RecruitingPhase 2NCT07623616

A Phase 2 Clinical Study of Ziftomenib in Patients With Relapsed or Refractory NPM1-Mutated Acute Myeloid Leukemia

A Phase 2, Multicenter, Open-Label Study of Ziftomenib Monotherapy in Japanese Patients With Relapsed or Refractory Acute Myeloid Leukemia With NPM1 Mutation


Sponsor

Kyowa Kirin Co., Ltd.

Enrollment

6 participants

Start Date

Apr 23, 2026

Study Type

INTERVENTIONAL

Conditions

Summary

This is the first study to administer ziftomenib to Japanese patients. In this study, the efficacy, safety, and pharmacokinetics of ziftomenib will be evaluated in patients with relapsed or refractory NPM1-mutated acute myeloid leukemia


Eligibility

Min Age: 18 Years

Inclusion Criteria10

  • Voluntary written informed consent and willingness to comply with all study procedures
  • Age ≥ 18 years
  • Confirmed diagnosis of acute myeloid leukemia (AML)
  • Patients with R/R AML with NPM1-m
  • No available standard of care expected to provide clinical benefit, ineligible for or declined standard therapy.
  • ECOG performance status 0-2.
  • White blood cell count ≤ 30,000/mm³ at screening (hydroxyurea permitted for cytoreduction).
  • Adequate organ function according to protocol requirements.
  • Women of childbearing potential must be willing to use a highly effective method of contraception throughout the study and for at least 187 days after the last dose of study treatment.
  • Males with female partners of childbearing potential must agree to use a highly effective method of contraception throughout the study and for at least 97 days after the last dose of study treatment.

Exclusion Criteria16

  • Diagnosis of acute promyelocytic leukemia.
  • Donor lymphocyte infusion < 30 days prior to study entry.
  • Clinically active central nervous system (CNS) leukemia.
  • Prior hematopoietic stem cell transplantation (HSCT) without adequate hematologic recovery.
  • Active Grade ≥ 2 acute graft-versus-host disease or moderate/severe chronic graft-versus-host disease.
  • Prior treatment with a menin inhibitor.
  • Receipt of chemotherapy, immunotherapy, radiotherapy, or investigational therapy within 14 days or 5 half-lives prior to first dose.
  • Unresolved toxicities from prior therapy > Grade 1.
  • Requirement for strong CYP3A4 inducers.
  • Active or uncontrolled infection, including hepatitis B, hepatitis C, or HIV.
  • Conditions predisposing to serious or life-threatening infection or significant immunodeficiency.
  • Cardiovascular disease or QTcF > 480 ms.
  • Interstitial lung disease.
  • Major surgery within 4 weeks prior to first dose.
  • Women who are pregnant or lactating
  • Any medical, psychiatric, or social condition that may interfere with study participation or safety, or that makes the patient unsuitable in the investigator's judgment.

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Interventions

DRUGziftomenib

Oral adminitration once daily


Locations(20)

Chiba Aoba Municipal Hospital

Chiba, Japan

Gifu Municipal Hospital

Gifu, Japan

Hyogo Medical University Hospital

Hyōgo, Japan

Mito Medical Center

Ibaraki, Japan

Imamura General Hospital

Kagoshima, Japan

Kanagawa Cancer Center

Kanagawa, Japan

Kyoto University Hospital

Kyoto, Japan

Tohoku University Hospital

Miyagi, Japan

Matsumoto National Hospital

Nagano, Japan

Nagasaki University Hospital

Nagasaki, Japan

Kurashiki Central Hospital

Okayama, Japan

Okayama University Hospital

Okayama, Japan

Kansai Medical University Hospital

Osaka, Japan

Osaka Metropolitan University Hospital

Osaka, Japan

Jichi Medical University Saitama Medical Center

Saitama, Japan

Dokkyo Medical University Hospital

Tochigi, Japan

Jichi Medical University Hospital

Tochigi, Japan

Keio University Hospital

Tokyo, Japan

Nippon Medical School Hospital

Tokyo, Japan

Tokyo Metropolitan Cancer and Infectious Diseases Center Komagome Hospital

Tokyo, Japan

View Full Details on ClinicalTrials.gov

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NCT07623616


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