RecruitingPhase 3NCT05646862

A Study Evaluating the Efficacy and Safety of Inavolisib Plus Fulvestrant Compared With Alpelisib Plus Fulvestrant in Participants With HR-Positive, HER2-Negative, PIK3CA Mutated, Locally Advanced or Metastatic Breast Cancer Post CDK4/6i and Endocrine Combination Therapy

A Phase III, Multicenter, Randomized, Open-Label Study Evaluating the Efficacy and Safety of Inavolisib Plus Fulvestrant Versus Alpelisib Plus Fulvestrant in Patients With Hormone Receptor-Positive, HER2-Negative, PIK3CA Mutated, Locally Advanced or Metastatic Breast Cancer Who Progressed During or After CDK4/6 Inhibitor and Endocrine Combination Therapy


Sponsor

Hoffmann-La Roche

Enrollment

420 participants

Start Date

Jun 7, 2023

Study Type

INTERVENTIONAL

Conditions

Summary

This is a Phase III, multicenter, randomized, open-label, global study designed to evaluate the efficacy and safety of inavolisib plus fulvestrant compared with alpelisib plus fulvestrant in patients with hormone receptor (HR)-positive, human epidermal growth factor receptor 2 (HER2) -negative, PIK3CA-mutated, locally advanced (LA) or metastatic breast cancer (mBC), who progressed during or after cyclin dependent kinase 4/6i (CDK4/6i)-based therapy. Enrollment for the main study is now complete.


Eligibility

Min Age: 18 Years

Plain Language Summary

Simplified for easier understanding

This clinical trial is studying a drug called Alpelisib, a drug called Bupropion, and others for people with breast cancer. The study is currently recruiting participants at 210 locations.

This summary was AI-generated to explain the trial in plain language. It is not medical advice. Always discuss eligibility with your doctor before enrolling in a clinical trial.

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Interventions

DRUGInavolisib

Participants will be administered a 9 milligram (mg) inavolisib tablet orally once a day (PO QD) on Days 1-28 of each 28-day cycle of main study and sub-study.

DRUGFulvestrant

Participants will be administered 500 mg of fulvestrant on Days 1 and 15 of Cycle 1 and then on Day 1 of each subsequent 28-day cycle of main study and sub-study.

DRUGAlpelisib

Alpelisib will be administered to participants at the approved dose in combination with fulvestrant: 300 mg taken PO QD and on days 1-28 of each 28-day cycle.

DRUGBupropion

Participants will be administered bupropion PO on Day -3 and Day 12 of Cycle 1 of the sub-study.

DRUGOmeprazole

Participants will be administered omerprazole PO on Day -4 and Day 11 of Cycle 1 of sub-study.

DRUGMidazolam

Participants will be administered midazolam PO on Day -4 and Day 11 of Cycle 1 of sub-study.


Locations(210)

Marin Cancer Care Inc

Greenbrae, California, United States

Cancer Blood and Specialty Clinic

Los Alamitos, California, United States

Los Angeles Cancer Network

Los Angeles, California, United States

University of California, Irvine Medical Center

Orange, California, United States

UC Davis Comprehensive Cancer Center

Sacramento, California, United States

Rocky Mountain Cancer Centers

Denver, Colorado, United States

Banner MD Anderson Cancer Center

Greeley, Colorado, United States

Eastern CT Hematology and Oncology Associates

Norwich, Connecticut, United States

Cancer Care Centers of Brevard

Palm Bay, Florida, United States

Cleveland Clinic Florida

Weston, Florida, United States

Grady Health System

Atlanta, Georgia, United States

Midtown West Medical

Atlanta, Georgia, United States

Emory University Hospital

Atlanta, Georgia, United States

Winship Cancer Institute at Emory Saint Joseph's Hospital

Atlanta, Georgia, United States

University of Louisville Hospital

Louisville, Kentucky, United States

Massachusetts General Hospital

Boston, Massachusetts, United States

Karmanos Cancer Institute.

