RecruitingPhase 3NCT06757634

Phase 3 Study of Gedatolisib as First-Line Treatment for Patients With HR-Positive, HER2-Negative Advanced Breast Cancer (VIKTORIA-2)

VIKTORIA-2: A Randomized, Open-Label, Phase 3 Study of Fulvestrant and CDK4/6 Inhibitors With or Without Gedatolisib as First-Line Treatment in Patients With HR-Positive and HER2-Negative Advanced Breast Cancer


Sponsor

Celcuity Inc

Enrollment

674 participants

Start Date

Jul 24, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This is a Phase 3, open-label, randomized, clinical trial evaluating the efficacy and safety of gedatolisib plus fulvestrant and CDK4/6 Inhibitors for the treatment of patients with locally advanced or metastatic HR+/HER2- advanced breast cancer.


Eligibility

Min Age: 18 Years

Inclusion Criteria13

  • Histologically or cytologically confirmed diagnosis of metastatic or locally advanced HR+/HER2- breast cancer
  • Adult females, pre- and/or post-menopausal, and adult males. Pre-menopausal (and peri-menopausal) women can be enrolled if amenable to treatment with an LHRH agonist. Patients are to have commenced concomitant treatment with LHRH agonist prior to or on Cycle 1, Day 1 and must be willing to continue for the duration of the study.
  • Negative pregnancy test for females of childbearing potential. Female subjects who are not surgically sterile must use a medically effective contraceptive method from screening until 2 years after the last dose of study treatment.
  • Progression of disease during or within 12 months of completing (neo)adjuvant ET.
  • Adequate archival, fresh tumor tissue, or liquid biopsy for the analysis of PIK3CA mutational status.
  • Permitted prior therapies:
  • (neo)adjuvant fulvestrant or any selective ER degrader only if the treatment duration \< 6 months
  • (neo)adjuvant chemotherapy
  • (neo)adjuvant CDK4/6 inhibitor, unless PD was on or within 6 months of discontinuation of CDK4/6i
  • Subject has radiologically measurable disease according to RECIST v1.1, per local assessment. Patients with evaluable bone-only disease are not eligible. Patients with bone-only disease that has lytic or mixed lytic/blastic lesions and at least one measurable soft tissue component per RECIST v1.1 may be eligible.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0-2.
  • Life expectancy of at least \>6 months.
  • Adequate bone marrow, hepatic, renal and coagulation function.

Exclusion Criteria7

  • Concurrent malignancies other than adequately treated non-melanoma skin cancer. Previous malignancies in remission but curatively treated with no evidence of disease progression and judged by local Investigator to be at low risk of impacting health or survival while on study.
  • Prior treatment with a phosphoinositide 3-kinase (PI3K) inhibitor, a protein kinase B (Akt) inhibitor, or a mechanistic target of rapamycin (mTOR) inhibitor
  • Prior treatment with systemic anticancer therapy for ABC
  • Subjects with type 1 diabetes
  • Known and untreated, or active, brain or leptomeningeal metastases
  • History of clinically significant cardiovascular abnormalities
  • History of drug-induced symptomatic interstitial lung disease (pneumonitis) or hepatitis

Interventions

DRUGArm A: Gedatolisib + Palbociclib or Ribociclib + Fulvestrant

Drug: Gedatolisib Participants will receive intravenous (IV) gedatolisib once weekly for 3 weeks (Days 1, 8, 15) followed by 1 week off Other Names: • PF-05212384 Drug: Palbociclib Participants will receive oral palbociclib on days 1-21 of each 28-day cycle. Other Names: • IBRANCE Drug: Ribociclib Participants will receive oral ribociclib on Days 1-21 of each 28-day cycle Other Names: • KISQALI® Drug: Fulvestrant Participants will receive intramuscular (IM) fulvestrant every 2 weeks during Cycle 1 and then every 4 weeks Other Names: • Faslodex

DRUGArm B: Palbociclib or Ribociclib + Fulvestrant

Drug: Palbociclib Participants will receive oral palbociclib on Days 1-21 of each 28-day cycle Other Names: • IBRANCE Drug: Ribociclib Participants will receive oral ribociclib on Days 1-21 of each 28-day cycle Other Names: • KISQALI® Drug: Fulvestrant Participants will receive intramuscular (IM) fulvestrant approximately every 2 weeks during Cycle 1 then approximately every 4 Other Names: • Faslodex


