RecruitingPhase 3NCT07211633

A Study to Evaluate the Pharmacokinetics, Pharmacodynamics, Safety, Radiological and Clinical Effects of Subcutaneous Ublituximab in Participants With Relapsing Multiple Sclerosis (RMS)

A Phase 3, Non-Inferiority, Randomized, Open-Label, Parallel Group, Multicenter Study to Evaluate the Pharmacokinetics, Pharmacodynamics, Safety, Radiological and Clinical Effects of Subcutaneous Ublituximab Versus Intravenous Ublituximab in Patients With Multiple Sclerosis


Sponsor

TG Therapeutics, Inc.

Enrollment

360 participants

Start Date

Jul 9, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to assess the pharmacokinetics of ublituximab when administered subcutaneously (SC) compared to intravenous (IV) administration in participants with RMS.


Eligibility

Min Age: 18 YearsMax Age: 65 Years

Inclusion Criteria4

  • Diagnosis of RMS (2017 Revised McDonald criteria).
  • Expanded Disability Status Scale (EDSS) score ≤ 5.5 at screening.
  • Neurologically stable for \> 30 days prior to Screening and Day 1.
  • Female participants of childbearing potential must consent to use a highly effective method of contraception from consent and for 6 months after the last dose of ublituximab.

Exclusion Criteria4

  • Primary-progressive Multiple Sclerosis (PPMS) or inactive Secondary Progressive Multiple Sclerosis (SPMS).
  • Active chronic disease of the immune system other than MS or immunodeficiency syndrome.
  • Participants with significantly impaired bone marrow function or significant leukopenia or thrombocytopenia.
  • Participants who previously received anti-CD20 therapy at any time; any approved therapy to treat MS within 5 half-lives of the medication prior to screening.

Interventions

BIOLOGICALUblituximab

Administered as an IV infusion.

BIOLOGICALUblituximab

Administered as an SC injection.


Locations(42)

TG Therapeutics Investigational Trial Site

Banja Luka, Bosnia and Herzegovina

TG Therapeutics Investigational Trial Site

Bihać, Bosnia and Herzegovina

TG Therapeutics Investigational Trial Site

Mostar, Bosnia and Herzegovina

TG Therapeutics Investigational Trial Site

Saravejo, Bosnia and Herzegovina

TG Therapeutics Investigational Trial Site

Pleven, Bulgaria

TG Therapeutics Investigational Trial Site

Plovdiv, Bulgaria

TG Therapeutics Investigational Trial Site

Sofia, Bulgaria

TG Therapeutics Investigational Trial Site

Veliko Tarnovo, Bulgaria

TG Therapeutics Investigational Trial Site

Varaždin, Croatia

TG Therapeutics Investigational Trial Site

Zagreb, Croatia

TG Therapeutics Investigational Trial Site

Brno, Czechia

TG Therapeutics Investigational Trial Site

Hradec Králové, Czechia

TG Therapeutics Investigational Trial Site

Jihlava, Czechia

TG Therapeutics Investigational Trial Site

Ostrava, Czechia

TG Therapeutics Investigational Trial Site

Pardubice, Czechia

TG Therapeutics Investigational Trial Site

Zlín, Czechia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Tbilisi, Georgia

TG Therapeutics Investigational Trial Site

Budapest, Hungary

TG Therapeutics Investigational Trial Site

Budapest, Hungary

TG Therapeutics Investigational Trial Site

Kaposvár, Hungary

TG Therapeutics Investigational Trial Site

Kistarsca, Hungary

TG Therapeutics Investigational Trial Site

Pécs, Hungary

TG Therapeutics Investigational Trial Site

Shtip, North Macedonia

TG Therapeutics Investigational Trial Site

Skopje, North Macedonia

TG Therapeutics Investigational Trial Site

Cherkasy, Ukraine

TG Therapeutics Investigational Trial Site

Ivano-Frankivsk, Ukraine

TG Therapeutics Investigational Trial Site

Ivano-Frankivsk, Ukraine

TG Therapeutics Investigational Trial Site

Ivano-Frankivsk, Ukraine

TG Therapeutics Investigational Trial Site

Kyiv, Ukraine

TG Therapeutics Investigational Trial Site

Kyiv, Ukraine

TG Therapeutics Investigational Trial Site

Lviv, Ukraine

TG Therapeutics Investigational Trial Site

Lviv, Ukraine

TG Therapeutics Investigational Trial Site

Ternopil, Ukraine

TG Therapeutics Investigational Trial Site

Vinnytsia, Ukraine

TG Therapeutics Investigational Trial Site

Vinnytsia, Ukraine

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NCT07211633


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