setting.


Eligibility

Sex: MALEMin Age: 18 Years

Inclusion Criteria5

  • Male participants aged ≥18 years (or the minimum age of consent in accordance with local regulations) at screening.
  • Histologically or cytologically confirmed adenocarcinoma of the prostate without small cell features.
  • Metastatic prostate cancer documented by positive bone scan (for bone disease) or metastatic lesion(s) on CT or MRI (for soft tissue/visceral disease).
  • Resolution of acute effects of any prior therapy to either baseline severity or CTCAE Grade ≤1 (except for AEs which do not constitute a safety risk in the investigator's judgement).
  • Participants must have ECOG PS 0 or 1.

Exclusion Criteria7

  • Any medical or psychiatric condition including recent (within the past year) or active suicidal ideation/behavior or laboratory abnormality that may increase the risk of study participation or, in the investigator's judgment, make the participant inappropriate for the study.
  • Clinically significant cardiovascular disease.
  • Known or suspected brain metastasis or active leptomeningeal disease.
  • Participants must be treatment naïve at the mCSPC stage, eg, participants cannot have received any cytotoxic chemotherapy with the following exceptions: Treatment with first-generation antiandrogen (ADT) agents is allowed for mCSPC.
  • Previous administration with an investigational product (drug or vaccine) within 30 days.
  • Current use or anticipated need for drugs that are known strong CYP3A4/5 inhibitors and inducers (with exception of enzalutamide as part of this study).
  • Inadequate organ function.

Interventions

DRUGMevrometostat

Oral continuous

DRUGPlacebo

Oral continuous

DRUGEnzalutamide

Oral continuous


Locations(188)

Ironwood Cancer & Research Centers

Chandler, Arizona, United States

Ironwood Cancer & Research Centers

Gilbert, Arizona, United States

Ironwood Cancer & Research Centers

Glendale, Arizona, United States

Ironwood Cancer & Research Centers

Goodyear, Arizona, United States

Ironwood Cancer & Research Centers

Mesa, Arizona, United States

Ironwood Cancer & Research Centers

Mesa, Arizona, United States

Ironwood Cancer & Research Centers

Phoenix, Arizona, United States

Ironwood Cancer & Research Centers

Scottsdale, Arizona, United States

Highlands Oncology Group, PA

Fayetteville, Arkansas, United States

Highlands Oncology Group, PA

Rogers, Arkansas, United States

Highlands Oncology Group, PA

Springdale, Arkansas, United States

UCLA Hematology/Oncology - Alhambra

Alhambra, California, United States

UCLA Hematology/Oncology - Atascadero

Atascadero, California, United States

UCLA Hematology/Oncology - Beverly Hills

Beverly Hills, California, United States

UCLA Hematology/Oncology - Burbank

Burbank, California, United States

UCLA Hematology/Oncology - Encino

Encino, California, United States

UCLA Hematology/Oncology - Irvine

Irvine, California, United States

UCLA Hematology/Oncology - Laguna Hills

Laguna Hills, California, United States

Ronald Reagan UCLA Medical Center - Drug Information Center

Los Angeles, California, United States

UCLA Department of Medicine - Hematology/Oncology

Los Angeles, California, United States

UCLA Hematology/Oncology

Los Angeles, California, United States

UCLA Hematology/Oncology - Marina del Rey

Marina del Rey, California, United States

UCLA Hematology/Oncology - Pasadena

Pasadena, California, United States

UCLA Hematology/Oncology - Porter Ranch

Porter Ranch, California, United States

UCLA Hematology/Oncology - San Luis Obispo

San Luis Obispo, California, United States

UCLA Hematology/Oncology - Santa Barbara

Santa Barbara, California, United States

UCLA Hematology/Oncology- Santa Monica

Santa Monica, California, United States

UCLA Hematology/Oncology - Torrance

Torrance, California, United States

UCLA Hematology/Oncology - Santa Clarita

Valencia, California, United States

UCLA Hematology/Oncology - Ventura

Ventura, California, United States

UCLA Hematology/Oncology - Westlake

Westlake Village, California, United States

AdventHealth Medical Group Urology of Denver

Denver, Colorado, United States

Cancer Care Specialists of Illinois

Decatur, Illinois, United States

Cancer Care Specialists of Illinois

O'Fallon, Illinois, United States

University of Rochester Medical Center

Rochester, New York, United States

University of Rochester, Cancer Center Pharmacy (Investigational Product)

