RecruitingPhase 2NCT06189209

Efficacy and Safety of Tenalisib in Patients With Metastatic Triple Negative Breast Cancer (TNBC)

A Phase II, Multi-center, Single-arm, Open-label Study to Assess the Efficacy and Safety of Tenalisib, a PI3K δ/γ, and SIK3 Inhibitor, in Patients With Metastatic Triple Negative Breast Cancer (TNBC)


Sponsor

Rhizen Pharmaceuticals SA

Enrollment

40 participants

Start Date

Mar 4, 2024

Study Type

INTERVENTIONAL

Summary

This is a Phase II, open-label, single-arm, study, designed to evaluate the efficacy and safety of tenalisib in patients with metastatic TNBC, who have received at least one but not more than 3 prior therapies in a metastatic setting.


Eligibility

Sex: FEMALEMin Age: 18 Years

Inclusion Criteria5

  • Patients who have histologically confirmed TNBC.
  • Patients who have received at least 1 but not more than 3 prior chemotherapy regimens in a metastatic setting.
  • Patients with at least one measurable lesion, per RECIST version 1.1 at baseline . Bone-only disease is not permitted.
  • ECOG performance status 0 to 2.
  • Adequate bone marrow, liver, and renal function

Exclusion Criteria10

  • Cancer therapy/ any cancer investigational drug within 3 weeks (21 days) or 5 half-lives (whichever is shorter).
  • Patient who has not recovered from acute toxicities of previous therapy except treatment-related alopecia.
  • Prior exposure to PI3K inhibitors (e.g., alpelisib, buparlisib) for breast cancer.
  • Major surgery within 4 weeks of starting study treatment.
  • Patient with symptomatic uncontrolled brain metastasis.
  • Ongoing immunosuppressive therapy including systemic corticosteroids.
  • History of severe cutaneous reactions.
  • Concurrent disease or condition that would interfere with study participation
  • Pregnancy or lactation.
  • Any severe and/or uncontrolled medical conditions or other conditions that could affect patient participation

Interventions

DRUGTenalisib

Tenalisib will be administered 800mg/ 400mg BID, orally


Locations(9)

HCG City Cancer Center

Vijayawada, Andhra Pradesh, India

Narayana Hrudayala Majumdar Shaw Hospital

Bangalore, Karnataka, India

Tata Memorial Centre

Mumbai, Maharashtra, India

Mumbai Oncocare Centre

Mumbai, Maharashtra, India

Sahyadri Super Speciality Hospital

Pune, Maharashtra, India

Nobel Hospital

Pune, Maharashtra, India

Meenakshi Mission Hospital & Research Center

Madurai, Tamil Nadu, India

Nizams Institute of Medical Science

Hyderabad, Telangana, India

Health Point Hospital

Kolkata, West Bengal, India

View Full Details on ClinicalTrials.gov

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NCT06189209