RecruitingPhase 3NCT06881784

Study of Daraxonrasib (RMC-6236) in Patients With RAS Mutated NSCLC (RASolve 301)

RASolve 301: Phase 3 Multicenter, Open Label, Randomized Study of RMC-6236 Versus Docetaxel in Patients With Previously Treated Locally Advanced or Metastatic RAS[MUT] NSCLC


Sponsor

Revolution Medicines, Inc.

Enrollment

420 participants

Start Date

May 6, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to evaluate the safety and efficacy of a novel RAS(ON) inhibitor compared to docetaxel.


Eligibility

Min Age: 18 Years

Inclusion Criteria8

  • At least 18 years old and has provided informed consent.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  • Pathologically confirmed NSCLC, either locally advanced or metastatic, not amenable to curative surgery or radiotherapy.
  • Measurable disease per RECIST v1.1.
  • Adequate organ function (bone marrow, liver, kidney, coagulation).
  • One to two prior lines of therapy including an anti-PD-1/anti-PD(L)-1 agent and platinum-based chemotherapy.
  • Documented RAS mutation status, defined as Nonsynonymous mutations in KRAS, NRAS, or HRAS at codons 12, 13, or 61 (G12, G13, or Q61).
  • Able to take oral medications.

Exclusion Criteria5

  • Prior therapy with direct RAS-targeted therapy or docetaxel.
  • Untreated central nervous system (CNS) metastases.
  • Medically significant comorbidities (significant cardiovascular disease, lung disease, or impaired GI function).
  • Ongoing anticancer therapy.
  • Pregnant or breastfeeding.

Interventions

DRUGdaraxonrasib

oral tablets

DRUGdocetaxel

intravenous (IV) infusion


Locations(129)

Alabama Oncology

Birmingham, Alabama, United States

MemorialCare Long Beach Medical Center

Long Beach, California, United States

Yale University, Smillow Cancer Center

New Haven, Connecticut, United States

Florida Cancer Specialists & Research Institute - South

Fort Myers, Florida, United States

BRCR Global

Plantation, Florida, United States

Cancer Care Centers of Breevard

Rockledge, Florida, United States

Florida Cancer Specialists & Research Institute - North

St. Petersburg, Florida, United States

Cleveland Clinic Martin North

Stuart, Florida, United States

Florida Cancer Specialists & Research Institute - East

West Palm Beach, Florida, United States

University Cancer and Blood Center

Athens, Georgia, United States

Center for Care and Discovery

Chicago, Illinois, United States

The University of Kansas Cancer Center

Westwood, Kansas, United States

Johns Hopkins University of Medicine

Baltimore, Maryland, United States

Karmanos Cancer Institute

Detroit, Michigan, United States

Henry Ford Health

Detroit, Michigan, United States

Washington University School of Medicine - Siteman Cancer Center

St Louis, Missouri, United States

St. Vincent Frontier Cancer Center

Billings, Montana, United States

Dartmouth-Hitchcock Medical Center

Lebanon, New Hampshire, United States

Morristown Medical Center (MMCORC)