Locations(203)

City of Hope Medical Center

Duarte, California, United States

Providence Medical Foundation

Fullerton, California, United States

UCLA Hematology Oncology Santa Monica

Los Angeles, California, United States

BRCR Medical Center, Inc- Internal Medicine

Plantation, Florida, United States

BRCR Medical Center, INC

Tamarac, Florida, United States

The University of Kansas Cancer Center

Westwood, Kansas, United States

Mercy Health-Paducah Cancer Center

Paducah, Kentucky, United States

American Oncology Partners, P.A.

Bethesda, Maryland, United States

Massachusetts General Hospital Cancer Center

Boston, Massachusetts, United States

Henry Ford Health System

Detroit, Michigan, United States

Saint Luke's Cancer Institute

Kansas City, Missouri, United States

Washington University School of Medicine in Saint Louis

St Louis, Missouri, United States

SCL Health - Cancer Centers of Montana

Billings, Montana, United States

Weill Cornell Medical College - NewYork-Presbyterian Hospital

New York, New York, United States

Clinical Research Alliance, Inc.

Westbury, New York, United States

Stefanie Spielman Comprehensive Breast Center at Olentangy River Road

Columbus, Ohio, United States

Rittenhouse Hematology/Oncology

Philadelphia, Pennsylvania, United States

Sanford Health

Sioux Falls, South Dakota, United States

University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Mays Cancer Center

San Antonio, Texas, United States

Bon Secours St. Francis Medical Oncology Center

Midlothian, Virginia, United States

Fred Hutchinson Cancer Center

Seattle, Washington, United States

Centro de Oncologia e Investigacion Buenos Aires COIBA

Buenos Aires, Argentina

Pergamino Clinic

Buenos Aires, Argentina

CENIT Foundation

Buenos Aires, Argentina

Fleischer Medical Center (Centro Medico Fleischer)

Buenos Aires, Argentina

Fundacion Respirar

Buenos Aires, Argentina

Centro Oncológico Korben

Buenos Aires, Argentina

Alexander Fleming Institute

Buenos Aires, Argentina

Center for Medical Education and Clinical Research (CEMIC)

Buenos Aires, Argentina

Cordoba Oncology Institute (IONC)

Córdoba, Argentina

Centro Oncologico de Excelencia

La Plata, Argentina

Fundación CORI

La Rioja, Argentina

Center of Nuclear and Molecular Medicine of Entre Rios (CEMENER)

Paraná, Argentina

Rosario's Oncology Institute and Medical Specialities (IOR)

Rosario, Argentina

GenesisCare - St Andrews

Adelaide, Australia

Breast Cancer Research Centre

Nedlands, Australia

Icon Cancer Centre Southport

Southport, Australia

Sydney Adventist Hospital

Wahroonga, Australia

Westmead Hospital

Westmead, Australia

The Queen Elizabeth Hospital

Woodville, Australia

Cliniques Universitaires Saint-Luc

Brussels, Belgium

Grand Hopital De Charleroi

Charleroi, Belgium

Universitair Ziekenhuis Gent - Medische Oncologie

Ghent, Belgium

Jessa Ziekenhuis - Campus Virga Jesse - Medische Oncologie

Hasselt, Belgium

Universitaire Ziekenhuizen Leuven - Campus Gasthuisberg

Leuven, Belgium

CTO Centro de Tratamento Oncológico

Belém, Brazil

Oncocentro Belo Horizonte

Belo Horizonte, Brazil

Centro Regional Integrado de Oncologia - CRIO

Fortaleza, Brazil

Pronutrir Oncologia e Nutrição

Fortaleza, Brazil

ONCOSITE - Centro de Pesquisa Clinica em Oncologia LTDA

Ijuí, Brazil

Catarina Pesquisa Clinica

Itajaí, Brazil

Hospital Sao Lucas da PUCRS

Porto Alegre, Brazil

Hospital Das Clinicas da Faculdade de Medicina de Ribeirão Preto - USP

Ribeirão Preto, Brazil

Bahia Oncology Center

Salvador, Brazil

Hospital A.C.Camargo

São Paulo, Brazil

Instituto D'or de Pesquisa e Ensino - ONCO STAR

São Paulo, Brazil

Complex Oncology Center - Burgas

Burgas, Bulgaria

Multi-profile Hospital For Active Treatment-Uni Hospital Ltd.

