RecruitingPhase 1Phase 2NCT06850922

A Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Efficacy of RO7446603 Administered Alone or in Combination With Aflibercept or Faricimab in Participants With Diabetic Macular Edema

A Phase I/II Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Efficacy of RO7446603 Administered Alone or in Combination With Aflibercept or Faricimab in Patients With Diabetic Macular Edema


Sponsor

Genentech, Inc.

Enrollment

546 participants

Start Date

Jun 22, 2022

Study Type

INTERVENTIONAL

Conditions

Summary

This study aims to evaluate the ocular and systemic safety, tolerability and efficacy of RO7446603 in participants with diabetic macular edema (DME). The study consists of 2 segments: Phase I (Parts 1-4) and Phase II (Part 5). Phase I investigated the safety of RO7446603 following a single and multiple intravitreal (IVT) doses as monotherapy or co-administered with IVT aflibercept or IVT faricimab (in separate injections). Phase II will investigate the safety, tolerability, pharmacokinetics (PK) and efficacy of two dose levels of RO7446603 in combination with faricimab, with the two drugs co-mixed and administered as a single IVT injection, compared to faricimab alone. The first participant was enrolled in the Phase I segment on June 22, 2022. Phase I has been completed.


Eligibility

Min Age: 18 Years

Inclusion Criteria3

  • Documented diagnosis of diabetes mellitus (DM) (Type 1 or Type 2) with glycated hemoglobin (HbA1c) \< 12%
  • Macular thickening secondary to DME involving the center of the fovea \> 325 microns
  • Decreased VA attributable primarily to DME between 25 and 73 ETDRS letters

Exclusion Criteria8

  • Currently untreated DM or previously untreated participants who initiated oral anti-diabetic medication or insulin within 90 days prior to Day 1
  • Uncontrolled blood pressure (BP)
  • Pregnancy or breastfeeding, or intention to become pregnant during the study
  • For Parts 1-4: IVT anti-VEGF treatment within 90 days prior to Day 1; For Part 5: IVT anti-VEGF treatment within 120 days prior to Day 1 or IVT anti-VEGF treatment prior to Day 1 for treatment naïve participants
  • Treatment with SUSVIMOTM (ranibizumab injection) prior to Day 1
  • Any IVT or periocular (sub-tenons) corticosteroid treatment within 6 months prior to Day 1
  • Any current or history of ocular disease other than DME that may confound assessment of the macula or affect central vision
  • Proliferative diabetic retinopathy (PDR) in the study eye

Interested in this trial?

Get notified about updates and connect with the research team.

Interventions

DRUGRO7446603

Participants will receive RO7446603 as an IVT injection per the schedule described in the treatment arms.

DRUGAflibercept

Participants will receive aflibercept as an IVT injection per the schedule described in the treatment arm.

DRUGFaricimab

Participants will receive faricimab as an IVT injection per the schedule described in the treatment arms.


Locations(78)

