RecruitingPhase 3NCT07221188

A Clinical Study to Investigate the Safety and Tolerability of Efimosfermin Alfa Injection in Participants With Known or Suspected F2- or F3-stage MASH

A Phase 3, Randomized, Double-Blind, Placebo-Controlled, 3-Arm Study to Investigate the Safety and Tolerability of Efimosfermin Alfa in Participants With Known or Suspected F2- or F3-Stage Metabolic Dysfunction-Associated Steatohepatitis (MASH) (ZENITH-2)


Sponsor

GlaxoSmithKline

Enrollment

1,250 participants

Start Date

Dec 12, 2025

Study Type

INTERVENTIONAL

Summary

This study will evaluate the safety and tolerability of Efimosfermin Alfa for participants with known or suspected MASH with fibrosis consistent with stage F2 or F3.


Eligibility

Min Age: 18 YearsMax Age: 75 Years

Inclusion Criteria4

  • Able and willing to understand and sign a written informed consent form (ICF) that must be obtained prior to the initiation of study procedures
  • Age >=18 through <=75 years at enrolment
  • History or presence of 2 or more of the 5 components of metabolic syndrome per American Heart Association definition
  • History or presence of known or suspected MASH with evidence of fibrosis

Exclusion Criteria14

  • ALT or AST >=5 × upper limit of normal (ULN)
  • Total bilirubin (BILI) >=1.3 milligram per deciliter (mg/dL). Individuals with documented Gilbert's syndrome may be enrolled if they experienced an isolated increase in total BILI of >=1.3 mg/dL and direct BILI is <=20% of total BILI; otherwise, the individual will be excluded.
  • Serum albumin <=3.5 grams per deciliter (g/dL)
  • International normalized ratio (INR) >=1.3 not due to therapeutic anticoagulation. Individuals receiving chronic anticoagulant treatment with higher INR values may be enrolled at the discretion of the Investigator and Study Medical Monitor.
  • Alkaline phosphatase (ALP) >=2 × ULN
  • Platelet (PLT) count <140 000 per (/) cubic millimeter (mm\^3); individuals with a PLT count between 110,000/mm\^3 and 140,000/mm\^3 may be enrolled after discussion with the Study Medical Monitor
  • Serum creatinine >=1.5 mg/dL or creatinine clearance <=60 milliliter (mL)/minute (min)/1.73 square meter by Chronic Kidney Disease Epidemiology Collaboration equation.
  • Alpha-fetoprotein >=20 nanogram per milliliter (ng/mL)
  • HbA1c >=9.0%
  • Model for End-Stage Liver Disease (MELD) 3.0 score >=12 unless the score is elevated in the absence of liver dysfunction (eg, Gilbert's syndrome)
  • Phosphatidylethanol (PEth) >=80 nanogram per milliliter (ng/mL) at Screening
  • Known co-infection with any of the following: a. Human immunodeficiency virus; b. Hepatitis B virus; c. Hepatitis C virus (HCV); d. Hepatitis D virus; or e. Hepatitis E virus.
  • Chronic liver disease from any other cause including, but not limited to, alcoholic liver disease; evidence of portal hypertension; viral hepatitis, or any history or evidence of cirrhosis; or decompensated liver disease such as clinical ascites, bleeding gastroesophageal varices, hepatorenal syndrome, or hepatic encephalopathy prior to Screening or Day 1.
  • Current or history of excessive alcohol intake for >=3 months within the 12-month period prior to Screening

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Interventions

DRUGEfimosfermin Alfa

Efimosfermin Alfa will be administered

DRUGPlacebo

Placebo will be administered


Locations(43)

GSK Investigational Site

Arcadia, California, United States

GSK Investigational Site

Covina, California, United States

GSK Investigational Site

Los Angeles, California, United States

GSK Investigational Site

Santa Maria, California, United States

GSK Investigational Site

Cape Coral, Florida, United States

GSK Investigational Site

Doral, Florida, United States

GSK Investigational Site

Hialeah, Florida, United States

GSK Investigational Site

Inverness, Florida, United States

GSK Investigational Site

Jacksonville, Florida, United States

GSK Investigational Site

Kissimmee, Florida, United States

GSK Investigational Site

Lakeland, Florida, United States

GSK Investigational Site

Maitland, Florida, United States

GSK Investigational Site

Miami, Florida, United States

GSK Investigational Site

Miami, Florida, United States

GSK Investigational Site

Miami, Florida, United States

GSK Investigational Site

Miami, Florida, United States

GSK Investigational Site

Miami Lakes, Florida, United States

GSK Investigational Site

Ocala, Florida, United States

GSK Investigational Site

Palmetto Bay, Florida, United States

GSK Investigational Site

Topeka, Kansas, United States

GSK Investigational Site

Springfield, Missouri, United States

GSK Investigational Site

St Louis, Missouri, United States

GSK Investigational Site

Jersey City, New Jersey, United States

GSK Investigational Site

East Syracuse, New York, United States

GSK Investigational Site

New York, New York, United States

GSK Investigational Site

Morehead City, North Carolina, United States

GSK Investigational Site

Akron, Ohio, United States

GSK Investigational Site

Springboro, Ohio, United States

GSK Investigational Site

Austin, Texas, United States

GSK Investigational Site

Austin, Texas, United States

GSK Investigational Site

Brownsville, Texas, United States

GSK Investigational Site

Dallas, Texas, United States

GSK Investigational Site

DeSoto, Texas, United States

GSK Investigational Site

Richmond, Texas, United States

GSK Investigational Site

San Antonio, Texas, United States

GSK Investigational Site

San Antonio, Texas, United States

GSK Investigational Site

Seabrook, Texas, United States

GSK Investigational Site

Tomball, Texas, United States

GSK Investigational Site

Waco, Texas, United States

GSK Investigational Site

Waco, Texas, United States

GSK Investigational Site

West Jordan, Utah, United States

GSK Investigational Site

Manassas, Virginia, United States

GSK Investigational Site

Seattle, Washington, United States

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NCT07221188