Panagyurishte, Bulgaria

Complex Oncological Centre Ruse

Rousse, Bulgaria

MHAT Nadezhda - Medical Oncology Clinic

Sofia, Bulgaria

MHAT "Serdika" EOOD, Base 2 - Second Department of Medical Oncology

Sofia, Bulgaria

USHAT of Oncology

Sofia, Bulgaria

Masarykuv onkologicky ustav - Oddeleni klinickych hodnoceni

Brno, Czechia

Multiscan s.r.o. - Ambulance klinicke onkologie se stacionarem

Hořovice, Czechia

FN Hradec Kralove - Klinika onkologie a radioterap

Hradec Králové, Czechia

Fakultni nemocnice Olomouc - Onkologicka klinika

Olomouc, Czechia

FN Kralovske Vinohrady - Radioterapeuticka a onkologicka klinika

Prague, Czechia

Fakultni Thomayerova Nemocnice - Onkologicka klinika

Prague, Czechia

Fakultni Nemocnice v Motole

Prague, Czechia

Centre Hospitalier Universitaire D'Amiens (Hopital Sud) - Oncologie Medicale - Cancerolo

Amiens, France

Centre Georges François Baclesse

Caen, France

Centre Georges Francois Leclerc - service d'oncologie médicale

Dijon, France

Clinique Victor Hugo / Centre Jean Bernard

Le Mans, France

CHU La Timone

Marseille, France

Centre Hospitalier Lyon Sud

Pierre-Bénite, France

Centre Hospitalier Universitaire de Poitiers - Médico-Chirurgical De Cardiol

Poitiers, France

Centre de Lutte Contre le Cancer (CLCC) - Institut de Cancerologie de l'Ouest (ICO) - Rene Gauducheau - Oncology

Saint-Herblain, France

Institut Gustave Roussy

Villejuif, France

Universitätsklinikum Düsseldorf - Gynecology

Düsseldorf, Germany

Universitätsmedizin Johannes Gutenberg

Mainz, Germany

CaritasKlinikum Saarbrücken St. Theresia

Saarbrücken, Germany

Helios Klinikum Wuppertal

Wuppertal, Germany

Areteio Hospital

Athens, Greece

University General Hospital of Heraklion

Heraklion, Greece

Iaso Thessalia General Clinic Private Obstetrics S.A.

Larissa, Greece

General University Hospital Of Larissa

Larissa, Greece

Metropolitan Hospital

Piraeus, Greece

Athens Medical Center S.A.

Thessaloniki, Greece

Theageneio Cancer Hospital

Thessaloniki, Greece

Debreceni Egyetem Klinikai Központ Nagyerdei Campus - Onkológiai Klinika

Debrecen, Hungary

Gyor-Moson-Sopron Varmegyei Petz Aladar Egyetemi Oktatokorhaz

Győr, Hungary

Békés Megyei Központi Kórház Pándy Kálmán Tagkórház - Oncology

Gyula, Hungary

Bacs-Kiskun Varmegyei Oktatakorhaz

Kecskemét, Hungary

University of Pecs- Oncology Dept.

Pécs, Hungary

Tolna Varmegyei Balassa Janos Korhaz

Szekszárd, Hungary

Presidio Ospedaliero S. Croce - Oncologia

Fano, Italy

IRCCS Ospedale Policlinico San Martino - Clinica di Oncologia Medica

Genova, Italy

IRST IRCCS - Oncologia Medica

Meldola, Italy

IEO - Istituto Europeo di Oncologia, IRCCS

Milan, Italy

Istituto Clinico Humanitas

Milan, Italy

AOU di Modena, Policlinico di Modena - Attività Integrata di Oncologia ed Ematologia