Barnet Dulaney Perkins Eye Center

Phoenix, Arizona, United States

Arizona Retina and Vitreous Consultants

Phoenix, Arizona, United States

Associated Retinal Consultants PC

Phoenix, Arizona, United States

Retinal Research Institute, LLC

Phoenix, Arizona, United States

Retinal Diagnostic Center

Campbell, California, United States

The Retina Partners

Encino, California, United States

Retina Consultants of Orange County

Fullerton, California, United States

Retinal Consultants Medical Group

Modesto, California, United States

Northern California Retina-Vitreous Associates

Mountain View, California, United States

Retinal Consultants Medical Group

Sacramento, California, United States

University of California San Francisco

San Francisco, California, United States

Macula Retina Vitreous Research Institute

Torrance, California, United States

University of Colorado - Eye Center - PPDS

Aurora, Colorado, United States

Retina Consultants of Southern Colorado PC

Colorado Springs, Colorado, United States

Retina Specialists of Colorado

Denver, Colorado, United States

Advanced Vision Research Institute

Longmont, Colorado, United States

Retina Group of New England

Waterford, Connecticut, United States

Blue Ocean Clinical Research

Clearwater, Florida, United States

National Ophthalmic Research Institute

Fort Myers, Florida, United States

Florida Retina Institute

Jacksonville, Florida, United States

Retina Associates of Florida;Retina Associates of Florida

Tampa, Florida, United States

Southeast Retina Center

Augusta, Georgia, United States

Georgia Retina PC

Marietta, Georgia, United States

Retina Consultants of Hawaii

‘Aiea, Hawaii, United States

Illinois Eye and Ear Infirmary

Chicago, Illinois, United States

University Retina and Macula Associates, PC

Oak Forest, Illinois, United States

Raj K. Maturi, MD PC

Indianapolis, Indiana, United States

The Retina Care Center

Baltimore, Maryland, United States

Johns Hopkins Hospital

Baltimore, Maryland, United States

Retina Group of Washington

Chevy Chase, Maryland, United States

Cumberland Valley Retina Consultants

Hagerstown, Maryland, United States

Chesapeake Retina Centers - Waldorf

Waldorf, Maryland, United States

Associated Retinal Consultants - Royal Oak

Royal Oak, Michigan, United States

Retina Consultants Minnesota

Saint Louis Park, Minnesota, United States

Long Island Vitreoretinal Consultants;Opthalmology

Hauppauge, New York, United States

Retina Vitreous Surgeons of CNY PC

Liverpool, New York, United States

Opthalmic Consultants of LI

Lynbrook, New York, United States

Western Carolina Retinal Associate PA

Asheville, North Carolina, United States

North Carolina Retina Associates

Cary, North Carolina, United States

Duke University Medical Center

Durham, North Carolina, United States

Graystone Eye

Hickory, North Carolina, United States

North Carolina (NC) Retina Associates - Wake Forest Office

Wake Forest, North Carolina, United States

Piedmont Retina Specialists

Winston-Salem, North Carolina, United States

Cincinnati Eye Institute

Blue Ash, Ohio, United States

University Hospitals Cleveland Medical Center

Cleveland, Ohio, United States

Ohio State Eye and Ear Institute

Columbus, Ohio, United States

Tulsa Retina Consultants

Tulsa, Oklahoma, United States

Cascade Medical Research Institute LLC

Springfield, Oregon, United States

Erie Retina Research

Erie, Pennsylvania, United States

Wills Eye Hospital

Philadelphia, Pennsylvania, United States

Sewickely Eye Group

Sewickley, Pennsylvania, United States

Palmetto Retina Center

West Columbia, South Carolina, United States

Charles Retina Institute

Germantown, Tennessee, United States

Retina Research Institute of Texas

Abilene, Texas, United States

Texas Retina Associates

Arlington, Texas, United States

Austin Retina Associates

Austin, Texas, United States

Austin Clinical Research LLC

Austin, Texas, United States

Retina & Vitreous of Texas

Bellaire, Texas, United States

Texas Retina Associates

Dallas, Texas, United States

Valley Retina Institute P.A.

McAllen, Texas, United States

Medical Center Ophthalmology Associates

San Antonio, Texas, United States

Retina Consultants of Texas - San Antonio

San Antonio, Texas, United States

Brown Retina Institute

San Antonio, Texas, United States

Retina Consultants of Texas

The Woodlands, Texas, United States

Strategic Clinical Research Group, LLC

Willow Park, Texas, United States

Retina Associates of Utah, PLLC;Clinical Research

Salt Lake City, Utah, United States

Piedmont Eye Center

Lynchburg, Virginia, United States

Wagner Kapoor Institute

Norfolk, Virginia, United States

Virginia Eye Institute - Richmond - 7301 Forest Ave

Richmond, Virginia, United States

Retina Institute of Virginia

Richmond, Virginia, United States

Spokane Eye Clinical Research

Spokane, Washington, United States

Beijing Tongren Hospital, Capital Medical University

Beijing, Beijing Municipality, China

Tianjin Medical University Eye Hospital

Tianjin, Tianjin Municipality, China

Eye Hospital,WMU(Zhejiang Eye Hospital)

Wenzhou, Zhejiang, China

Beijing Hospital

Beijing, China

Peking Union Medical College Hospital

Beijing, China

Shanghai General Hospital - North Campus

Shanghai, China

Emanuelli Research and Development Center LLC

Arecibo, Puerto Rico

View Full Details on ClinicalTrials.gov

For the most up-to-date information, visit the official listing.

Visit

NCT06850922


Related Trials