Detroit, Michigan, United States

Cancer & Hematology Centers of Western Michigan

Grand Rapids, Michigan, United States

Minnesota Oncology Hematology

Saint Paul, Minnesota, United States

MD Anderson Cancer Center at Cooper

Camden, New Jersey, United States

Novant Health Presbyterain Medical Center

Charlotte, North Carolina, United States

Novant Health Forsyth Medical Center

Winston-Salem, North Carolina, United States

Gabrail Cancer Center

Canton, Ohio, United States

Asante Rogue Regional Medical Center

Medford, Oregon, United States

Bryn Mawr Hospital

Bryn Mawr, Pennsylvania, United States

St. Lukes Hospital and Health Network

Easton, Pennsylvania, United States

Paoli Memorial Hospital

Paoli, Pennsylvania, United States

Abramson Cancer Center Chester County Hospital

West Chester, Pennsylvania, United States

Lankenau Medical Center, Cancer Center

Wynnewood, Pennsylvania, United States

Main Line Health System

Wynnewood, Pennsylvania, United States

WellSpan Oncology Research

York, Pennsylvania, United States

Texas Oncology West

Amarillo, Texas, United States

Texas Oncology - Dallas Presbyterian Hospital

Dallas, Texas, United States

Texas Tech University Health Sciences Center

El Paso, Texas, United States

Texas Oncology (Flower Mound) - USOR

Flower Mound, Texas, United States

The Center for Cancer and Blood Disorders - Fort Worth

Fort Worth, Texas, United States

Lumi Research

Kingwood, Texas, United States

Texas Oncology McKinney

McKinney, Texas, United States

Kadlec Clinic Hematology and Oncology

Kennewick, Washington, United States

Centro de Investigaciones Médicas y Desarrollo LC S.R.L

Buenos Aires, Argentina

Centro Oncologico Korben

Ciudad Autonoma Buenos Aires, Argentina

Fundacion CORI para la Investigacion y Prevencion del Cancer

La Rioja, Argentina

Instituto de Oncología de Rosario

Rosario, Argentina

Sanatorio Parque S.A.

Rosario, Argentina

Hosp Provincial D. Centenarios

Rosario, Argentina

CER San Juan Centro Polivalente de Asistencia e Investigacion Clinica

San Juan, Argentina

Clinica Viedma S.A.

Viedma, Argentina

Campbelltown Hospital

Campbelltown, New South Wales, Australia

Coffs Harbour Health Campus

Coffs Harbour, New South Wales, Australia

Concord Repatriation General Hospital

Concord, New South Wales, Australia

Kinghorn Cancer Centre

Darlinghurst, New South Wales, Australia

Gosford Hospital

Gosford, New South Wales, Australia

Icon Cancer Care Wesley

Auchenflower, Queensland, Australia

University of the Sunshine Coast

Sippy Downs, Queensland, Australia

Bendigo Cancer Centre

Bendigo, Victoria, Australia

Sir Charles Gairdner Hospital

Perth, Western Australia, Australia

Cliniques Universitaires St-Luc

Brussels, Belgium

GHdC Site Les Viviers

Charleroi, Belgium

UZ Antwerpen

Edegem, Belgium

UZ Gent

Ghent, Belgium

UZ Leuven Gasthuisberg

Leuven, Belgium

Clinique Ste-Elisabeth

Namur, Belgium

Hospital da Bahia

Salvador, Estado de Bahia, Brazil

Instituto D?Or de Pesquisa e Ensino ? Hospital DF STAR

Brasília, Federal District, Brazil

NUPEC

Belo Horizonte, Minas Gerais, Brazil

Hospital Santa Cruz / Centro de Oncologia D'Or

Curitiba, Paraná, Brazil

Hospital do Cancer de Pernambuco - HCP

Recife, Pernambuco, Brazil

Instituto D?Or de Pesquisa e Ensino ? Hospital Esperança Recife

Recife, Pernambuco, Brazil

Vencer Oncoclínica - Centro de Pesquisa do Piauí

Teresina, Piauí, Brazil

Liga Norte Riograndense Contra O Câncer

Natal, Rio Grande do Norte, Brazil

Santa Casa de Misericordia de Porto Alegre

Porto Alegre, Rio Grande do Sul, Brazil

Hospital Sao Lucas - PUCRS

Porto Alegre, Rio Grande do Sul, Brazil

Hospital de Base de Sao Jose do Rio Preto

São José do Rio Preto, São Paulo, Brazil

Hospital Sírio-Libanês

São Paulo, São Paulo, Brazil

Arthur J.E. Child Comprehensive Cancer Center-Calgary

Calgary, Alberta, Canada

Cross Cancer Institute

Edmonton, Alberta, Canada

BC Cancer ? Vancouver

Vancouver, British Columbia, Canada

The Moncton Hospital

Moncton, New Brunswick, Canada

Juravinski Hospital

Hamilton, Ontario, Canada

The Ottawa Hospital - General Campus

Ottawa, Ontario, Canada

CIUSSS de l Est de l Ile de Montreal - Hopital Maisonneuve Rosemont

Montreal, Quebec, Canada

Centre Hospitalier de l'Universite de Montreal (CHUM)