Modena, Italy

Istituto Nazionale dei Tumori - Fondazione Pascale, IRCCS

Napoli, Italy

Ospedale Maggiore, AOU Parma

Parma, Italy

IRCCS Policlinico San Matteo, Università degli studi di Pavia

Pavia, Italy

Ospedale "Santa Maria delle Croci" di Ravenna - Oncologia

Ravenna, Italy

Fondazione Policlinico Universitario Campus Bio-Medico

Roma, Italy

Umberto I Policlinico di Roma, Università La Sapienza

Roma, Italy

Istituto Clinico Humanitas

Rozzano, Italy

Azienda Ospedaliera Santa Maria di Terni

Terni, Italy

Borgo Trento, Ospedale Civile Maggiore, AOU Integrata Verona

Verona, Italy

Penang Adventist Hospital

George Town, Malaysia

Hospital Universiti Sains Malaysia

Kota Bharu, Malaysia

Hospital Kuala Lumpur - Surgery

Kuala Lumpur, Malaysia

Pantai Hospital Kuala Lumpur

Kuala Lumpur, Malaysia

Hospital Umum Sarawak

Kuching, Malaysia

Beacon Hospital

Petaling Jaya, Malaysia

National Cancer Institute - Radiotherapy and Oncology

Putrajaya, Malaysia

San Peregrino Unidad de Investigacion

Aguascalientes, Mexico

Office of Emanuel de la Mora Jimenez, MD/equiv

Guadalajara, Mexico

Clinical Research Center Chapultepec Mexico City

Mexico City, Mexico

Centro de Atencion Oncologica Viva

Mexico City, Mexico

Avix Clinical Research

Monterrey, Mexico

Filios High Medicine

Monterrey, Mexico

Administrative Society of Health Services, SC

Morelia, Mexico

Centrum Onkologii im. prof. F. Lukaszczyka - Ambulatorium Chemioterapii

Bydgoszcz, Poland

Przychodnia Lekarska KOMED

Konin, Poland

Pratia MCM Kraków

Krakow, Poland

Instytut Medyczny Santa Familia

Lodz, Poland

SP ZOZ Opolskie Centrum Onkologii - Oddzial Onkologii Klinicznej z Odcinkiem Dziennym

Opole, Poland

Zachodniopomorskie Centrum Onkologii - Osrodek Innowacyjnosci, Rozwoju i Badan Klinicznych

Szczecin, Poland

LUX MED Onkologia Sp. z o.o., Szpital Szamocka - Oddzial Onkologii Klinicznej/Chemioterapii

Warsaw, Poland

Narodowy Instytut Onkologii im. Marii SkÅ'odowskiej-Curie â€" PaÅ"stwowy Instytut Badawczy - Klinika Nowotworow Piersi i Chirurg

Warsaw, Poland

Centro Hospitalar e Universitário de Coimbra

Coimbra, Portugal

Instituto Portugues de Oncologia de Lisboa Francisco Gentil - Oncologia Medica

Lisbon, Portugal

Hospital da Luz de Lisboa - Learning Health

Lisbon, Portugal

H. de Santa Maria. Centro Hospitalar Lisboa Norte - Oncologia

Lisbon, Portugal

Hospital CUF Descobertas

Lisbon, Portugal

Centro Hospitalar Universitario do Porto - H. Santo Antonio

Porto, Portugal

Centrul de Oncologie Sf Nectarie - Medical Oncology

Baia Mare, Romania

Oncopremium Team - Medical Oncology

Baia Mare, Romania

Institutul Oncologic Prof Dr Ion Chiricuta Cluj-Napoca

Bucharest, Romania

Institutul Oncologic Prof Dr Alexandru Trestioreanu Bucuresti

Cluj-Napoca, Romania

Onco Clinic Consult

Craiova, Romania

Radiotherapy Center Cluj

Floreşti, Romania

Centrul de Oncologie Euroclinic

Iași, Romania

Institutul Regional de Oncologie Iasi - Medical Oncology

Iași, Romania

National Cancer Center - Breast Cancer

Goyang, South Korea

Gachon University Gil Medical Center - Oncology

Incheon, South Korea

CHA Bundang Medical Center - Oncology

Seongnam-si, South Korea

Korea University Anam Hospital - Gastroenterological Surgery

Seoul, South Korea

Seoul National University Hospital

Seoul, South Korea

Yonsei University Health System, Severance hospital

Seoul, South Korea

Asan Medical Center - Oncology

Seoul, South Korea

Gangnam Severance Hospital

Seoul, South Korea

Samsung Medical Center - Hematology & Oncology

Seoul, South Korea

Korea University Guro Hospital

Seoul, South Korea

The Catholic University of Korea, Seoul St. Mary's Hospital - Hematology and Oncology

