RecruitingPhase 1NCT07164313

A Study of ZW251 in Participants With Advanced Solid Tumors

A First-In-Human, Phase 1, Open-Label, Multicenter Study of ZW251, a Novel Glypican-3 Targeting Antibody-Drug Conjugate, in Participants With Advanced Solid Tumors, Including Hepatocellular Carcinoma


Sponsor

Zymeworks BC Inc.

Enrollment

100 participants

Start Date

Oct 21, 2025

Study Type

INTERVENTIONAL

Conditions

Summary

The purpose of this study is to find out if ZW251, an antibody-drug conjugate targeting glypican-3 (GPC3), is safe and can treat participants with advanced cancers, including hepatocellular carcinoma (HCC).


Eligibility

Min Age: 18 Years

Inclusion Criteria5

  • Pathologically or cytologically confirmed diagnosis of HCC with evidence of locally advanced (unresectable, and ineligible for transplant) and/or metastatic disease. Noninvasive methods may be used to confirm diagnosis
  • Measurable disease per RECIST v1.1
  • Eastern Cooperative Oncology Group (ECOG) Performance Status score of 0 or 1
  • Liver function status of Child-Pugh Class A
  • Adequate organ function

Exclusion Criteria5

  • Known additional malignancy that is progressing or that has required active treatment within the last year
  • History of hepatic encephalopathy within the past 6 months or requirement for medications to control encephalopathy
  • Portal vein thrombosis within 3 months prior to Cycle 1 Day 1 that require coagulation therapy or is not stable
  • Known gastrointestinal bleeding within 3 months
  • Acute or chronic uncontrolled renal disease, pancreatitis, or non-malignant liver disease

Interventions

DRUGZW251

Administered intravenously


Locations(20)

UCSF Comprehensive Cancer Center

San Francisco, California, United States

Norton Cancer Institute

Louisville, Kentucky, United States

START Midwest

Grand Rapids, Michigan, United States

Hackensack University Medical Center

Hackensack, New Jersey, United States

MD Anderson Cancer Center

Houston, Texas, United States

START San Antonio

San Antonio, Texas, United States

START - Dublin Mater Misericordiae University Hospital (MMUH)

Dublin, Ireland

National Cancer Center East

Kashiwa, Japan

Kyoto University Hospital

Kyoto, Japan

Kansai Medical University Hospital

Osaka, Japan

National Cancer Center Hospital

Tokyo, Japan

START Lisboa a - Unidade de Ensaios ClÃnicos - Hospital de Santa Maria

Lisbon, Portugal

Hospital Universitario Vall d'Hebron

Barcelona, Spain

START Barcelona

Barcelona, Spain

START - Rioja Hospital Universitario San Pedro

Logroño, Spain

START Madrid Hospital Universitario Fundacion Jimenez Diaz

Madrid, Spain

START Madrid Hospital Universitario HM Sanchinarro - CIOCC

Madrid, Spain

NEXT Oncology Madrid

Madrid, Spain

National Taiwan University Hospital

Taipei, Taiwan

Taipei Veterans General Hospital

Taipei, Taiwan

View Full Details on ClinicalTrials.gov

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NCT07164313


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