RecruitingPhase 1Phase 2NCT07038343

AVENTINE-1: Study of AVZO-1418 as a Single Agent and in Combination Therapy in Patients With Locally Advanced or Metastatic Solid Tumors (AVZO-1418-1001)

A Phase 1/2, First-in-human Study to Assess the Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Antitumor Activity of AVZO-1418 as a Single Agent and in Combination Therapy in Patients With Locally Advanced or Metastatic Solid Tumors


Sponsor

Avenzo Therapeutics, Inc.

Enrollment

430 participants

Start Date

Jun 4, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This study, the first clinical trial of AVZO-1418, aims to determine the safety, tolerability, pharmacokinetics, pharmacodynamics, maximum tolerated dose, and antitumor activity of AVZO-1418 when administered intravenously as a monotherapy and potentially in combination therapy to patients with locally advanced or metastatic epithelial solid tumors.


Eligibility

Min Age: 18 YearsMax Age: 75 Years

Inclusion Criteria5

  • Patient must be an adult, between 18 and 75 years of age with an Eastern Cooperative Oncology Group (ECOG) Performance Status of ≤ 1 and a life expectancy of \> 3 months.
  • Patients with histologically or cytologically confirmed locally advanced/metastatic malignancies for tumor types of preferred indications:
  • o Locally advanced or metastatic epithelial solid tumors (as specified in the protocol).
  • Measurable disease as assessed by Investigator using RECIST v1.1.
  • Agree to provide molecular test report results to confirm eligibility and archival tumor samples and/or fresh biopsy, as applicable.

Exclusion Criteria6

  • Uncontrolled hypertension.
  • Patients with active central nervous system (CNS) metastases are not eligible. Patients with asymptomatic and treated brain metastases may participate if they are radiologically stable for at least 4 weeks prior to the first dose of this study and do not require steroid treatment. Patients with suspected or confirmed leptomeningeal disease are not eligible, even if treated.
  • History of drug-induced interstitial lung disease (ILD).
  • History of any serious cardiovascular condition.
  • Infection requiring IV antibiotics, antivirals, or antifungals within 2 weeks prior to first dose.
  • History of a solid organ transplant.

Interventions

DRUGAVZO-1418

Specific dose in protocol specified schedule

DRUGCombination Agent 1

Per label based on combination agent used

DRUGCombination Agent 2

Per label based on combination agent used


Locations(16)

Avenzo Therapeutics Recruiting Site

Gilbert, Arizona, United States

Avenzo Therapeutics Recruiting Site

Los Angeles, California, United States

Avenzo Therapeutics Recruiting Site

Denver, Colorado, United States

Avenzo Therapeutics Recruiting Site

New Haven, Connecticut, United States

Avenzo Therapeutics Recruiting Site

Washington D.C., District of Columbia, United States

Avenzo Therapeutics Recruiting Site

Orlando, Florida, United States

Avenzo Therapeutics Recruiting Site

Sarasota, Florida, United States

Avenzo Therapeutics Recruiting Site

Atlanta, Georgia, United States

Avenzo Therapeutics Recruiting Site

Boston, Massachusetts, United States

Avenzo Therapeutics Recruiting Site

Philadelphia, Pennsylvania, United States

Avenzo Therapeutics Recruiting Site

Dallas, Texas, United States

Avenzo Therapeutics Recruiting Site

Houston, Texas, United States

Avenzo Therapeutics Recruiting Site

San Antonio, Texas, United States

Avenzo Therapeutics Recruiting Site

West Valley City, Utah, United States

Avenzo Therapeutics Recruiting Site

Fairfax, Virginia, United States

Avenzo Therapeutics Recruiting Site

Seattle, Washington, United States

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NCT07038343


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