RecruitingPhase 1NCT05800665

A Study Evaluating the Safety, Pharmacokinetics, and Activity of RO7656594 In Participants With Advanced or Metastatic Prostate Cancer

A Phase 1, Open-Label, Multicenter, Dose-Escalation and Expansion Study Evaluating the Safety, Pharmacokinetics, and Activity of RO7656594 in Patients With Advanced or Metastatic Prostate Cancer


Sponsor

Genentech, Inc.

Enrollment

210 participants

Start Date

May 2, 2023

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics, and preliminary activity of RO7656594 in participants with advanced or metastatic prostate cancer. It will also identify recommended doses and regimens for RO7656594 for subsequent studies.


Eligibility

Sex: MALEMin Age: 18 Years

Inclusion Criteria5

  • Eastern Cooperative Oncology Group (ECOG) performance status ≤1.
  • Metastatic prostate adenocarcinoma without small-cell carcinoma or neuroendocrine features.
  • Prior therapy with a second-generation androgen receptor (AR)-targeted therapy (e.g., abiraterone, enzalutamide, apalutamide, darolutamide).
  • Prior therapy with a taxane regimen or are considered ineligible for treatment with a taxane regimen or have refused treatment with a taxane regimen, unless otherwise specified.
  • For participants with a known pathogenic breast cancer gene 1 (BRCA1) or BRCA2 mutation: prior therapy with a poly (adenosine diphosphate (ADP)-ribose) polymerase (PARP) inhibitor, or are considered ineligible for treatment with a PARP inhibitor, if such therapy is approved and available.

Exclusion Criteria4

  • Treatment with any approved systemic anti-cancer therapy within 14 days or 5 drug elimination half-lives (whichever is longer, not to exceed 28 days) prior to the first study treatment.
  • Treatment with any investigational agent within 28 days prior to the first study treatment.
  • Treatment with any previous AR protein degrader.
  • Untreated central nervous system (CNS) metastases or leptomeningeal disease.

Interventions

DRUGRO7656594

RO7656594 will be administered orally at specified dose on specified days.


Locations(25)

HonorHealth

Scottsdale, Arizona, United States

Yale Cancer Center

New Haven, Connecticut, United States

Sarah Cannon Research Institute @ Florida Cancer

Orlando, Florida, United States

University of Illinois Hospital & Health Sciences System

Chicago, Illinois, United States

SCRI Oncology Partners

Nashville, Texas, United States

St Vincent's Hospital Sydney

Darlinghurst, New South Wales, Australia

Macquarie University Hospital

New South Wales, New South Wales, Australia

Monash Health Monash Medical Centre

Clayton, Victoria, Australia

Austin Hospital

Heidelberg, Victoria, Australia

British Columbia Cancer Agency

Vancouver, British Columbia, Canada

Princess Margaret Hospital

Toronto, Ontario, Canada

Centre Léon Bérard

Lyon, France

Institut Paoli Calmettes

Marseille, France

Seoul National University Hospital

Seoul, South Korea

Severance Hospital Yonsei University Health System - PPDS

Seoul, South Korea

Asan Medical Center - PPDS

Seoul, South Korea

Samsung Medical Center - PPDS

Seoul, South Korea

Clinica Universidad de Navarra

Pamplona, Navarre, Spain

Hospital Universitario Vall d'Hebron - PPDS

Barcelona, Spain

Clinica Universidad de Navarra-Madrid

Madrid, Spain

Hospital Clinico San Carlos

Madrid, Spain

Cambridge Clinical Research Centre

Cambridge, United Kingdom

Leicester Royal Infirmary

Leicester, United Kingdom

The Christie

Manchester, United Kingdom

Royal Marsden Hospital - Surrey

Sutton, United Kingdom

View Full Details on ClinicalTrials.gov

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NCT05800665


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