RecruitingPhase 3NCT07611110

AZD2265 Compared With Standard of Care in PSMA-positive Metastatic Castration-resistant Prostate Cancer (VECTRA-01)

A Phase III, Multicentre, Randomised Controlled Study to Evaluate the Efficacy and Safety of AZD2265 (FPI-2265) ²²⁵Ac-PSMA-I&T Compared With Standard of Care in Patients With PSMA-positive Metastatic Castration-resistant Prostate Cancer (VECTRA-01)


Sponsor

AstraZeneca

Enrollment

670 participants

Start Date

May 4, 2026

Study Type

INTERVENTIONAL

Conditions

Summary

The intention of the study is to demonstrate superiority of AZD2265 relative to standard of care treatments by assessment of radiographic progression-free survival (rPFS) and overall survival (OS) in participants with mCRPC.


Eligibility

Sex: MALEMin Age: 18 Years

Inclusion Criteria12

  • ≥ 18 years of age.
  • Diagnosis of adenocarcinoma of prostate.
  • Must have had prior orchiectomy and/or ongoing ADT and a castrate level of plasma/serum testosterone.
  • Progressive mCRPC following the most recent treatment at the time of study entry, with at least 1 metastatic lesion (measurable and/or non-measurable) that is suitable for repeated assessment by CT and/or MRI and/or bone scan.
  • Previously treated with at least 2 cycles of PSMA-directed β-emitting radioconjugate.
  • Previously treated with at least 1 taxane-based chemotherapy regimen for either metastatic hormone-sensitive prostate cancer or CRPC.
  • Previously treated with at least 1 ARPI (eg, enzalutamide, abiraterone, etc.).
  • Positive PSMA PET/CT scans, obtained with PSMA ligands (⁶⁸Ga-PSMA-11 or ¹⁸F-DCFPyL).
  • ECOG performance status of 0 to 2.
  • Adequate organ and bone marrow function as described in study protocol.
  • Participants must not father children or donate sperm from signing ICF, during the study intervention and for 6 months after the last dose of study intervention.
  • Participants must use a condom from signing ICF, during study intervention, and for 6 months after the last dose of study drug, with all sexual partners.

Exclusion Criteria7

  • Prior treatment with an α-emitting molecular targeted therapeutic radioconjugate (prior treatment with radium-223 is permitted).
  • Progression on PSMA-directed β-emitting radioconjugate prior to the administration of Cycle 3.
  • Receipt of > 6 cycles of PSMA-directed β-emitting therapeutic RC.
  • History of another primary malignancy, with exceptions.
  • Persistent toxicities (CTCAE Grade ≥ 2) caused by previous anticancer therapy, with exceptions.
  • Spinal cord compression or brain metastases unless asymptomatic, stable, and not requiring steroids for at least 4 weeks prior to start of study intervention.
  • Clinically significant ECG abnormalities, with exceptions.

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Interventions

DRUGAZD2265

IV

DRUGCabazitaxel

IV in combination with oral prednisone/prednisolone

DRUGAbiraterone

Oral in combination with prednisone/prednisolone

DRUGEnzalutamide

Oral

DRUGApalutamide

Oral

DRUGDarolutamide

Oral

DRUGRezvilutamide

Oral

DRUGRadium-223

IV


Locations(90)

Research Site

Dothan, Alabama, United States

Research Site

Phoenix, Arizona, United States

Research Site

Irvine, California, United States

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Loma Linda, California, United States

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San Francisco, California, United States

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Aurora, Colorado, United States

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Miami, Florida, United States

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O'Fallon, Illinois, United States

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Metairie, Louisiana, United States

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Detroit, Michigan, United States

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Grand Rapids, Michigan, United States

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Omaha, Nebraska, United States

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Omaha, Nebraska, United States

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Albuquerque, New Mexico, United States

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New Hyde Park, New York, United States

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New York, New York, United States

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Cleveland, Ohio, United States

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Dayton, Ohio, United States

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Portland, Oregon, United States

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Pittsburgh, Pennsylvania, United States

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Myrtle Beach, South Carolina, United States

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Nashville, Tennessee, United States

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Houston, Texas, United States

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Salt Lake City, Utah, United States

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Darlinghurst, Australia

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Melbourne, Australia

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Linz, Austria

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Salzburg, Austria

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São Paulo, Brazil

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São Paulo, Brazil

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Edmonton, Alberta, Canada

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Halifax, Nova Scotia, Canada

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Hamilton, Ontario, Canada

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Toronto, Ontario, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Beijing, China

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Chengdu, China

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Chongqing, China

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Fuzhou, China

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Guangzhou, China

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Guangzhou, China

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Guangzhou, China

Research Site

Nanjing, China

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Nanjing, China

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Shanghai, China

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Shanghai, China

Research Site

Wuhan, China

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Wuhan, China

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Villejuif, France

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Berlin, Germany

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Bonn, Germany

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Dresden, Germany

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Essen, Germany

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Karlsruhe, Germany

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Münster, Germany

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Rostock, Germany

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Tübingen, Germany

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Würzburg, Germany

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Bangalore, India

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Gurgaon, India

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Gurgaon, India

Research Site

Navi Mumbai, India

Research Site

Fukuoka, Japan

Research Site

Kanazawa, Japan

Research Site

Kashiwa, Japan

Research Site

Sapporo, Japan

Research Site

Goyang-si, South Korea

Research Site

Seoul, South Korea

Research Site

Seoul, South Korea

Research Site

Barcelona, Spain

Research Site

Barcelona, Spain

Research Site

L'Hospitalet de Llobregat, Spain

Research Site

Madrid, Spain

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Málaga, Spain

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Santiago de Compostela, Spain

Research Site

Kaohsiung City, Taiwan

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Taipei, Taiwan

Research Site

Taipei, Taiwan

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Taipei, Taiwan

Research Site

Taoyuan, Taiwan

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Bangkok, Thailand

Research Site

Bangkok, Thailand

Research Site

Ankara, Turkey (Türkiye)

Research Site

Ankara, Turkey (Türkiye)

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Istanbul, Turkey (Türkiye)

Research Site

Istanbul, Turkey (Türkiye)

Research Site

London, United Kingdom

Research Site

Middlesbrough, United Kingdom

Research Site

Southampton, United Kingdom

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