Rochester, New York, United States

Montefiore Einstein Comprehensive Cancer Center

The Bronx, New York, United States

Montefiore Medical Center- Montefiore Medical Park

The Bronx, New York, United States

University Hospitals Seidman Cancer Center at UH Avon Health Center

Avon, Ohio, United States

TriState Urologic Services PSC Inc. dba The Urology Group

Cincinnati, Ohio, United States

University Hospitals Cleveland Medical Center

Cleveland, Ohio, United States

University Hospitals Seidman Cancer Center at UH Mentor Health Center

Mentor, Ohio, United States

UH Minoff Health Center at Chagrin Highlands

Orange, Ohio, United States

The Centers for Advanced Urology, LLP d/b/a Keystone Urology Specialists

Lancaster, Pennsylvania, United States

Grand Strand Medical Center

Myrtle Beach, South Carolina, United States

Carolina Urologic Research Center, LLC

Myrtle Beach, South Carolina, United States

Parkway Surgery Center

Myrtle Beach, South Carolina, United States

Urology Associates, P.C.

Nashville, Tennessee, United States

University of Texas Southwestern Medical Center - Simmons Cancer Center

Dallas, Texas, United States

University of Texas Southwestern Medical Center - William P. Clements, Jr., University Hospital

Dallas, Texas, United States

University of Texas Southwestern Simmons Cancer Center - Redbird

Dallas, Texas, United States

University of Texas Southwestern Medical Center-Zale Lipshy University Hospital

Dallas, Texas, United States

University of Texas Southwestern Simmons Cancer Center - Fort Worth

Fort Worth, Texas, United States

US Oncology Investigational Product Center (IPC)

Irving, Texas, United States

Palmerston North Hospital

Palmerston North, New Zealand

University of Texas Southwestern Simmons Cancer Center - Richardson/Plano

Richardson, Texas, United States

Huntsman Cancer Institute

Salt Lake City, Utah, United States

Blue Ridge Cancer Care

Blacksburg, Virginia, United States

Blue Ridge Cancer Care

Low Moor, Virginia, United States

Blue Ridge Cancer Care

Roanoke, Virginia, United States

Blue Ridge Cancer Care

Salem, Virginia, United States

Blue Ridge Cancer Care

Wytheville, Virginia, United States

Northwest Medical Specialties, PLLC

Bonney Lake, Washington, United States

Northwest Medical Specialties, PLLC

Federal Way, Washington, United States

Northwest Medical Specialties, PLLC

Gig Harbor, Washington, United States

Northwest Medical Specialties, PLLC

Puyallup, Washington, United States

Northwest Medical Specialties, PLLC

Tacoma, Washington, United States

University of Wisconsin Carbone Cancer Center - Eastpark Medical Center

Madison, Wisconsin, United States

University of Wisconsin Carbone Cancer Center - University Hospital

Madison, Wisconsin, United States

Asociación de Beneficencia Hospital Sirio Libanés

Ciudad Autonoma de Buenos Aires, Buenos Aires, Argentina

Centro Oncologico Korben

Buenos Aires, Argentina

Orange Health Service

Orange, New South Wales, Australia

Sydney Adventist Hospital

Wahroonga, New South Wales, Australia

Icon Cancer Centre Chermside

Chermside, Queensland, Australia

Mater Misericordiae Limited Mater Cancer Care Centre

South Brisbane, Queensland, Australia

ICON Cancer Centre - Kurralta Park

Kurralta Park, South Australia, Australia

Sir Charles Gairdner Hospital

Perth, Western Australia, Australia

UZ Leuven

Leuven, Vlaams-brabant, Belgium

CEPHO - Centro de Estudos e Pesquisas de Hematologia e Oncologia

Santo André, São Paulo, Brazil

MBAL Uni Hospital

Panagyurishte, Pazardzhik, Bulgaria

Medical Center Futuremeds

Plovdiv, Bulgaria

Complex Oncology Center - Plovdiv EOOD

Plovdiv, Bulgaria

Prostate Cancer Centre

Calgary, Alberta, Canada

Centre of Applied Urology Research/Nova Scotia Health Authority

Halifax, Nova Scotia, Canada

Centre Intégré de Santé et de Services Sociaux de la Montérégie-Centre

Greenfield Park, Quebec, Canada

Centre Hospitalier de l'Université de Montréal

Montreal, Quebec, Canada

Jewish General Hospital

Montreal, Quebec, Canada

Centre intégré de cancérologie du CHU de Québec Université Laval, Hôpital de l'Enfant-Jésus

