RecruitingPhase 1NCT07069725

The Phase 1, Open-label, PET Trial Designed to Investigate the Effect of AZD2389 on FAP Occupancy in the Liver in Participants With Advanced Liver Fibrosis.

A Phase 1, Open-label Positron Emission Tomography Trial to Assess Changes in Liver Uptake of [68Ga]Ga-FAPI-46 Following Oral Administration of Single Doses of AZD2389 to Patients With Advanced Liver Fibrosis (PECHORA).


Sponsor

AstraZeneca

Enrollment

12 participants

Start Date

May 26, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

This is a phase 1, open-label, PET trial. The study is designed to investigate the effect of AZD2389 on FAP occupancy in the liver in participants with advanced liver fibrosis.


Eligibility

Min Age: 20 Years

Inclusion Criteria4

  • Male or female (of non-childbearing potential) participant aged ≥ 20 years and willing and able to give written informed consent for participation in the trial.
  • History confirming compensated liver cirrhosis.
  • Females must have a negative pregnancy test.
  • Barrier contraceptives use by males.

Exclusion Criteria10

  • A condition that would interfere with evaluation of the trial intervention, put the participant at risk, influence the participant's ability to participate or affect the interpretation of the results of the trial.
  • Any clinically significant illness, medical or major surgical procedure or trauma prior randomization.
  • Hepatitis B , hepatitis C and/or HIV infection.
  • Significant elevations in liver blood test, MELD score \>12 and platelets \<100 x109/L g).
  • eGFR) \< 60 ml/min/1.73m2.
  • History of decompensated liver cirrhosis.
  • Any participants with an aetiology of liver cirrhosis where the Investigator considers that PET signal uptake may be impacted.
  • History of bleeding disorders and major bleeding risk.
  • History of severe dermatological disorders or wound healing.
  • Positive screening result for drugs of abuse or alcohol.

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Interventions

DRUGAZD2389

Doses of AZD2389 will be administrated orally

DIAGNOSTIC_TESTPET scan and radioligand

PET scan and radioligand


Locations(2)

Research Site

Solna, Sweden

Research Site

Stockholm, Sweden

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NCT07069725


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