Seoul, South Korea

Ajou University Hospital - Hematology/Oncology

Suwon, South Korea

Ulsan University Hospital

Ulsan, South Korea

Complexo Hospitalario Universitario A Coruña

A Coruña, Spain

Hospital Universitario de Badajoz

Badajoz, Spain

Hospital Del Mar

Barcelona, Spain

Hospital Clinic De Barcelona

Barcelona, Spain

Caceres Hospital Complex - San Pedro de Alcantara General Hospital

Cáceres, Spain

Hospital Clínico Universitario Virgen De La Arrixaca

El Palmar, Spain

Institut Catala D'oncologia

L'Hospitalet de Llobregat, Spain

H.U Arnau De Vilanova Lleida

Lleida, Spain

Hospital Beata Maria Ana de Jesus

Madrid, Spain

Hospital Universitario Ramon y Cajal - Oncología Médica

Madrid, Spain

Hospital Universitario Fundacion Jimenez Diaz

Madrid, Spain

Complejo Hospitalario Universitario De Santiago

Santiago de Compostela, Spain

Fundacion Instituto Valenciano de Oncologia

Valencia, Spain

Changhua Christian Medical Foundation - Changhua Christian Hospital - Neurology

Changhua, Taiwan

National Taiwan University Hospital - Yunlin Branch - Oncology

Douliu, Taiwan

Kaohsiung Medical University - Chung-Ho Memorial Hospital - Breast Surgery

Kaohsiung City, Taiwan

China Medical University Hospital - Breast Surgery

Taichung, Taiwan

Taichung Veterans General Hospital - General Surgery

Taichung, Taiwan

National Cheng Kung University Hospital - Gynecology/Obstetrics

Tainan, Taiwan

Chi Mei Medical Center - YongKang - Oncology and Hematology

Tainan, Taiwan

National Taiwan University Hospital - Oncology

Taipei, Taiwan

Taipei Medical University - Shuang Ho Hospital Ministry of Health and Welfare - Nephrology

Taipei, Taiwan

Taipei Veterans General Hospital - Hematology

Taipei, Taiwan

Taipei Municipal Wanfang Hospital - Managed by Taipei Medical University - Hematology and Oncology

Taipei, Taiwan

King Chulalongkorn Memorial Hospital [Medical Oncology]

Bangkok, Thailand

Rajavithi Hospital

Bangkok, Thailand

Siriraj Hospital - Medical Oncology

Bangkok, Thailand

Prince of Songkla University - Internal Medicine

Hat Yai, Thailand

Banphaeo General Hospital

Samut Sakhon, Thailand

Adana Baskent Practice and Research Hospital - Oncology

Adana, Turkey (Türkiye)

Gulhane Training and Research Hospital - Medical Oncology

Ankara, Turkey (Türkiye)

Hacettepe University Medical Faculty - Hematology

Ankara, Turkey (Türkiye)

Dr Abdurrahman Yurtaslan Training and Research Hospital - Medical Oncology

Ankara, Turkey (Türkiye)

Memorial Ankara Hastanesi

Ankara, Turkey (Türkiye)

Ankara University Medical Faculty - Oncology

Ankara, Turkey (Türkiye)

Dicle University Medical Faculty Hospital Medical Oncology

Diyarbakır, Turkey (Türkiye)

Trakya University Medical Faculty - Oncology

Edirne, Turkey (Türkiye)

Medical Park Hastaneler Grubu - I.A.U. VM Medical Park Florya

Istanbul, Turkey (Türkiye)

Medipol Mega Hospital - Medical Oncology

Istanbul, Turkey (Türkiye)

Istanbul Goztepe Prof. Dr. Suleyman Yalcin City Hospital - Medical Oncology

Istanbul, Turkey (Türkiye)

Kocaeli Uni Egt ve Uyg Hast

İzmit, Turkey (Türkiye)

Necmettin Erbakan University Meram Medical Faculty - Oncology

Konya, Turkey (Türkiye)

VM Medical Park Mersin Hastanesi

Mezitli, Turkey (Türkiye)

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NCT06757634


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