RecruitingPhase 1Phase 2NCT06445062

Study of RAS(ON) Inhibitors in Patients With Gastrointestinal Solid Tumors

A Platform Study of RAS(ON) Inhibitors in Patients With Gastrointestinal Solid Tumors


Sponsor

Revolution Medicines, Inc.

Enrollment

1,130 participants

Start Date

May 24, 2024

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this platform study is to evaluate the safety, tolerability, pharmacokinetics (PK), and preliminary antitumor activity of novel RAS(ON) inhibitors combined with Standard(s) of Care (SOC) or with novel agents. The current subprotocols include the following: Subprotocol A: RMC-6236 + 5-fluorouracil-based regimens Subprotocol B: RMC-6236 + cetuximab with or without mFOLFOX6 Subprotocol C: RMC-6236 + gemcitabine + nab-paclitaxel Subprotocol D: RMC-9805 with or without RMC-6236 + 5-fluorouracil-based regimens Subprotocol E: RMC-9805 with or without RMC-6236 + cetuximab with or without mFOLFOX6 Subprotocol F: RMC-9805 with or without RMC-6236 + gemcitabine + nab-paclitaxel


Eligibility

Min Age: 18 Years

Inclusion Criteria6

  • All Patients (unless otherwise noted):
  • ≥ 18 years of age
  • ECOG PS is 0 to 1
  • Adequate organ function as outlined by the study
  • Pathologically or cytologically documented pancreatic carcinoma or poorly differentiated pancreatic carcinoma with metastatic disease or RAS-mutated, histologically or cytologically confirmed colorectal adenocarcinoma with documented unresectable or metastatic disease (Subprotocol A, B, and C)
  • Presence of RAS G12D mutation (Subprotocol D, E, F)

Exclusion Criteria4

  • All Patients:
  • Primary central nervous system (CNS) tumors
  • Impaired gastrointestinal (GI) function that may significantly alter the absorption of RMC drugs
  • Major surgery within 28 days of first dose

Interventions

DRUGRMC-6236

Oral tablet

DRUGmFOLFOX6 regimen

IV infusion

DRUGbevacizumab

IV infusion

DRUGmFOLFIRINOX regimen

IV infusion

DRUGcetuximab

IV infusion

DRUGgemcitabine

IV infusion

DRUGnab-paclitaxel

IV infusion

DRUGRMC-9805

Oral Tablet


Locations(32)

Ironwood Cancer and Research Centers

Chandler, Arizona, United States

Mayo Clinic Hospital

Phoenix, Arizona, United States

HonorHealth Research Institute

Scottsdale, Arizona, United States

UC San Diego Moores Cancer Center

La Jolla, California, United States

Cedars-Sinai Cancer at Cedars-Sinai Medical Center

Los Angeles, California, United States

UCLA Hematology/Oncology- Santa Monica

Los Angeles, California, United States

University of Colorado Hospital-Anschutz Cancer Pavilion

Aurora, Colorado, United States

Yale-New Haven Hospital-Yale Cancer Center

New Haven, Connecticut, United States

Mayo Clinic Cancer Center

Jacksonville, Florida, United States

Moffitt Cancer Center

Tampa, Florida, United States

The University of Kansas Clinical Research Center

Westwood, Kansas, United States

The Sidney Kimmel Comprehensive Cancer Center at John Hopkins

Baltimore, Maryland, United States

Massachusetts General Hospital

Boston, Massachusetts, United States

Dana Farber Cancer Institute

Boston, Massachusetts, United States

Mayo Clinic

Rochester, Minnesota, United States

Nebraska Cancer Specialists

Omaha, Nebraska, United States

University of Nebraska Medical Center

Omaha, Nebraska, United States

Atlantic Health System

Morristown, New Jersey, United States

Northwell Health / RJ Zuckerberg Cancer Center

Lake Success, New York, United States

Columbia University Medical Center

New York, New York, United States

Memorial Sloan Kettering Cancer Center Main Campus

New York, New York, United States

Duke University Medical Center

Durham, North Carolina, United States

University of Cincinnati Medical Center

Cincinnati, Ohio, United States

Stephenson Cancer Center

Oklahoma City, Oklahoma, United States

Hospital of the University of Pennsylvania

Philadelphia, Pennsylvania, United States

SCRI Oncology Partners

Nashville, Tennessee, United States

Baylor College of Medicine

Houston, Texas, United States

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States

NEXT Oncology Dallas

Irving, Texas, United States

Huntsman Cancer Institute, University of Utah

Salt Lake City, Utah, United States

Virginia Cancer Specialists

Fairfax, Virginia, United States

Fred Hutchinson Cancer Center

Seattle, Washington, United States

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NCT06445062


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