Morristown, New Jersey, United States

Roswell Park Cancer Institute

Buffalo, New York, United States

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Montefiore Medical Center

The Bronx, New York, United States

UNC Lineberger Comprehensive Cancer Center at University of North Carolina

Chapel Hill, North Carolina, United States

TriHealth Cancer & Blood Institute Research

Cincinnati, Ohio, United States

Taylor Cancer Research Center

Maumee, Ohio, United States

Oncology Associates of Oregon PC

Eugene, Oregon, United States

Avera Cancer Institute

Sioux Falls, South Dakota, United States

SCRI Oncology Partners - Tennessee

Nashville, Tennessee, United States

Texas Oncology - South Austin

Austin, Texas, United States

Texas Oncology Dallas

Dallas, Texas, United States

MD Anderson Cancer Center

Houston, Texas, United States

Texas Oncology - Gulf Coast

The Woodlands, Texas, United States

Utah Cancer Specialists

Salt Lake City, Utah, United States

Virginia Cancer Specialists

Fairfax, Virginia, United States

Blacktown Medical Oncology Research

Blacktown, New South Wales, Australia

Chris O'Brien Lifehouse

Camperdown, New South Wales, Australia

Calvary Mater Newcastle

Waratah, New South Wales, Australia

Mater Misericordiae Limited

South Brisbane, Queensland, Australia

The Alfred Hospital

Melbourne, Victoria, Australia

Sir Charles Gairdner Hospital

Perth, Western Australia, Australia

Institut Jules Bordet

Anderlecht, Belgium, Belgium

Grand Hôpital de Charleroi - Les Viviers

Gilly, Belgium

AZ Groeninge

Kortrijk, Belgium

UZ Leuven-Campus Gasthuisberg

Leuven, Belgium

AZ Delta

Roeselare, Belgium

CHU Strasbourg - Nouvel Hôpital Civil

Strasbourg, Bas Rhin, France

Hopital Nord - CHU Marseille

Marseille, Bouches-du-Rhône, France

Institut régional du Cancer de Montpellier

Montpellier, Herault, France

CHU Rennes Hôpital Pontchaillou

Rennes, Ille et Vilaine, France

CHU de Grenoble - Hôpital Albert Michallon

La Tronche, Isere, France

CHU Nantes - Hôpital Guillaume et René Laënnec

Saint-Herblain, Loire Atlantique, France

Institut de Cancerologie de l Ouest

Saint-Herblain, Loire Atlantique, France

Centre Leon Berard

Léon, Lyon, France

Hopital Albert Calmette - CHU Lille

Lille, Nord, France

Hôpital Bichat - Claude Bernard

Paris, Paris, France

Hopital Louis Pradel

Bron, Rhone, France

Centre Hospitalier Intercommunal de Créteil

Créteil, Val de Marne, France

Institut Gustave Roussy

Vaillant, Villejuif, France

CHU Brest - Hôpital Morvan

Brest, France

Institut Bergonie

Gironde, France

CHU de Toulouse - Hopital Larrey

Toulouse, France

LKI Lungenfachklinik Immenhausen

Immenhausen, Hesse, Germany

Universitaetsklinikum Essen

Essen, North Rhine-Westphalia, Germany

Universitaetsklinikum Carl Gustav Carus TU Dresden

Dresden, Saxony, Germany

Thoraxklinik Heidelberg gGmbH

Baden, Wuerttemberg, Germany

Klinikum Esslingen GmbH

Baden, Germany

Evangelische Lungenklinik Berlin

Berlin, Germany

Hong Kong United Oncology Centre

Hong Kong, Hong Kong

Queen Mary Hospital

Hong Kong, Hong Kong

Mater Private Hospital

Dublin, Dublin, Ireland

University Hospital Limerick

Cork, Limerick, Ireland

Beaumont Hospital Cancer Clinical

Dublin, Ireland

IEO Istituto Europeo di Oncologia

Milan, Milano, Italy

Azienda Socio Sanitaria Territoriale Niguarda

Milan, Milano, Italy

Istituto Clinico Humanitas

Rossano, Milano, Italy

Fondazione IRCCS San Gerardo dei Tintori

Monza, Milan, Italy

Istituto Nazionale Tumori Fondazione G. Pascale

Napoli, Napoli, Italy

Azienda Ospedaliero Universitaria Pisana (Presidio di Cisanello)

Pisa, Pisa, Italy

Istituto Nazionale dei Tumori Regina Elena IRCCS

Roma, Roma, Italy

Fondazione Policlinico Universitario Agostino Gemelli IRCCS

Rome, Italy

Aichi Cancer Center Hospital

Nagoya, Aichi-ken, Japan

Fujita Health University Hospital

Toyoake-shi, Aichi-ken, Japan

National Cancer Center Hospital East

Kashiwa-shi, Chiba, Japan

NHO Shikoku Cancer Center

Matsuyama, Ehime, Japan

National Hospital Organization Hokkaido Cancer Center

Sapporo, Hokkaido, Japan

Hyogo Cancer Center

Akashi, Hyōgo, Japan

Kanazawa University Hospital

Kanazawa, Ishikawa-ken, Japan

Kanagawa Cancer Center

Yokohama, Kanagawa, Japan

Tohoku University Hospital

Sendai, Miyagi, Japan

Nara Medical University Hospital

Kashihara-shi, Nara, Japan

Niigata Cancer Center

Niigata, Niigata, Japan

Kansai Medical University Hospital

Hirakata-shi, Osaka, Japan

Kindai University Hospital

Osakasayama-shi, Osaka, Japan

Shizuoka Cancer Center

Nagaizumi-chō, Shizuoka, Japan

National Cancer Center Hospital

Chuo Ku, Tokyo, Japan

Cancer Institute Hospital of JFCR

Koto-Ku, Tokyo, Japan

Wakayama Medical University Hospital

Wakayama, Wakayama, Japan

Amsterdam UMC, Locatie VUMC

Amsterdam, Netherlands, Netherlands

Erasmus Medisch Centrum

Rotterdam, Netherlands, Netherlands

Antoni van Leeuwenhoek

Amsterdam, Netherlands

Maastricht University Medical Center P. Debyelaan 25

Maastricht, Netherlands

Radboudumc

Nijmegen, Netherlands

Auckland City Hospital - Cancer and Blood Research

Grafton, Auckland, New Zealand

INSTYTUT GENETYKI I IMMMUNOLOGII GENIM sp. z o.o.

Lublin, Poland

Med-Polonia Sp. z o.o.

Poznan, Poland

Aidport Sp. z o.o.

Skorzewo, Poland

Pan American Center for Oncology Trials

San Juan, Puerto Rico, Puerto Rico

National University Hospital

Singapore, Singapore, Singapore

National Cancer Centre Singapore

Singapore, Singapore

Ajou University Hospital

Gyeonggi-do, Suwon-si, South Korea

Chungbuk National University Hospital

Cheongju-si, South Korea

Chonnam National University Hwasun Hospital

Hwasun, South Korea

Korea University Anam Hospital

Seoul, South Korea

Severance Hospital, Yonsei University Health System

Seoul, South Korea

Samsung Medical Center

Seoul, South Korea

Complejo Hospitalario Universitario A Coruña

A Coruña, A Coruña, Spain

Hospital Universitari Dexeus

Barcelona, Barcelona, Spain

Hospital Universitario La Paz

Fuencarral-El Pardo, Madrid, Spain

Hospital Universitario HM Madrid Sanchinarro

Madrid, Madrid, Spain

Hospital de la Santa Creu i Sant Pau

Barcelona, Spain

Universitätsspital Basel

Basel, Switzerland

HFR Fribourg/Kantonsspital Fribourg

Fribourg, Switzerland

Kantonsspital St. Gallen

Sankt Gallen, Switzerland

Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung, Taiwan, Taiwan

National Cheng Kung University Hospital

Tainan, Taiwan, Taiwan

National Taiwan University Hospital

Taipei, Taiwan, Taiwan

Taipei Medical University Hospital

Taipei, Taiwan

Chang Gung Medical Foundation Linkou

Taoyuan District, Taiwan

The Christie NHS Foundation Trust

Manchester, United Kingdom

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