RecruitingPhase 1Phase 2NCT07148128

Phase 1/2a Study to Assess the Safety, Tolerability, Pharmacokinetics, and Preliminary Efficacy of WEF-001 as Monotherapy in Advanced KRAS-Mutant Solid Tumours.

An Open-label, Multicenter, Phase 1/2a Study to Investigate the Safety, Tolerability, Pharmacokinetics, and Antitumour Activity of WEF-001 in Participants With Advanced KRAS- Mutant Solid Tumours.


Sponsor

Auricula Biosciences Inc.

Enrollment

110 participants

Start Date

Jul 28, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This is a study designed to assess the safety, tolerability, pharmacokinetics and preliminary efficacy of WEF-001 as monotherapy in patients with Advanced KRAS-mutant solid tumours.


Eligibility

Min Age: 18 Years

Inclusion Criteria4

  • Advanced KRAS-mutant solid tumor: pancreatic ductal adenocarcinoma, colorectal cancer, non small cell lung cancer, platinum-resistant serous ovarian cancer, cholangiocarcinoma or urothelial bladder cancer
  • Progressive disease following at least one line of standard of care therapy
  • Measurable disease as defined by RECIST v1.1
  • ECOG ≤ 1

Exclusion Criteria8

  • Active systemic infection requiring anti-infective therapy within 28 days prior to first dose of IMP
  • Active cardiovascular disease
  • Having a second active primary malignancy, requiring systemic administration of any cancer-related therapy
  • Liver dysfunction
  • Untreated brain metastasis and/or unstable neurological dysfunction
  • Inflammatory bowel disease
  • Active and untreated hyperthyroidism
  • Lupus erythematosus within past 5 years

Interventions

DRUGWEF-001

Starting dose of 0.3 mg/m2 q4wks IV, dose escalation


Locations(4)

NEXT Oncology Dallas

Dallas, Texas, United States

Next Oncology, San Antonio

San Antonio, Texas, United States

Princess Margareth Cancer Center

Toronto, Ontario, Canada

Oxford University Hospital

Headington, Oxford, United Kingdom

View Full Details on ClinicalTrials.gov

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NCT07148128


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