Montreal, Quebec, Canada

Jewish General Hospital

Montreal, Quebec, Canada

Hôpital du Sacré-Coeur de Montreal

Montreal, Quebec, Canada

The First Hospital of Jilin University

Changchun, China

Sichuan Provincial Cancer Hospital

Chengdu, China

The First Affiliated Hospital, Chongqing Medical University

Chongqing, China

Sun yat-sen University Cancer Center

Guangzhou, China

Guangdong Provincial People's Hospital

Guangzhou, China

The Second Affiliated Hospital of Zhejiang University School of Medicine

Hangzhou, China

Sir Run Run Shaw Hospital Zhejiang University

Hangzhou, China

Harbin Medical University Tumor Hospital

Harbin, China

Shandong Cancer Hospital

Jinan, China

The Second Affiliated Hospital to Nanchang University

Nanchang, China

Jiangsu Cancer Hospital

Nanjing, China

Tianjin Cancer Hospital

Tianjin, China

Union Hospital Tongji Medical College Huazhong University of Science and Technology

Wuhan, China

Hubei Cancer Hospital

Wuhan, China

First Affiliated Hospital of Medical College of Xi'an Jiaotong University

Xi'an, China

Zhejiang Cancer Hospital

Zhejiang, China

Institut Sainte Catherine

Avignon, France

Centre Hospitalier de La Cote Basque

Bayonne, France

Polyclinique Bordeaux Nord

Bordeaux, France

Centre Leon Berard

Lyon, France

ICM

Montpellier, France

Centre Eugene Marquis

Rennes, France

IUCT Oncopole

Toulouse, France

Uniklinik RWTH Aachen Klinik für Gynäkologie und Geburtsmedizin

Aachen, Germany

Onkologische Schwerpunktpraxis Bielefeld

Bielefeld, Germany

Universitätsklinikum Essen

Essen, Germany

Praxis für Interdisziplinäre Onkologie und Hämatologie GbR

Freiburg im Breisgau, Germany

Niels-Stensen-Kliniken Franziskus-Hospital Harderberg GmbH

Georgsmarienhütte, Germany

Universitätsmedizin Göttingen Georg-August-Universität

Göttingen, Germany

Mammazentrum Hamburg am Krankenhaus Jerusalem

Hamburg, Germany

Medizinische Hochschule Zentrum Frauenheilkunde Abt.Gynäkologische Onkologie

Hanover, Germany

Nationales Centrum für Tumorerkrankungen (NCT)

Heidelberg, Germany

Brustzentrum Rhein-Ruhr Servicegesellschaft mbH

Mönchengladbach, Germany

Klinik & Poliklinik für Frauenheilkunde und Geburtshilfe, Campus Innenstadt

München, Germany

St. Vincenz-Krankenhaus GmbH Paderborn Frauen- und Kinderklinik St. Louise

Paderborn, Germany

MVZ für Hämatologie und Onkologie Ravensburg GmBH

Ravensburg, Germany

A.O. S. Anna e San Sebastiano

Caserta, Campania, Italy

IRST Istituto Scientifico Romagnolo Per Lo Studio E Cura Dei Tumori, Sede Meldola

Meldola, Emilia-Romagna, Italy

AUSL della Romagna

Ravenna, Emilia-Romagna, Italy

Irccs Centro Di Riferimento Oncologico (CRO)

Aviano, Friuli Venezia Giulia, Italy

Ospedale San Raffaele

Milan, Lombardy, Italy

ASL AL - Azienda Sanitaria Locale AL

Alessandria, Piedmont, Italy

AOU Città della Salute e della Scienza di Torino

Turin, Piedmont, Italy

Humanitas Centro Catanese Di Oncologia

Misterbianco (CT), Sicily, Italy

Ospedale Di Macerata

Province of Macerata, The Marches, Italy

Ospedale Santa Chiara

Trento, Trentino-Alto Adige, Italy

Ospedale S. Giuseppe

Empoli (FI), Tuscany, Italy

Panamerican Clinical Research S.A de C.V.

Guadalajara, Jalisco, Mexico

RENATI INNOVATION S.A.P.I. de C.V

Guadalajara, Jalisco, Mexico

COI Centro Oncologico Internacional Santa Fe

Mexico City, Mexico CITY (federal District), Mexico

Health Pharma Professional Research

Mexico City, Mexico CITY (federal District), Mexico

OncoMed

Mexico City, Mexico CITY (federal District), Mexico

ARKE Estudios Clínicos S.A. de C.V.

Mexico City, Mexico CITY (federal District), Mexico

Instituto Nacional de Cancerologia

Distrito Federal, Mexico

CENEIT Oncologicos

Mexico City, Mexico

Antiguo Hospital Civil de Guadalajara Fray Antonio Alcalde

Morelia, Mexico

New Zealand Clinical Research - Auckland

Auckland, New Zealand

Centrum Onkologii im. Prof. Franciszka ?ukaszczyka

Bydgoszcz, Poland

Szpital Morski im.PCK

Gdynia, Poland

Narodowy Instytut Onkologii Odzia? w Gliwicach

Gliwice, Poland

Przychodnia Lekarska KOMED, Roman Karaszewski

Konin, Poland

Szpital Wojewódzki im. Miko?aja Kopernika

Koszalin, Poland

Szpital Uniwersytecki w Krakowie

Krakow, Poland

MRUKMED Lekarz Beata Madej-Mruk i Partner Spolka Partnerska Oddzial nr 1 w Rzeszowie

