RecruitingPhase 1NCT05304377

A Phase 1a/1b Study of ELVN-001 for the Treatment Chronic Myeloid Leukemia

A Phase 1a/1b Study of ELVN-001 for the Treatment of Chronic Myeloid Leukemia


Sponsor

Enliven Therapeutics

Enrollment

200 participants

Start Date

May 22, 2022

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to evaluate the safety, tolerability and determine the recommended dose for further clinical evaluation of ELVN-001 in patients with chronic myeloid leukemia with and without T315I mutations in patients who are relapsed, refractory or intolerant to TKIs.


Eligibility

Min Age: 18 Years

Inclusion Criteria5

  • BCR-ABL1 positive CML in chronic phase, with or without T315I mutation.
  • US: The patient has failed or is intolerant to at least one prior second-generation tyrosine kinase inhibitor (TKI) or asciminib. Rest of World: The patient has failed, is intolerant to, or not a candidate for, available therapies known to be active for treatment of their CML (country-specific criteria may vary).
  • ECOG performance status of 0 to 2.
  • Adequate hematologic, hepatic and renal function.
  • Prior bone marrow transplant allowed if ≥ 6 months prior to the first dose of ELVN-001.

Exclusion Criteria3

  • Treatment with anti-cancer or anti-CML therapy within 7 days or 5 half-lives, whichever is longer.
  • History of acute tyrosine kinase inhibitor (TKI)-related pancreatitis within 6 months of study entry. Active chronic pancreatitis, or pancreatic disease due to any cause.
  • QTc \>470 ms.

Interventions

DRUGELVN-001

orally once or twice daily


Locations(46)

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Montefiore Medical Center

The Bronx, New York, United States

Oregon Health & Science University-Knight Cardiovascular Institute

Portland, Oregon, United States

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Royal Adelaide Hospital

Adelaide, Australia

UZ Gent

Ghent, Belgium

UZ Leuven

Leuven, Belgium

CHU Liege

Liège, Belgium

University Health Network (UHN) - Princess Margaret Cancer Centre

Toronto, Ontario, Canada

CHU Amiens Picardie Site Sud

Amiens, France

Institut Bergonie - Centre Regional de Lutte Contre Le Cancer de Bordeaux et Sud Ouest

Bordeaux, France

Centre Hospitalier de Versailles (CHV)

Le Chesnay, France

CHRU de Lille - Hopital Calmette-Boulevard du Pr Leclercq CHRU Lille

Lille, France

Centre Hospitalier Universitaire (CHU) De Limoges Hopital Dupuytren

Limoges, France

Centre Leon Berard

Lyon, France

Centre Hospitalier Lyon Sud

Pierre-Bénite, France

Uniklinik RWTH Aachen Medizinische

Aachen, Germany

Charite Campus Virchow

Berlin, Germany

Klinikum der Goethe Universitat

Frankfurt, Germany

Universitaetsklinikum Des Saarlandes Und Medizinische Fakultaet Der Universitaet Des Saarlandes

Homburg, Germany

Universitaetsklinikum Jena

Jena, Germany

Medizinische Universitatsklinik Mannheim der Universitat Heidelberg

Mannheim, Germany

Universitaetsmedizin Rostock

Rostock, Germany

Semmelweis Egyetem, Belgyogyaszati es Onkologiai Klinika

Budapest, Hungary

Pecsi Tudomanyegyetem Klinikai Kozpont (University of Pecs, Clinical Centre)

Pécs, Hungary

Hadassah Medical Center

Jerusalem, Israel

The Galilee Medical Center

Nahariya, Israel

Rabin Medical Center

Petah Tikva, Israel

Azienda Ospedaliero Universitaria Delle Marche

Ancona, Italy

Radboud University Medical Center

Nijmegen, Netherlands

Szpital Specjalistycnzy im. Jedrzeja Sniadeckiego w Nowym Saczu

Nowy Sącz, Poland

MICS Centrum Medyczne Torun

Torun, Poland

Instytut Hematologii I Transfuzjologii

Warsaw, Poland

Chonbuk National University Hospital

Jeonju, Jeollabuk-do, South Korea

Keimyung University Dongsan Hospital

Daegu, South Korea

Uijeongbu Eulji Medical Center

Gyeonggi-do, South Korea

Chonnam National University Hwasun Hospital

Hwasun, South Korea

Samsung Medical Center

Seoul, South Korea

Hospital Del Mar

Barcelona, Spain

Hospital Universitario de Gran Canaria Dr. Negrin, Servicio Canario e Salud (SCS)

Las Palmas de Gran Canaria, Spain

Hospital Universitario La Paz

Madrid, Spain

Complejo Hospitalario de Toledo - Hospital Virgen de la Salud

Toledo, Spain

Universitat de Valencia - Hospital Universitari i Politecnic La Fe de Valencia (Hospital La Fe Bulevar Sur)

Valencia, Spain

Beatson West of Scotland Cancer Centre, Gartnavel General Hospital

Glasgow, United Kingdom

Hammersmith Hospital Imperial College Healthcare NHS Trust

London, United Kingdom

The Christie NHS Foundation Trust

Manchester, United Kingdom

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