Québec, Quebec, Canada

Centre intégré universitaire de santé et de services sociaux de l'Estrie - Centre Hospitalier Univer

Sherbrooke, Quebec, Canada

Diex Recherche Trois-Rivieres

Trois-Rivières, Quebec, Canada

Wannan Medical College Yijishan Hospital

Wuhu, Anhui, China

Peking University First Hospital

Beijing, Beijing Municipality, China

Beijing Friendship Hospital Affiliate of Capital University

Beijing, Beijing Municipality, China

The First Affiliated Hospital of Chongqing Medical University

Chongqing, Chongqing Municipality, China

Chongqing University Cancer Hospital

Chongqing, Chongqing Municipality, China

Lanzhou university second hospital

Lanzhou, Gansu, China

The First Affiliated Hospital of Guangzhou Medical University

Guangzhou, Guangdong, China

Sun Yat-sen University Cancer Center

Guangzhou, Guangdong, China

Union Hospital Tongji Medical College Huazhong University of Science and Technology

Wuhan, Hubei, China

Hunan Cancer Hospital

Changsha, Hunan, China

First Huai'an Hospital Affiliated to Nanjing Medical University

Huai'an, Jiangsu, China

Nanjing Drum Tower Hospital The Affiliated Hospital of Nanjing University Medical School

Nanjing, Jiangsu, China

Nantong Tumor Hospital

Nantong, Jiangsu, China

The Second Affiliated Hospital of Soochow University

Suzhou, Jiangsu, China

The First Affiliated Hospital of Xi'an Jiaotong University

Xi'an, Shaanxi, China

Qilu Hospital of Shandong University

Jinan, Shandong, China

Fudan University Shanghai Cancer Center

Shanghai, Shanghai Municipality, China

Suining Central Hospital

Suining, Sichuan, China

Zhejiang Provincial People's Hospital

Hangzhou, Zhejiang, China

Sir Run Run Shaw Hospital of Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

The first affiliated hospital of Ningbo university

Ningbo, Zhejiang, China

The First Affiliated Hospital of Wenzhou Medical University

Wenzhou, Zhejiang, China

The Third Affiliated Hospital of Southern Medical University

Guangzhou, China

Masarykuv onkologicky ustav

Brno, Czechia

Fakultni nemocnice Hradec Kralove

Hradec Králové, Czechia

Urocentrum Praha s.r.o.

Prague, Czechia

Fakultni Thomayerova nemocnice

Prague, Czechia

Fakultni nemocnice v Motole

Prague, Czechia

Institut Bergonié - Centre Régional de Lutte Contre Le Cancer de Bordeaux et Sud Ouest