Rzeszów, Poland

Narodowy Instytut Onkologii im. M.Sklodowskiej-Curie

Warsaw, Poland

Dr. W.M. Szpak Incorporated trading as Rainbow Oncology

Durban, South Africa

Hopelands Cancer Centre

Hilton, South Africa

Medical Oncology Centre of Rosebank

Johannesburg, South Africa

Richards Bay Oncology Centre

KwaZulu Natal, South Africa

Mountain View Oncology

Paarl, South Africa

Kyungpook National University Chilgok Hospital

Daegu, South Korea

National Cancer Center

Goyang-si, South Korea

CHA Bundang Medical Center

Gyeonggi-do, South Korea

Catholic Univ. of Incheon St.Mary's Hospital

Incheon, South Korea

Inha University Hospital

Incheon, South Korea

Korea University Anam Hospital

Seoul, South Korea

Seoul National University Hospital

Seoul, South Korea

Severance Hospital, Yonsei University Health System

Seoul, South Korea

Asan Medical Center

Seoul, South Korea

Gangnam Severance Hospital

Seoul, South Korea

Samsung Medical Center

Seoul, South Korea

Seoul St Mary's Hospital

Seoul, South Korea

ICO L'Hospitalet

L'Hospitalet de Llobregat, Barcelona, Spain

Complejo Hospitalario Universitario de Santiago (CHUS)

Santiago de Compostela, LA Coruna, Spain

Hospital Universitario de Canarias

San Cristóbal de La Laguna, Tenerife, Spain

Hospital Universitari Vall d'Hebron

Barcelona, Spain

Hospital San Pedro De Alcantara

Cáceres, Spain

Hospital General Universitario Gregorio Marañon

Madrid, Spain

Hospital Ramon y Cajal

Madrid, Spain

Hospital Universitario 12 de Octubre

Madrid, Spain

Hospital Regional Universitario Carlos Haya

Málaga, Spain

Hospital Universitario Virgen de Arrixaca

Murcia, Spain

Hospital Universitario Virgen Macarena

Seville, Spain

China Medical University Hospital

Taichung, Taiwan

National Cheng Kung University Hospital

Tainan, Taiwan

Taipei Veterans General Hospital

Taipei, Taiwan

Chang Gung Memorial Hosipital at Linkou

Taoyuan City, Taiwan

Veterans General Hospital - Taichung

Xitun Dist., Taiwan

National Taiwan University Hospital

Zhongzheng Dist., Taiwan

Chulalongkorn Hospital

Bangkok, Thailand

Maharaj Nakorn Chiang Mai Hospital

Chiang Mai, Thailand

Chulabhorn Hospital

Lak Si, Thailand

Songklanagarind Hospital

Songkhla, Thailand

Gulhane Training and Applicaton Hospital

Ankara, Turkey (Türkiye)

Memorial Ankara Hastanesi

Ankara, Turkey (Türkiye)

Dicle University Faculty of Medicine

Diyarbakır, Turkey (Türkiye)

Trakya University Medical Faculty

Edirne, Turkey (Türkiye)

Medipol Mega Üniversite Hastanesi Göztepe

Istanbul, Turkey (Türkiye)

Marmara Uni Faculty of Medicine

Istanbul, Turkey (Türkiye)

Ege Uni Medical Faculty Hospital

Izmir, Turkey (Türkiye)

Izmir Ataturk Training and Research Hospital

Izmir, Turkey (Türkiye)

Goztepe Prof.Dr. Suleyman Yalcin City Hospital

Kadiköy, Turkey (Türkiye)

Medical Park Seyhan Hospital

Seyhan, Turkey (Türkiye)

Hacettepe Uni Medical Faculty Hospital

Sihhiye/Ankara, Turkey (Türkiye)

Basingstoke and North Hampshire Hospital

Basingstoke, United Kingdom

Blackpool Victoria Hospital

Blackpool, United Kingdom

Dumfries and Galloway Royal Infirmary

Dumfries, United Kingdom

Western General Hospital

Edinburgh, United Kingdom

Princess Alexandra Hospital

Harlow, United Kingdom

St John's Hospital

Livingston, United Kingdom

St Bartholomew's Hospital

London, United Kingdom

Maidstone & Tonbridge Wells Hospital

Maidstone, United Kingdom

Mount Vernon & Watford Hospital Trust

Northwood, United Kingdom

Churchill Hospital

Oxford, United Kingdom

Royal Preston Hosptial

Preston, United Kingdom

Royal Hampshire County Hospital

Winchester, United Kingdom

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NCT05646862


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