Bordeaux, Aquitaine, France

Centre Leon Berard

Lyon Cedex08, Auvergne-Rhône-Alpes, France

Centre Hospitalier de la Côte Basque

Bayonne, Pyrénées-atlantiques, France

Urologie Neandertal - Praxis Mettmann

Mettmann, North Rhine-Westphalia, Germany

Universitätsklinikum Münster - Albert Schweitzer Campus

Münster, North Rhine-Westphalia, Germany

Rabin Medical Center

Petah Tikva, Central District, Israel

Sheba Medical Center

Ramat Gan, Central District, Israel

Yitzhak Shamir Medical Center

Ẕerifin, Central District, Israel

Shaare Zedek Medical Center

Jerusalem, Jerusalem, Israel

Hadassah Medical Center

Jerusalem, Jerusalem, Israel

Rambam Health Care Campus

Haifa, Northern District, Israel

Sourasky Medical Center

Tel Aviv, TELL ABĪB, Israel

Chiba cancer center

Chiba, Chiba, Japan

National Hospital Organization Shikoku Cancer Center

Matsuyama, Ehime, Japan

National Hospital Organization Hokkaido Cancer Center

Sapporo, Hokkaido, Japan

Hokkaido University Hospital

Sapporo, Hokkaido, Japan

Kobe University Hospital

Kobe, Hyōgo, Japan

Kanazawa University Hospital

Kanazawa, Ishikawa-ken, Japan

Yokohama City University Medical Center

Yokohama, Kanagawa, Japan

Yokosuka Kyosai Hospital

Yokosuka, Kanagawa, Japan

The University of Osaka Hospital

Suita, Osaka, Japan

Keio university hospital

Shinjuku-ku, Tokyo, Japan

National Hospital Organization Kyushu Cancer Center

Fukuoka, Japan

National Hospital Organization Kumamoto Medical Center

Kumamoto, Japan

Osaka International Cancer Institute

Osaka, Japan

Yamagata University Hospital

Yamagata, Japan

Canisius-Wilhelmina Ziekenhuis

Nijmegen, Gelderland, Netherlands

Tergooi MC

Hilversum, North Holland, Netherlands

Reinier de Graaf Ziekenhuis, locatie Delft

Delft, South Holland, Netherlands

Tauranga Hospital

Tauranga, Bay of Plenty, New Zealand

Waikato Hospital

Hamilton, Waikato Region, New Zealand

Clinical Research Center Spółka z ograniczoną odpowiedzialnością MEDIC-R Sp.k

Poznan, Greater Poland Voivodeship, Poland

Szpital Specjalistyczny im. Ludwika Rydygiera w Krakowie

Krakow, Lesser Poland Voivodeship, Poland

Zachodniopomorskie Centrum Onkologii

Szczecin, West Pomeranian Voivodeship, Poland

Clinical Best Solutions Sp. z o.o. S.K.

Lublin, Poland

Centrum Medyczne MEDYK

Rzeszów, Poland

EMC Instytut Medyczny S.A.

Wroclaw, Poland

MILAB, s.r.o., Urologicka ambulancia

Prešov, Slovakia

Privatna urologicka ambulancia, s.r.o.

Trenčín, Slovakia

Chonnam National University Hwasun Hospital

Hwasun-gun, Jeonranamdo, South Korea

National Cancer Center

Goyang-si, Kyǒnggi-do, South Korea

Seoul National University Bundang Hospital

Seongnam, Kyǒnggi-do, South Korea

Seoul National University Hospital

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Severance Hospital, Yonsei University Health System

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Asan Medical Center

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Samsung Medical Center

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Ewha Womans University Mokdong Hospital

Seoul, Seoul-teukbyeolsi [seoul], South Korea

Kyungpook National University Chilgok Hospital

Deagu, Taegu-kwangyǒkshi, South Korea

Chungnam national university hospital

Junggu, Taejǒn-kwangyǒkshi, South Korea

Parc de Salut Mar - Hospital del Mar

Barcelona, Barcelona [barcelona], Spain

Althaia, Xarxa Assistencial Universitària de Manresa

Manresa, Barcelona, Spain

Hospital Clínic de Barcelona

Barcelona, Catalunya [cataluña], Spain

Hospital Universitario Ramón y Cajal

Madrid, Madrid, Comunidad de, Spain

Hospital Universitario Virgen de la Victoria

Málaga, Málaga, Spain

CHUVI- Hospital Alvaro Cunqueiro

Vigo, Pontevedra [pontevedra], Spain

Fundación Instituto Valenciano de Oncología

Valencia, Valenciana, Comunitat, Spain

Hospital Clinico San Carlos

Madrid, Spain

Inselspital Bern

Bern, Canton of Bern, Switzerland

UniversitätsSpital Zürich

Zurich, Switzerland

Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung City, Taiwan

Taichung Veterans General Hospital

Taichung, Taiwan

National Cheng Kung University Hospital

Tainan, Taiwan

National Taiwan University Hospital

Taipei, Taiwan

Taipei Veterans General Hospital

Taipei, Taiwan

Royal Blackburn Hospital

Blackburn, Blackburn WITH Darwen, United Kingdom

Torbay Hospital

Torquay, Devon, United Kingdom

Imperial College Healthcare NHS Trust, Charing Cross Hospital

London, Hammersmith and Fulham, United Kingdom

Maidstone Hospital

Maidstone, KENT, United Kingdom

Guy's & St Thomas' NHS Foundation Trust

London, London, CITY of, United Kingdom

The Christie NHS Foundation Trust

Manchester, United Kingdom

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NCT07028853


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